Foto del docente

Manuela Bartolini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Bartolini, M.; Naldi, M.; Andrisano, V., ON-LINE GLYCAN RELEASE AND ANALYSIS BY AN INTEGRATED PNGASE F-IMER LC-ESI-Q-TOF APPROACH, in: IMASS PHARMA NETWORK 2015 Book of Abstracts, 2015, pp. 10 - 10 (atti di: IMASS PHARMA NETWORK 2015, Verona, Italia, 26-28 ottobre 2015) [Contribution to conference proceedings]

Bartolini, M.; Naldi, M.; Andrisano, V., PROTEIN GLYCOSILATION ANALYSIS BY AN INTEGRATED PNGASE-F-IMER-LC-ESI-Q-TOF APPROACH, in: Abstract Book - RDPA 2015, 2015, pp. 26 - 26 (atti di: RDPA 2015 - Recent Developments in Pharmaceutical Analysis, Perugia, June 28 - July 1, 2015) [Contribution to conference proceedings]

Diego Muñoz-Torrero; Irene Sola; Elisabet Viayna; Manuela Bartolini; Angela De Simone; Cheril Tapia-Rojas; Felipe G. Serrano; Raimon Sabaté; Jordi Juárez-Jiménez; Belén Pérez; F. Javier Luque; Vincenza Andrisano; M. Victòria Clos; Nibaldo C. Inestrosa, Synthesis, in vitro biological profiling and in vivo efficacy studies of novel multitarget disease-modifyng anti-Alzheimer drug candidates., in: I Simposio de Jóvenes Investigadores de la Sociedad Española de Química Terapéutica, 2014(atti di: I Simposio de Jóvenes Investigadores de la Sociedad Española de Química Terapéutica, Madrid, Maggio 2014) [Poster]

Viayna, E.; Sola, I.; Bartolini, M.; De Simone, A.; Tapia-Rojas, C.; Carvajal, F. J.; Serrano, F. G.; Sabate, R.; Juárez, J.; Pérez, B.; Badia, A.; Luque, F. J.; Andrisano, V.; Clos, M. V.; Inestrosa, N. C.; Muñoz-Torrero, D. ., Synthesis, molecular modelling, in vitro biological profiling, and in vivo efficacy studies of a novel family of huprine-based multi-target anti-alzheimer compounds., in: XVII National Meeting of the Spanish Society of Medicinal Chemistry., 2013(atti di: XVII National Meeting of the Spanish Society of Medicinal Chemistry., Madrid, Spagna, 2-4 Ottobre 2013) [Poster]

Andrisano, V.; Seidl, C.; Santos, C.; De Simone, A.; Bartolini, M. ., Uleine an indole alkaloid from Himatanthus lancifolius as acetylcholinesterase, butyrylcholinesterase, beta-secretase and beta-amyloid(1-42) spontaneous aggregation inhibitor., in: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, 2013(atti di: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, Florence, 6-10 Marzo 2013 .) [Poster]

De Simone, A; Mancini, F; Belluti, F; Bartolini, M; Bottegoni, G.; Rampa, A.; Cavalli, A.; Andrisano, V., Curcumin derivatives as beta-secretase (BACE1) inhibitors., in: Nuove Prospettive in Chimica Farmaceutica 6, 2012(atti di: Nuove Prospettive in Chimica Farmaceutica 6, Riccione, 11-13 Aprile) [Poster]

Rosini M.; Andrisano V.; Bartolini M.; Bolognesi M.L.; Hrelia P.; Minarini A.; Tarozzi A.; Melchiorre C., Lipocrine, a multipotent drug for the investigation of Alzheimer's disease, in: Trends in Drug Research, NOORDWIJKERHOUT, s.l., 2005(atti di: 15th Noordwijkerhout-Camerino Symposium, Noordwijkerhout, 8-13 May 2005) [Abstract]

Andrisano, V.; Bartolini, M.; Bertucci, C.; Cavrini, V.; Luppi, B.; Cerchiara, T., Analytical methods for the determination of folic acid in a polymeric micellar carrier, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2003, 32, pp. 983 - 989 [Scientific article]

Andrisano V.; Bartolini M.; Bertucci C.; Cavrini V.; Luppi B.; Cerchiara T., Analytical methods for the determination of folic acid in a polymeric micellar carrier, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2003, 32, pp. 983 - 989 [Scientific article]

Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valenti P.; Recanatini M., 3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy, «JOURNAL OF MEDICINAL CHEMISTRY», 2003, 46, pp. 2279 - 2282 [Scientific article]

Bolognesi M.L.; Bixel M.G.; Marucci G.; Bartolini M.; Krauss M.; Angeli P.; Antonello A.; Rosini M.; Tumiatti V.; Hucho F.; Melchiorre C., Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure, «JOURNAL OF MEDICINAL CHEMISTRY», 2002, 45, pp. 3286 - 3295 [Scientific article]

Rampa A.; Piazzi L.; Belluti F.; Gobbi S.; Bisi A.; Bartolini M.; Andrisano V.; Cavrini V.; Cavalli A.; Recanatini M.; Valenti P., Acetylcholinesterase inhibitors: SAR and kinetic studies on ω-[N-methyl-N-(3-alkylcarbamoyloxyphenyl]methyl] aminoalkoxyaryl derivatives, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 3810 - 3820 [Scientific article]

Recanatini M.; Cavalli A.; Belluti F.; Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Valenti P.; Andrisano V.; Bartolini M.; Cavrini V., SAR of 9-amino-1,2,3-4-tetrahydroacridine-based acetylcholinesterase inhibitors: Synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues, «JOURNAL OF MEDICINAL CHEMISTRY», 2000, 43, pp. 2007 - 2018 [Scientific article]