Foto del docente

Manuela Bartolini

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [Scientific article]Open Access

Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela, Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease, «CHEMMEDCHEM», 2016, 11, pp. 1309 - 1317 [Scientific article]Open Access

Wang, C.H.; Alluri, S.; Nikogosyan, G.; Decarlo, C.; Monteiro, C.; Mabagos, G.; Feng, H.H.; White, A.R.; Bartolini, M.; Andrisano, V.; Zhang, L.K.; Ganguly, A.K, Novel synthesis of physovenine and physostigmine analogs, «TETRAHEDRON LETTERS», 2016, 57, pp. 3046 - 3049 [Scientific article]

Zha, Xiaoming; Lamba, Doriano; Zhang, Lili; Lou, Yinghan; Xu, Changxu; Kang, Di; Chen, Li; Xu, Yungen; Zhang, Luyong; De Simone, Angela; Samez, Sarah; Pesaresi, Alessandro; Stojan, Jure; Lopez, Manuela G.; Egea, Javier; Andrisano, Vincenza; Bartolini, Manuela, Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimers Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 114 - 131 [Scientific article]Open Access

Prati, Federica; Bergamini, Christian; Fato, Romana; Soukup, Ondrej; Korabecny, Jan; Andrisano, Vincenza; Bartolini, Manuela; Bolognesi, Maria Laura, Novel 8-Hydroxyquinoline Derivatives as Multitarget Compounds for the Treatment of Alzheimer's Disease, «CHEMMEDCHEM», 2016, 11, pp. 1284 - 1295 [Scientific article]

Simoni, Elena; Caporaso, Roberta; Bergamini, Christian; Fiori, Jessica; Fato, Romana; Miszta, Przemyslaw; Filipek, Sławomir; Caraci, Filippo; Giuffrida, Maria Laura; Andrisano, Vincenza; Minarini, Anna; Bartolini, Manuela; Rosini, Michela, Polyamine Conjugation as a Promising Strategy To Target Amyloid Aggregation in the Framework of Alzheimer’s Disease, «ACS MEDICINAL CHEMISTRY LETTERS», 2016, 7, pp. 1145 - 1150 [Scientific article]

De Simone, Angela; Bartolini, Manuela; Fiori, Jessica; D’Urzo, Annalisa; Naldi, Marina.; Andrisano, Vincenza, Analytical approaches in Alzheimer’s disease Drug Discovery, in: SIMCC 2015 - Spanish-Italian Medicinal Chemistry Congress - Book of Abstracts, 2015, pp. 35 - 35 (atti di: SIMCC 2015 - Spanish-Italian Medicinal Chemistry Congress, BARCELONA (SPAIN), JULY 12-15, 2015) [Contribution to conference proceedings]

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Aráoz, Rómulo; Bouet, Monika; Bartolini, Manuela; Coquelle, Nicolas; Colletier, Jacques-Philippe; Servent, Denis; Molgo, Jordi; Jean, Ludovic; Renard, Pierre-Yves, Multi-target directed ligands: Electrophysiological characterization of an anticholinesterase inhibitor coupled to an agonist of α7 nicotinic acetylcholine receptor, «BIOCHEMICAL PHARMACOLOGY», 2015, 97, pp. 621 - 621 [Abstract]

Bartolini, Manuela; Naldi, Marina; Andrisano, Vincenza, New analytical tools to investigate the role of protein glycosylation in Alzheimer’s disease, in: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, 2015, pp. 167 - 167 (atti di: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, Barcelona Biomedical Research Park, Barcellona, Spagna, July 12-15 2015) [Poster]

Bartolini, M.; Naldi, M.; Andrisano, V., ON-LINE GLYCAN RELEASE AND ANALYSIS BY AN INTEGRATED PNGASE F-IMER LC-ESI-Q-TOF APPROACH, in: IMASS PHARMA NETWORK 2015 Book of Abstracts, 2015, pp. 10 - 10 (atti di: IMASS PHARMA NETWORK 2015, Verona, Italia, 26-28 ottobre 2015) [Contribution to conference proceedings]

Bartolini, M.; Naldi, M.; Andrisano, V., PROTEIN GLYCOSILATION ANALYSIS BY AN INTEGRATED PNGASE-F-IMER-LC-ESI-Q-TOF APPROACH, in: Abstract Book - RDPA 2015, 2015, pp. 26 - 26 (atti di: RDPA 2015 - Recent Developments in Pharmaceutical Analysis, Perugia, June 28 - July 1, 2015) [Contribution to conference proceedings]

Diego Muñoz-Torrero; Irene Sola; Elisabet Viayna; Manuela Bartolini; Angela De Simone; Cheril Tapia-Rojas; Felipe G. Serrano; Raimon Sabaté; Jordi Juárez-Jiménez; Belén Pérez; F. Javier Luque; Vincenza Andrisano; M. Victòria Clos; Nibaldo C. Inestrosa, Synthesis, in vitro biological profiling and in vivo efficacy studies of novel multitarget disease-modifyng anti-Alzheimer drug candidates., in: I Simposio de Jóvenes Investigadores de la Sociedad Española de Química Terapéutica, 2014(atti di: I Simposio de Jóvenes Investigadores de la Sociedad Española de Química Terapéutica, Madrid, Maggio 2014) [Poster]

Viayna, E.; Sola, I.; Bartolini, M.; De Simone, A.; Tapia-Rojas, C.; Carvajal, F. J.; Serrano, F. G.; Sabate, R.; Juárez, J.; Pérez, B.; Badia, A.; Luque, F. J.; Andrisano, V.; Clos, M. V.; Inestrosa, N. C.; Muñoz-Torrero, D. ., Synthesis, molecular modelling, in vitro biological profiling, and in vivo efficacy studies of a novel family of huprine-based multi-target anti-alzheimer compounds., in: XVII National Meeting of the Spanish Society of Medicinal Chemistry., 2013(atti di: XVII National Meeting of the Spanish Society of Medicinal Chemistry., Madrid, Spagna, 2-4 Ottobre 2013) [Poster]

Andrisano, V.; Seidl, C.; Santos, C.; De Simone, A.; Bartolini, M. ., Uleine an indole alkaloid from Himatanthus lancifolius as acetylcholinesterase, butyrylcholinesterase, beta-secretase and beta-amyloid(1-42) spontaneous aggregation inhibitor., in: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, 2013(atti di: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, Florence, 6-10 Marzo 2013 .) [Poster]