Foto del docente

Manuela Bartolini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease, «MOLECULES», 2018, 23, Article number: 1902 , pp. 1 - 22 [Scientific article]Open Access

Daniele Tedesco, Federica Ierardi, Aleš Štrancar, Urh Černigoj, Manuela Bartolini, Extraction of human serum albumin for functional studies using novel immunoaffinity-based CIMac-αHSA monolithic columns, in: Monolith Summer School and Symposium 2018 (MSS 2018), 2018(atti di: Monolith Summer School and Symposium 2018 (MSS 2018), Portorož (Slovenia), 18-20/06/2018) [Poster]Open Access

Naldi, Marina; Tramarin, Anna; Bartolini, Manuela*, Immobilized enzyme-based analytical tools in the -omics era: recent advances, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2018, 160, pp. 222 - 237 [Scientific article]

Galdeano, Carles; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Bartolini, Manuela; Pérez, Belén; Victòria Clos, M.; Silman, Israel; Jean, Ludovic*; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Munoz-Torrero, Diego, Increasing polarity in tacrine and huprine derivatives: Potent anticholinesterase agents for the treatment of myasthenia gravis, «MOLECULES», 2018, 23, Article number: 634 , pp. 1 - 19 [Scientific article]Open Access

Angela De Simone, Marina Naldi, Daniele Tedesco, Manuela Bartolini, Vincenza Andrisano, Integrated analytical methodologies for Alzheimer's disease drug discovery, in: DA-PBA 2018 book of abstracts, 2018, pp. 148 - 148 (atti di: DA-PBA 2018, Leuven, Belgio, 9-12 Settembre 2018) [Contribution to conference proceedings]

Anna Tramarin, Edoardo Fabini, Marina Naldi, Loredana Lupu, Pascal Wiegand, Genny Degani, Laura Popolo, Giancarlo Aldini, Michael Przybylski, Manuela Bartolini, RAGE IN DIABETES MELLITUS: A MULTIMETHODOLOGICAL STRATEGY TO STUDY GLYCATED HSA-RAGE INTERACTION, in: XVIII GIORNATA DELLA CHIMICA DELL’EMILIA ROMAGNA, 2018(atti di: XVIII GIORNATA DELLA CHIMICA DELL’EMILIA ROMAGNA, Parma, 17/12/2018) [Poster]

m BARTOLINI, a DE SIMONE, V ANDRISANO, Synthesis and pharmacological evaluation of a novel class of multi target Huprine-based anti-Alzheimer hybrids, in: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily 2018 book of abstracts, 2018, pp. 13 - 13 (atti di: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily 2018, palermo, 17-20 July 2018) [Contribution to conference proceedings]

Chioua, Mourad; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tramarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jóźwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José; Bartolini, Manuela*, Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, as multi-target-directed ligands for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2018, 155, pp. 839 - 846 [Scientific article]

Gandini, Annachiara; Bartolini, Manuela; Tedesco, Daniele; Martinez-Gonzalez, Loreto; Roca, Carlos; Campillo, Nuria E.; Zaldivar-Diez, Josefa; Perez, Concepción; Zuccheri, Giampaolo; Miti, Andrea; Feoli, Alessandra; Castellano, Sabrina; Petralla, Sabrina; Monti, Barbara; Rossi, Martina; Moda, Fabio; Legname, Giuseppe; Martinez, Ana; Bolognesi, Maria Laura*, Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 7640 - 7656 [Scientific article]

Terra, Bruna S.; Da Silva, Pedro H. C.; Tramarin, Anna; Franco, Lucas L.; Da Cunha, Elaine F. F.; Macedo, Fernando; Ramalho, Teodorico C.; Bartolini, Manuela; Bolognesi, Maria L.; De Fátima, Ângelo, Two novel donepezil-lipoic acid hybrids: Synthesis, anticholinesterase and antioxidant activities and theoretical studies, «JOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY», 2018, 29, pp. 738 - 747 [Scientific article]

A De Simone; M Naldi; D Tedesco; M Bartolini; V Andrisano, β-Amyloid-CORMs interaction monitoring by LC-ESI/MS and Circular Dichroism studies, in: Med Chem Sicily 2018, 2018, pp. 18 - 18 (atti di: Med Chem Sicily 2018, Palermo, 17-20 July 2018) [Contribution to conference proceedings]

Wang, Li; Moraleda, Ignacio; Iriepa, Isabel; Romero, Alejandro; López-Muñoz, Francisco; Chioua, Mourad; Inokuchi, Tsutomu; Bartolini, Manuela; Marco-Contelles, José, 5-Methyl-N-(8-(5,6,7,8-tetrahydroacridin-9-ylamino)octyl)-5 H -indolo[2,3- b] quinolin-11-amine: a highly potent human cholinesterase inhibitor, «MEDCHEMCOMM», 2017, 8, pp. 1307 - 1317 [Scientific article]

Anna Tramarin, Edoardo Fabini, Manuela Bartolini, AChE inhibitors: affinity and kinetic studies using SPR technology, in: Quick Guide, 2017(atti di: Recent Developments in Pharmaceutical Analysis, Rimini, 20-23/09/2017) [Poster]

Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli, Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Chalcone-based carbamates for Alzheimer's disease treatment, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 749 - 764 [Scientific article]

Pérez-Areales, Francisco Javier; Betari, Nibal; Viayna, Antonio; Pont, Caterina; Espargarã³, Alba; Bartolini, Manuela; DE SIMONE, Angela; Rinaldi Alvarenga, José Fernando; Pã©rez, Belã©n; Sabate, Raimon; Lamuela-Raventós, Rosa Maria; Andrisano, Vincenza; Luque, Francisco Javier; Muñoz-Torrero, Diego, Design, synthesis and multitarget biological profiling of second-generation anti-Alzheimer rhein-huprine hybrids, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 965 - 981 [Scientific article]