Foto del docente

Manuela Bartolini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Gandini, Annachiara; Bartolini, Manuela; Tedesco, Daniele; Martinez-Gonzalez, Loreto; Roca, Carlos; Campillo, Nuria E.; Zaldivar-Diez, Josefa; Perez, Concepción; Zuccheri, Giampaolo; Miti, Andrea; Feoli, Alessandra; Castellano, Sabrina; Petralla, Sabrina; Monti, Barbara; Rossi, Martina; Moda, Fabio; Legname, Giuseppe; Martinez, Ana; Bolognesi, Maria Laura*, Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 7640 - 7656 [Scientific article]

Terra, Bruna S.; Da Silva, Pedro H. C.; Tramarin, Anna; Franco, Lucas L.; Da Cunha, Elaine F. F.; Macedo, Fernando; Ramalho, Teodorico C.; Bartolini, Manuela; Bolognesi, Maria L.; De Fátima, Ângelo, Two novel donepezil-lipoic acid hybrids: Synthesis, anticholinesterase and antioxidant activities and theoretical studies, «JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY», 2018, 29, pp. 738 - 747 [Scientific article]

A De Simone; M Naldi; D Tedesco; M Bartolini; V Andrisano, β-Amyloid-CORMs interaction monitoring by LC-ESI/MS and Circular Dichroism studies, in: Med Chem Sicily 2018, 2018, pp. 18 - 18 (atti di: Med Chem Sicily 2018, Palermo, 17-20 July 2018) [Contribution to conference proceedings]

Wang, Li; Moraleda, Ignacio; Iriepa, Isabel; Romero, Alejandro; López-Muñoz, Francisco; Chioua, Mourad; Inokuchi, Tsutomu; Bartolini, Manuela; Marco-Contelles, José, 5-Methyl-N-(8-(5,6,7,8-tetrahydroacridin-9-ylamino)octyl)-5 H -indolo[2,3- b] quinolin-11-amine: a highly potent human cholinesterase inhibitor, «MEDCHEMCOMM», 2017, 8, pp. 1307 - 1317 [Scientific article]

Anna Tramarin, Edoardo Fabini, Manuela Bartolini, AChE inhibitors: affinity and kinetic studies using SPR technology, in: Quick Guide, 2017(atti di: Recent Developments in Pharmaceutical Analysis, Rimini, 20-23/09/2017) [Poster]

Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli, Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Chalcone-based carbamates for Alzheimer's disease treatment, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 749 - 764 [Scientific article]

Pérez-Areales, Francisco Javier; Betari, Nibal; Viayna, Antonio; Pont, Caterina; Espargarã³, Alba; Bartolini, Manuela; DE SIMONE, Angela; Rinaldi Alvarenga, José Fernando; Pã©rez, Belã©n; Sabate, Raimon; Lamuela-Raventós, Rosa Maria; Andrisano, Vincenza; Luque, Francisco Javier; Muñoz-Torrero, Diego, Design, synthesis and multitarget biological profiling of second-generation anti-Alzheimer rhein-huprine hybrids, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 965 - 981 [Scientific article]

De Simone, Angela; Bartolini, Manuela; Baschieri, Andrea; Apperley, Kim Y.P.; Chen, Huan Huan; Guardigni, Melissa; Montanari, Serena; Kobrlova, Tereza; Soukup, Ondrej; Valgimigli, Luca; Andrisano, Vincenza; Keillor, Jeffrey W.; Basso, Manuela; Milelli, Andrea, Hydroxy-substituted trans-cinnamoyl derivatives as multifunctional tools in the context of Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 139, pp. 378 - 389 [Scientific article]

Anna Tramarin, Edoardo Fabini, Genny Degani, Marina Naldi, Laura Popolo, Giancarlo Aldini, Manuela Bartolini, Interaction between commercial glycated HSA and the extracellular region of human RAGE: a SPR-based study, in: Quick Guide, 2017(atti di: Recent Developments in Pharmaceutical Analysis, Rimini, 20-23/09/2017) [Poster]

Ruolo editoriale nella rivista «Journal of Pharmaceutical and Biomedical Analysis, volume 144 - Special Issue in Honor of the Retirement of Prof. Carlo Bertucci»

Daniele Tedesco, Piotr Drączkowski, Mirko Zaffagnini, Dariusz Matosiuk, Krzysztof Jóźwiak, Manuela Bartolini, Lipid bilayer nanodiscs: a promising system for in-solution studies on GPCR binding, in: 2° Retreat Scientifico del Dipartimento di Farmacia e Biotecnologie - Università di Bologna, 2017(atti di: 2° Retreat Scientifico del Dipartimento di Farmacia e Biotecnologie - Università di Bologna, Bologna, 07-08/02/2017) [Poster]Open Access

Simoni, Elena; Bartolini, Manuela; Abu, Izuddin F; Blockley, Alix; Gotti, Cecilia; Bottegoni, Giovanni; Caporaso, Roberta; Bergamini, Christian; Andrisano, Vincenza; Cavalli, Andrea; Mellor, Ian R; Minarini, Anna; Rosini, Michela, Multitarget drug design strategy in Alzheimer's disease: focus on cholinergic transmission and amyloid-beta aggregation, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 953 - 963 [Scientific article]

Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Coluccia, Antonio; Di Santo, Roberto; Costi, Roberta; Andrisano, Vincenza; Alabiso, Francesco; Bergamini, Christian; Fato, Romana; Bartolini, Manuela; Scipione, Luigi, New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 141, pp. 197 - 210 [Scientific article]

Roldán-Peña, Jesús M.; Alejandre-Ramos, Daniel; López, O scar; Maya, Inés; Lagunes, Irene; Padrón, José M.; Peña-Altamira, Luis Emiliano; Bartolini, Manuela; Monti, Barbara; Bolognesi, Maria L.; Fernández-Bolaños, José G., New tacrine dimers with antioxidant linkers as dual drugs: Anti-Alzheimer's and antiproliferative agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 138, pp. 761 - 773 [Scientific article]Open Access

Andrisano, Vincenza; Bartolini, Manuela; Tedesco, Daniele; Wainer, Irving W., Preface, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2017, 144, pp. VI - VI [Scientific article]