Foto del docente

Manuela Bartolini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Pont, Caterina; Sampietro, Anna; Pérez-Areales, F. Javier; Cristiano, Nunzia; Albalat, Agustí; Pérez, Belén; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Barenys, Marta; Teixidó, Elisabet; Sabaté, Raimon; Loza, M. Isabel; Brea, José; Muñoz-Torrero, Diego, Stepwise Structural Simplification of the Dihydroxyanthraquinone Moiety of a Multitarget Rhein-Based Anti-Alzheimer Lead to Improve Drug Metabolism and Pharmacokinetic Properties, «PHARMACEUTICS», 2024, 16, Article number: 982 , pp. 1 - 20 [Scientific article]Open Access

Sanese, Paola; De Marco, Katia; Lepore Signorile, Martina; La Rocca, Francesca; Forte, Giovanna; Latrofa, Marialaura; Fasano, Candida; Disciglio, Vittoria; Di Nicola, Elisabetta; Pantaleo, Antonino; Bianco, Giusy; Spilotro, Vito; Ferroni, Claudia; Tubertini, Matilde; Labarile, Nicoletta; De Marinis, Lucia; Armentano, Raffaele; Gigante, Gianluigi; Lantone, Valerio; Lantone, Giuliano; Naldi, Marina; Bartolini, Manuela; Varchi, Greta; Del Rio, Alberto; Grossi, Valentina; Simone, Cristiano, The novel SMYD3 inhibitor EM127 impairs DNA repair response to chemotherapy-induced DNA damage and reverses cancer chemoresistance, «JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH», 2024, 43, Article number: 151 , pp. 1 - 23 [Scientific article]Open Access

Giordani B.; Naldi M.; Croatti V.; Parolin C.; Erdogan U.; Bartolini M.; Vitali B., Exopolysaccharides from vaginal lactobacilli modulate microbial biofilms, «MICROBIAL CELL FACTORIES», 2023, 22, Article number: 45 , pp. 1 - 19 [Scientific article]Open Access

Carola Parolin, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolini, Beatrice Vitali, Exopolysaccharides released by vaginal Lactobacillus strains: chemical characterization and modulation of biofilm formation., in: Microbiology 2023 Proceedings, 2023, pp. 135 - 136 (atti di: Microbiology 2023 - XXXIV SIMGBM Congress, Cagliari, Italy, September 21-24, 2023) [Contribution to conference proceedings]

Basagni, Filippo; Ortega, Jose A; Bertozzi, Sine M; Armirotti, Andrea; Summa, Maria; Bertorelli, Rosalia; Bartolini, Manuela; Mellor, Ian R; Bedeschi, Martina; Bottegoni, Giovanni; Lembo, Vittorio; Minarini, Anna; Cavalli, Andrea; Rosini, Michela, Galantamine-memantine hybrids for Alzheimer's disease: The influence of linker rigidity in biological activity and pharmacokinetic properties, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2023, 261, Article number: 115803 , pp. 1 - 14 [Scientific article]Open Access

Beatrice Vitali, Barbara Giordani, Marina Naldi, Ülfet Erdoğan, Vanessa Croatti, Manuela Bartolini, Carola Parolin, Impact of Lactobacillus exopolysaccharides on vaginal microbial biofilms, in: FEMS 2023 - ABSTRACT BOOK, 2023, pp. 845 - 845 (atti di: FEMS 2023 - 10th Congress of European Microbiologists, Hamburg, Germany, 9-13 July 2023) [Contribution to conference proceedings]

Protti, Michele; Varfaj, Ina; Carotti, Andrea; Tedesco, Daniele; Bartolini, Manuela; Favilli, Alessandro; Gerli, Sandro; Mercolini, Laura; Sardella, Roccaldo, Microsampling and enantioselective liquid chromatography coupled to mass spectrometry for chiral bioanalysis of novel psychoactive substances, «TALANTA», 2023, 257, Article number: 124332 , pp. 1 - 9 [Scientific article]Open Access

Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML, Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease, «BIOORGANIC & MEDICINAL CHEMISTRY», 2023, 91, Article number: 117419 , pp. 1 - 9 [Scientific article]Open Access

Codony S.; Pont C.; Grinan-Ferre C.; Di Pede-Mattatelli A.; Calvo-Tusell C.; Feixas F.; Osuna S.; Jarne-Ferrer J.; Naldi M.; Bartolini M.; Loza M.I.; Brea J.; Perez B.; Bartra C.; Sanfeliu C.; Juarez-Jimenez J.; Morisseau C.; Hammock B.D.; Pallas M.; Vazquez S.; Munoz-Torrero D., Discovery and in Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 4909 - 4925 [Scientific article]Open Access

Gandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janočková, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero, Diego; Monti, Barbara; Sabaté, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura, Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2022, 13, pp. 3314 - 3329 [Scientific article]Open Access

Parenti, Md; Naldi, M; Manoni, E; Fabini, E; Cederfelt, D; Talibov, Vo; Gressani, V; Guven, U; Grossi, V; Fasano, C; Sanese, P; De Marco, K; Shtil, Aa; Kurkin, Av; Altieri, A; Danielson, Uh; Caretti, G; Simone, C; Varchi, G; Bartolini, M; Del Rio, A, Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2022, 243, pp. 114683 - 114695 [Scientific article]Open Access

Rapozzi V.; Moret F.; Menilli L.; Guerrini A.; Tedesco D.; Naldi M.; Bartolini M.; Gani M.; Zorzet S.; Columbaro M.; Milani C.; Martini C.; Ferroni C.; Varchi G., HSA-Binding Prodrugs-Based Nanoparticles Endowed with Chemo and Photo-Toxicity against Breast Cancer, «CANCERS», 2022, 14, Article number: 877 , pp. 877 - 902 [Scientific article]Open Access

Basagni, Filippo; Naldi, Marina; Ginex, Tiziana; Luque, F Javier; Fagiani, Francesca; Lanni, Cristina; Iurlo, Matteo; Marcaccio, Massimo; Minarini, Anna; Bartolini, Manuela; Rosini, Michela, Inhibition of β-Amyloid Aggregation in Alzheimer's Disease: The Key Role of (Pro)electrophilic Warheads, «ACS MEDICINAL CHEMISTRY LETTERS», 2022, 13, pp. 1812 - 1818 [Scientific article]Open Access

Bisi, A.; Feoli, A.; Trezza, A.; Viejo, L.; Formaggio, F.; Bartolini, M.; Belluti, F.; Gobbi, S.; Spiga, O.; Caprini, M.; de los Rios, C.; Castellano, S.; Rampa, A., Targeting neuronal calcium channels and GSK3β for Alzheimer's disease with naturally-inspired Diels-Alder adducts, «BIOORGANIC CHEMISTRY», 2022, 129, Article number: 106152 , pp. 106152 - 106166 [Scientific article]Open Access

Ismaili, L.; Monnin, J.; Etievant, A.; Arribas, R. L.; Viejo, L.; Refouvelet, B.; Soukup, O.; Janockova, J.; Hepnarova, V.; Korabecny, J.; Kucera, T.; Jun, D.; Andrys, R.; Musilek, K.; Baguet, A.; Garcia-Frutos, E. M.; De Simone, A.; Andrisano, V.; Bartolini, M.; De Los Rios, C.; Marco-Contelles, J.; Haffen, E., (±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2021, 12, pp. 1328 - 1342 [Scientific article]Open Access