Tedesco D.; Maj M.; Malarczyk P.; Cingolani A.; Zaffagnini M.; Wnorowski A.; Czapinski J.; Benelli T.; Mazzoni R.; Bartolini M.; Jozwiak K., Application of the SMALP technology to the isolation of GPCRs from low-yielding cell lines, «BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES», 2021, 1863, Article number: 183641 , pp. 1 - 11 [Scientific article]
Naldi M.; Brusotti G.; Massolini G.; Andrisano V.; Temporini C.; Bartolini M., Bio-guided fractionation of stem bark extracts from phyllanthus muellarianus: Identification of phytocomponents with anti-cholinesterase activity, «MOLECULES», 2021, 26, Article number: 4376 , pp. 4376-1 - 4376-14 [Scientific article]Open Access
Baldassarre M.; Naldi M.; Zaccherini G.; Bartoletti M.; Antognoli A.; Laggetta M.; Gagliardi M.; Tufoni M.; Domenicali M.; Waterstradt K.; Paterini P.; Baldan A.; Leoni S.; Bartolini M.; Viale P.; Trevisani F.; Bernardi M.; Caraceni P., Determination of Effective Albumin in Patients With Decompensated Cirrhosis: Clinical and Prognostic Implications, «HEPATOLOGY», 2021, 74, pp. 2058 - 2073 [Scientific article]Open Access
Viayna, Elisabet; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Cisternas, Pedro; Oliva, Carolina A.; Sánchez-López, Elena; Ettcheto, Miren; Bartolini, Manuela; De Simone, Angela; Ricchini, Mattia; Rendina, Marisa; Pons, Mégane; Firuzi, Omidreza; Pérez, Belén; Saso, Luciano; Andrisano, Vincenza; Nachon, Florian; Brazzolotto, Xavier; García, Maria Luisa; Camins, Antoni; Silman, Israel; Jean, Ludovic; Inestrosa, Nibaldo C.; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero, Diego, Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 Mice, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 812 - 839 [Scientific article]Open Access
Talibov, Vladimir O; Fabini, Edoardo; FitzGerald, Edward A; Tedesco, Daniele; Cederfeldt, Daniela; Talu, Martin J; Rachman, Moira M; Mihalic, Filip; Manoni, Elisabetta; Naldi, Marina; Sanese, Paola; Forte, Giovanna; Lepore Signorile, Martina; Barril, Xavier; Simone, Cristiano; Bartolini, Manuela; Dobritzsch, Doreen; Del Rio, Alberto; Danielson, U Helena, Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase, «CHEMBIOCHEM», 2021, 22, pp. 1597 - 1608 [Scientific article]Open Access
Ramos, Gd; De Oliveira, As; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L; Fraser, Pe; Abreu, M; Kiametis, As; Gargano, R; Silveira, Er; Brand, Gd; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, Ml; Romeiro, Las, Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties, «RSC MEDICINAL CHEMISTRY», 2021, 12, pp. 1154 - 1163 [Scientific article]Open Access
Albertini C.; Naldi M.; Petralla S.; Strocchi S.; Grifoni D.; Monti B.; Bartolini M.; Bolognesi M.L., From combinations to single-molecule polypharmacology—cromolyn-ibuprofen conjugates for alzheimer’s disease, «MOLECULES», 2021, 26, Article number: 1112 , pp. 1 - 22 [Scientific article]Open Access
Pont, C.; Ginex, T.; Grinan-Ferre, C.; Scheiner, M.; Mattellone, A.; Martinez, N.; Arce, E. M.; Soriano-Fernandez, Y.; Naldi, M.; De Simone, A.; Barenys, M.; Gomez-Catalan, J.; Perez, B.; Sabate, R.; Andrisano, V.; Loza, M. I.; Brea, J.; Bartolini, M.; Bolognesi, M. L.; Decker, M.; Pallas, M.; Luque, F. J.; Munoz-Torrero, D., From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2021, 225, Article number: 113779 , pp. 1 - 25 [Scientific article]Open Access
Montanari S.; Allara M.; Scalvini L.; Kostrzewa M.; Belluti F.; Gobbi S.; Naldi M.; Rivara S.; Bartolini M.; Ligresti A.; Bisi A.; Rampa A., New Coumarin derivatives as cholinergic and cannabinoid system modulators, «MOLECULES», 2021, 26, Article number: 3254 , pp. 1 - 18 [Scientific article]Open Access
Gorecki L.; Uliassi E.; Bartolini M.; Janockova J.; Hrabinova M.; Hepnarova V.; Prchal L.; Muckova L.; Pejchal J.; Karasova J.Z.; Mezeiova E.; Benkova M.; Kobrlova T.; Soukup O.; Petralla S.; Monti B.; Korabecny J.; Bolognesi M.L., Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2021, 12, pp. 1698 - 1715 [Scientific article]Open Access
Rossi, M; Freschi, M; de Camargo Nascente, L; Salerno, A; de Melo Viana Teixeira, S; Nachon, F; Chantegreil, F; Soukup, O; Prchal, L; Malaguti, M; Bergamini, C; Bartolini, M; Angeloni, C; Hrelia, S; Soares Romeiro, La; Bolognesi, Ml., Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 4972 - 4990 [Scientific article]Open Access
Perone, R.; Albertini, C.; Uliassi, E.; Di Pietri, F.; de Sena Murteira Pinheiro, P.; Petralla, S.; Rizzardi, N.; Fato, R.; Pulkrabkova, L.; Soukup, O.; Tramarin, A.; Bartolini, M.; Bolognesi, M. L., Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy, «CHEMMEDCHEM», 2021, 16, pp. 187 - 198 [Scientific article]Open Access
De Simone, A.; Naldi, M.; Tedesco, D.; Bartolini, M.; Davani, L.; Andrisano, V., Advanced analytical methodologies in Alzheimer's disease drug discovery, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2020, 178, Article number: 112899 , pp. 1 - 25 [Scientific article]Open Access
Pérez-Areales, F Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer, Angel; Muñoz-Torrero, Diego, Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 9360 - 9390 [Scientific article]Open Access
Guzman, Laura; Besa, Gisela; Linares, Daniela; González, Lara; Pont, Caterina; Bartolini, Manuela; Haigis, Ann-Cathrin; Legradi, Jessica; Muñoz-Torrero, Diego; Gómez-Catalán, Jesús; Barenys, Marta, Evaluation of the effects of acetylcholinesterase inhibitors in the zebrafish touch-evoked response: quantitative vs. qualitative assessment, «ENVIRONMENTAL SCIENCES EUROPE», 2020, 32, Article number: 145 , pp. 1 - 12 [Scientific article]Open Access