Foto del docente

Manuela Bartolini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

de simone a, naldi m, tedesco d, bartolini m, andrisano v, A multi-methodological approach for the investigation of β-Amyloid-CORMs interaction: an LC-ESI/MS and Circular Dichroism study., in: 10° MS pharma day book of abstracts, 2018, pp. 15 - 16 (atti di: 10° MS pharma day, Colleretto Giacosa (TO), 24-26 Ottobre) [Contribution to conference proceedings]

Andrisano, Vincenza*; Naldi, Marina; De Simone, Angela; Bartolini, Manuela, A patent review of butyrylcholinesterase inhibitors and reactivators 2010–2017, «EXPERT OPINION ON THERAPEUTIC PATENTS», 2018, 28, pp. 455 - 465 [Scientific article]

Fabini, Edoardo; Tramarin, Anna; Bartolini, Manuela*, Combination of human acetylcholinesterase and serum albumin sensing surfaces as highly informative analytical tool for inhibitor screening, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2018, 155, pp. 177 - 184 [Scientific article]

Anna Tramarin, Marina Naldi, Loredana Lupu, Pascal Wiegand, Edoardo Fabini, Genny Degani, Laura Popolo, Giancarlo Aldini, Michael Przybylski, Manuela Bartolini, EPITOPE IDENTIFICATION OF GLYCATED HSA AND THE EXTRACELLULAR REGION OF HUMAN RAGE BY SPR AND AFFINITY-MS SPECTROMETRY, in: Abstract book, 2018(atti di: XXII International Mass Spectrometry Conference, Florence, 26-31/08/2018) [Poster]

Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease, «MOLECULES», 2018, 23, Article number: 1902 , pp. 1 - 22 [Scientific article]Open Access

Daniele Tedesco, Federica Ierardi, Aleš Štrancar, Urh Černigoj, Manuela Bartolini, Extraction of human serum albumin for functional studies using novel immunoaffinity-based CIMac-αHSA monolithic columns, in: Monolith Summer School and Symposium 2018 (MSS 2018), 2018(atti di: Monolith Summer School and Symposium 2018 (MSS 2018), Portorož (Slovenia), 18-20/06/2018) [Poster]Open Access

Naldi, Marina; Tramarin, Anna; Bartolini, Manuela*, Immobilized enzyme-based analytical tools in the -omics era: recent advances, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2018, 160, pp. 222 - 237 [Scientific article]

Galdeano, Carles; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Bartolini, Manuela; Pérez, Belén; Victòria Clos, M.; Silman, Israel; Jean, Ludovic*; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Munoz-Torrero, Diego, Increasing polarity in tacrine and huprine derivatives: Potent anticholinesterase agents for the treatment of myasthenia gravis, «MOLECULES», 2018, 23, Article number: 634 , pp. 1 - 19 [Scientific article]Open Access

Angela De Simone, Marina Naldi, Daniele Tedesco, Manuela Bartolini, Vincenza Andrisano, Integrated analytical methodologies for Alzheimer's disease drug discovery, in: DA-PBA 2018 book of abstracts, 2018, pp. 148 - 148 (atti di: DA-PBA 2018, Leuven, Belgio, 9-12 Settembre 2018) [Contribution to conference proceedings]

Anna Tramarin, Edoardo Fabini, Marina Naldi, Loredana Lupu, Pascal Wiegand, Genny Degani, Laura Popolo, Giancarlo Aldini, Michael Przybylski, Manuela Bartolini, RAGE IN DIABETES MELLITUS: A MULTIMETHODOLOGICAL STRATEGY TO STUDY GLYCATED HSA-RAGE INTERACTION, in: XVIII GIORNATA DELLA CHIMICA DELL’EMILIA ROMAGNA, 2018(atti di: XVIII GIORNATA DELLA CHIMICA DELL’EMILIA ROMAGNA, Parma, 17/12/2018) [Poster]

m BARTOLINI, a DE SIMONE, V ANDRISANO, Synthesis and pharmacological evaluation of a novel class of multi target Huprine-based anti-Alzheimer hybrids, in: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily 2018 book of abstracts, 2018, pp. 13 - 13 (atti di: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily 2018, palermo, 17-20 July 2018) [Contribution to conference proceedings]

Chioua, Mourad; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tramarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jóźwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José; Bartolini, Manuela*, Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, as multi-target-directed ligands for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2018, 155, pp. 839 - 846 [Scientific article]

Gandini, Annachiara; Bartolini, Manuela; Tedesco, Daniele; Martinez-Gonzalez, Loreto; Roca, Carlos; Campillo, Nuria E.; Zaldivar-Diez, Josefa; Perez, Concepción; Zuccheri, Giampaolo; Miti, Andrea; Feoli, Alessandra; Castellano, Sabrina; Petralla, Sabrina; Monti, Barbara; Rossi, Martina; Moda, Fabio; Legname, Giuseppe; Martinez, Ana; Bolognesi, Maria Laura*, Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 7640 - 7656 [Scientific article]

Terra, Bruna S.; Da Silva, Pedro H. C.; Tramarin, Anna; Franco, Lucas L.; Da Cunha, Elaine F. F.; Macedo, Fernando; Ramalho, Teodorico C.; Bartolini, Manuela; Bolognesi, Maria L.; De Fátima, Ângelo, Two novel donepezil-lipoic acid hybrids: Synthesis, anticholinesterase and antioxidant activities and theoretical studies, «JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY», 2018, 29, pp. 738 - 747 [Scientific article]

A De Simone; M Naldi; D Tedesco; M Bartolini; V Andrisano, β-Amyloid-CORMs interaction monitoring by LC-ESI/MS and Circular Dichroism studies, in: Med Chem Sicily 2018, 2018, pp. 18 - 18 (atti di: Med Chem Sicily 2018, Palermo, 17-20 July 2018) [Contribution to conference proceedings]