Perone, R.; Albertini, C.; Uliassi, E.; Di Pietri, F.; de Sena Murteira Pinheiro, P.; Petralla, S.; Rizzardi, N.; Fato, R.; Pulkrabkova, L.; Soukup, O.; Tramarin, A.; Bartolini, M.; Bolognesi, M. L., Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy, «CHEMMEDCHEM», 2021, 16, pp. 187 - 198 [Scientific article]Open Access
De Simone A.; Naldi M.; Tedesco D.; Bartolini M.; Davani L.; Andrisano V., Advanced analytical methodologies in Alzheimer's disease drug discovery, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2020, 178, Article number: 112899 , pp. 1 - 25 [Scientific article]
Pérez-Areales, F Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer, Angel; Muñoz-Torrero, Diego, Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 9360 - 9390 [Scientific article]Open Access
Guzman, Laura; Besa, Gisela; Linares, Daniela; González, Lara; Pont, Caterina; Bartolini, Manuela; Haigis, Ann-Cathrin; Legradi, Jessica; Muñoz-Torrero, Diego; Gómez-Catalán, Jesús; Barenys, Marta, Evaluation of the effects of acetylcholinesterase inhibitors in the zebrafish touch-evoked response: quantitative vs. qualitative assessment, «ENVIRONMENTAL SCIENCES EUROPE», 2020, 32, Article number: 145 , pp. 1 - 12 [Scientific article]Open Access
Cieslikiewicz-Bouet, Monika; Naldi, Marina; Bartolini, Manuela; Pérez, Belén; Servent, Denis; Jean, Ludovic; Aráoz, Rómulo; Renard, Pierre-Yves, Functional characterization of multifunctional ligands targeting acetylcholinesterase and alpha 7 nicotinic acetylcholine receptor, «BIOCHEMICAL PHARMACOLOGY», 2020, 177, Article number: 114010 , pp. 1 - 11 [Scientific article]Open Access
Palmerini, Tullio; Barozzi, Chiara; Tomasi, Luciana; Riva, Diego Della; Marengo, Mario; Cicoria, Gianfranco; Bruno, Antonio G.; Bacchi-Reggiani, Maria-Letizia; Naldi, Marina; Bartolini, Manuela; Fanti, Stefano; Galiè, Nazzareno; Stone, Gregg W., In vitro thrombogenicity of drug-eluting and bare metal stents, «THROMBOSIS RESEARCH», 2020, 185, pp. 43 - 48 [Scientific article]
Bua G.; Tedesco D.; Conti I.; Reggiani A.; Bartolini M.; Gallinella G., No G-Quadruplex Structures in the DNA of Parvovirus B19: Experimental Evidence versus Bioinformatic Predictions, «VIRUSES», 2020, 12, Article number: 935 , pp. 935 - 935 [Scientific article]Open Access
Marques C.S.; Lopez O.; Bagetta D.; Carreiro E.P.; Petralla S.; Bartolini M.; Hoffmann M.; Alcaro S.; Monti B.; Bolognesi M.L.; Decker M.; Fernandez-Bolanos J.G.; Burke A.J., N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study, «BIOORGANIC CHEMISTRY», 2020, 98, Article number: 103753 , pp. 103753 - 103765 [Scientific article]
Bertoni S.; Tedesco D.; Bartolini M.; Prata C.; Passerini N.; Albertini B., Solid Lipid Microparticles for Oral Delivery of Catalase: Focus on the Protein Structural Integrity and Gastric Protection, «MOLECULAR PHARMACEUTICS», 2020, 17, pp. 3609 - 3621 [Scientific article]Open Access
Sanese, Paola; Fasano, Candida; Buscemi, Giacomo; Bottino, Cinzia; Corbetta, Silvia; Fabini, Edoardo; Silvestri, Valentina; Valentini, Virginia; Disciglio, Vittoria; Forte, Giovanna; Lepore Signorile, Martina; De Marco, Katia; Bertora, Stefania; Grossi, Valentina; Guven, Ummu; Porta, Natale; Di Maio, Valeria; Manoni, Elisabetta; Giannelli, Gianluigi; Bartolini, Manuela; Del Rio, Alberto; Caretti, Giuseppina; Ottini, Laura; Simone, Cristiano, Targeting SMYD3 to Sensitize Homologous Recombination-Proficient Tumors to PARP-Mediated Synthetic Lethality, «ISCIENCE», 2020, 23, pp. 101604 - 101604 [Scientific article]Open Access
Tramarin, Anna; Naldi, Marina; Degani, Genny; Lupu, Loredana; Wiegand, Pascal; Mazzolari, Angelica; Altomare, Alessandra; Aldini, Giancarlo; Popolo, Laura; Vistoli, Giulio; Przybylski, Michael; Bartolini, Manuela, Unveiling the molecular mechanisms underpinning biorecognition of early-glycated human serum albumin and receptor for advanced glycation end products, «ANALYTICAL AND BIOANALYTICAL CHEMISTRY», 2020, 412, pp. 4245 - 4259 [Scientific article]
Perez-Areales F.J.; Turcu A.L.; Barniol-Xicota M.; Pont C.; Pivetta D.; Espargaro A.; Bartolini M.; De Simone A.; Andrisano V.; Perez B.; Sabate R.; Sureda F.X.; Vazquez S.; Munoz-Torrero D., A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 180, pp. 613 - 626 [Scientific article]
Oukoloff, K.; Coquelle, N.; Bartolini, M.; Naldi, M.; Le Guevel, R.; Bach, S.; Josselin, B.; Ruchaud, S.; Catto, M.; Pisani, L.; Denora, N.; Iacobazzi, R. M.; Silman, I.; Sussman, J. L.; Buron, F.; Colletier, J. -P.; Jean, L.; Routier, S.; Renard, P. -Y., Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 168, pp. 58 - 77 [Scientific article]
Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolini M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A., Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 178, pp. 243 - 258 [Scientific article]Open Access
Scheiner M.; Dolles D.; Gunesch S.; Hoffmann M.; Nabissi M.; Marinelli O.; Naldi M.; Bartolini M.; Petralla S.; Poeta E.; Monti B.; Falkeis C.; Vieth M.; Hubner H.; Gmeiner P.; Maitra R.; Maurice T.; Decker M., Dual-Acting Cholinesterase-Human Cannabinoid Receptor 2 Ligands Show Pronounced Neuroprotection in Vitro and Overadditive and Disease-Modifying Neuroprotective Effects in Vivo, «JOURNAL OF MEDICINAL CHEMISTRY», 2019, 62, pp. 9078 - 9102 [Scientific article]Open Access