Foto del docente

Maria Laura Bolognesi

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHEM-07/A Chimica farmaceutica

Coordinatrice del Corso di Dottorato in Drug discovery and development

Pubblicazioni

Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura*, A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential, «ACS CHEMICAL NEUROSCIENCE», 2019, 10, pp. 279 - 294 [articolo]

Carolina B. Moraes, Gesa Witt, Maria Kuzikov, Bernhard Ellinger, Theodora Calogeropoulou, Kyriakos C. Prousis, Stefano Mangani, Flavio Di Pisa, Giacomo Landi, Lucia Dello Iacono, Cecilia Pozzi, Lucio H. Freitas-Junior, Bruno dos Santos Pascoalino, Claudia P. Bertolacini, Birte Behrens, Oliver Keminer, Jennifer Leu, Markus Wolf, Jeanette Reinshagen, Anabela Cordeiro-da-Silva, Nuno Santarem, Alberto Venturelli, Stephen Wrigley, Deepa Karunakaran, Bethlehem Kebede, Ina Pöhner, Wolfgang Müller, Joanna Panecka-Hofman, Rebecca C. Wade, Martina Fenske, Joachim Clos, José María Alunda, María Jesús Corral, Elisa Uliassi, Maria Laura Bolognesi, Pasquale Linciano, Antonio Quotadamo, Stefania Ferrari, Matteo Santucci, Chiara Borsari, Maria Paola Costi, Sheraz Gul, Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform, «SLAS DISCOVERY», 2019, 24, pp. 346 - 361 [articolo]

Cerone M.; Uliassi E.; Prati F.; Ebiloma G.U.; Lemgruber L.; Bergamini C.; Watson D.G.; de A. M. Ferreira T.; Roth Cardoso G.S.H.; Soares Romeiro L.A.; de Koning H.P.; Bolognesi M.L., Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)-Based Hybrids Target Mitochondrial Function and ATP Production in Trypanosoma brucei, «CHEMMEDCHEM», 2019, 14, pp. 621 - 635 [articolo]

Alcaro S.; Bolognesi M.; Garcia-Sosa A.T.; Rapposelli S., Editorial: Multi-target-directed ligands (MTDL) as challenging research tools in drug discovery: From design to pharmacological evaluation, «FRONTIERS IN CHEMISTRY», 2019, 7, pp. 71 - 72 [replica/breve intervento]Open Access

Bolognesi M.L., Harnessing Polypharmacology with Medicinal Chemistry, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 273 - 275 [articolo]

Ivasiv, V.; Albertini, C.; Goncalves, A. E.; Rossi, M.; Bolognesi, M., Molecular hybridization as a tool for designing multitarget drug candidates for complex diseases, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2019, 19, pp. 1694 - 1711 [articolo]

Romeiro L.A.S.; Da Costa Nunes J.L.; De Oliveira Miranda C.; Simoies Heyn Roth Cardoso G.; De Oliveira A.S.; Gandini A.; Kobrlova T.; Soukup O.; Rossi Michele.; Senger J.; Jung M.; Gervasoni S.; Vistoli G.; Petralla S.; Massenzio F.; Monti B.; Bolognesi M.L., Novel Sustainable-by-Design HDAC Inhibitors for the Treatment of Alzheimer's Disease, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 671 - 676 [articolo]

Lanthier, Caroline; Payan, Hugo; Liparulo, Irene; Hatat, Bérénice; Lecoutey, Cédric; Since, Marc; Davis, Audrey; Bergamini, Christian; Claeysen, Sylvie; Dallemagne, Patrick; Bolognesi, Maria-Laura; Rochais, Christophe, Novel multi target-directed ligands targeting 5-HT4 receptors with in cellulo antioxidant properties as promising leads in Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 182, pp. 111596 - 111607 [articolo]

Moda F.; Bolognesi M.L.; Legname G., Novel screening approaches for human prion diseases drug discovery, «EXPERT OPINION ON DRUG DISCOVERY», 2019, 14, pp. 983 - 993 [articolo]

Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.-J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K., Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 168, pp. 491 - 514 [articolo]Open Access

Michela Freschi, Cristina Angeloni, Michele Rossi, Marco Malaguti, Luiz Antonio Soares Romeiro, Luciana de Camargo Nascente, Maria Laura Bolognesi, Silvana Hrelia, STUDY OF THE ANTI-INFLAMMATORY ACTIVITY OF NOVEL TACRINE DERIVATIVES WITH LIPIDS EXTRACTED FROM CASHEW NUT SHELL LIQUID, in: Comitato scientifico, 1st International Conference on Neuroprotection by Drugs, Nutraceuticals and Physical Activity, 2019, pp. 66 - 66 (atti di: 1st International Conference on Neuroprotection by Drugs, Nutraceuticals and Physical Activity, Rimini, 6-7 giugno) [atti di convegno-abstract]

Staderini M.; Piquero M.; Abengozar M.A.; Nacher-Vazquez M.; Romanelli G.; Lopez-Alvarado P.; Rivas L.; Bolognesi M.L.; Menendez J.C., Structure-activity relationships and mechanistic studies of novel mitochondria-targeted, leishmanicidal derivatives of the 4-aminostyrylquinoline scaffold, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 171, pp. 38 - 53 [articolo]

Bolognesi M.L., Sustainable anti-trypanosomatid drugs: An aspirational goal for medicinal chemistry, in: Annual Reports in Medicinal Chemistry, 525 B STREET, SUITE 1900, SAN DIEGO, CA 92101-4495 USA, Academic Press Inc., 2019, pp. 153 - 176 [capitolo di libro]

Roldan-Pena J.M.; Romero-Real V.; Hicke J.; Maya I.; Franconetti A.; Lagunes I.; Padron J.M.; Petralla S.; Poeta E.; Naldi M.; Bartolini M.; Monti B.; Bolognesi M.; Lopez O.; Fernandez-Bolanos J.G., Tacrine-O-protected phenolics heterodimers as multitarget-directed ligands against Alzheimer's disease: Selective subnanomolar BuChE inhibitors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 181, Article number: 111550, pp. 111550 - 111565 [articolo]

Bolognesi M.L.; Ganamet K.L.; Liu H.; Poulsen S.-A.; Georg G.I.; Wang S., Women in Medicinal Chemistry Special Issue Call for Papers, «JOURNAL OF MEDICINAL CHEMISTRY», 2019, 62, pp. 3783 - 3783 [replica/breve intervento]