Foto del docente

Maria Laura Bolognesi

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Coordinatrice del Corso di Dottorato in Scienze biotecnologiche, biocomputazionali, farmaceutiche e farmacologiche

Pubblicazioni

Rossi M, Freschi M, de Camargo Nascente L, Salerno A, de Melo Viana Teixeira S, Nachon F, Chantegreil F, Soukup O, Prchal L, Malaguti M, Bergamini C, Bartolini M, Angeloni C, Hrelia S, Soares Romeiro LA, Bolognesi ML., Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 4972 - 4990 [articolo]Open Access

Espro C.; Paone E.; Mauriello F.; Gotti R.; Uliassi E.; Bolognesi M.L.; Rodriguez-Padron D.; Luque R., Sustainable production of pharmaceutical, nutraceutical and bioactive compounds from biomass and waste, «CHEMICAL SOCIETY REVIEWS», 2021, 50, pp. 11191 - 11207 [articolo]

Perone R.; Albertini C.; Uliassi E.; Di Pietri F.; de Sena Murteira Pinheiro P.; Petralla S.; Rizzardi N.; Fato R.; Pulkrabkova L.; Soukup O.; Tramarin A.; Bartolini M.; Bolognesi M.L., Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy, «CHEMMEDCHEM», 2021, 16, pp. 187 - 198 [articolo]Open Access

Huryn D.M.; Bolognesi M.L., A Different Kind of Medicinal Chemistry Toolbox, «ACS MEDICINAL CHEMISTRY LETTERS», 2020, 11, pp. 245 - 248 [articolo]Open Access

Rodrigues D.A.; Pinheiro P.D.S.M.; Sagrillo F.S.; Bolognesi M.L.; Fraga C.A.M., Histone deacetylases as targets for the treatment of neurodegenerative disorders: Challenges and future opportunities, «MEDICINAL RESEARCH REVIEWS», 2020, 40, pp. 2177 - 2211 [articolo]

Linciano P.; Cullia G.; Borsari C.; Santucci M.; Ferrari S.; Witt G.; Gul S.; Kuzikov M.; Ellinger B.; Santarem N.; Cordeiro da Silva A.; Conti P.; Bolognesi M.L.; Roberti M.; Prati F.; Bartoccini F.; Retini M.; Piersanti G.; Cavalli A.; Goldoni L.; Bertozzi S.M.; Bertozzi F.; Brambilla E.; Rizzo V.; Piomelli D.; Pinto A.; Bandiera T.; Costi M.P., Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2020, 189, Article number: 112047, pp. N/A - N/A [articolo]

Zaccagnini L.; Rossetti G.; Tran T.H.; Salzano G.; Gandini A.; Colini Baldeschi A.; Bolognesi M.L.; Carloni P.; Legname G., In silico/in vitro screening and hit evaluation identified new phenothiazine anti-prion derivatives, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2020, 196, Article number: 112295, pp. 1 - 16 [articolo]

Rossi M.; Petralla S.; Protti M.; Baiula M.; Kobrlova T.; Soukup O.; Spampinato S.M.; Mercolini L.; Monti B.; Bolognesi M.L., α-linolenic acid-valproic acid conjugates: Toward single-molecule polypharmacology for multiple sclerosis, «ACS MEDICINAL CHEMISTRY LETTERS», 2020, 11, pp. 2406-2413 - 2413 [articolo]Open Access

Marques C.S.; Lopez O.; Bagetta D.; Carreiro E.P.; Petralla S.; Bartolini M.; Hoffmann M.; Alcaro S.; Monti B.; Bolognesi M.L.; Decker M.; Fernandez-Bolanos J.G.; Burke A.J., N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study, «BIOORGANIC CHEMISTRY», 2020, 98, Article number: 103753, pp. 103753 - 103765 [articolo]

Al-Tel T.H.; Srinivasulu V.; Ramanathan M.; Soares N.C.; Sebastian A.; Bolognesi M.L.; Abu-Yousef I.A.; Majdalawieh A., Stereocontrolled transformations of cyclohexadienone derivatives to access stereochemically rich and natural product-inspired architectures, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2020, 18, pp. 8526 - 8571 [articolo]

Bolognesi M.L.; Ganamet K.L.; Liu H.; Poulsen S.-A.; Georg G.I.; Wang S., Women in Medicinal Chemistry: Ad Maiora!, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 1777 - 1778 [replica/breve intervento]Open Access

Uliassi, Elisa; Pena-Altamira, Luis Emiliano; Morales, Aixa V.; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martinez Gonzalez, Loreto; Martinez, Ana; Monti, Barbara; Bolognesi, Maria Laura*, A Focused Library of Psychotropic Analogues with Neuroprotective and Neuroregenerative Potential, «ACS CHEMICAL NEUROSCIENCE», 2019, 10, pp. 279 - 294 [articolo]

Carolina B. Moraes, Gesa Witt, Maria Kuzikov, Bernhard Ellinger, Theodora Calogeropoulou, Kyriakos C. Prousis, Stefano Mangani, Flavio Di Pisa, Giacomo Landi, Lucia Dello Iacono, Cecilia Pozzi, Lucio H. Freitas-Junior, Bruno dos Santos Pascoalino, Claudia P. Bertolacini, Birte Behrens, Oliver Keminer, Jennifer Leu, Markus Wolf, Jeanette Reinshagen, Anabela Cordeiro-da-Silva, Nuno Santarem, Alberto Venturelli, Stephen Wrigley, Deepa Karunakaran, Bethlehem Kebede, Ina Pöhner, Wolfgang Müller, Joanna Panecka-Hofman, Rebecca C. Wade, Martina Fenske, Joachim Clos, José María Alunda, María Jesús Corral, Elisa Uliassi, Maria Laura Bolognesi, Pasquale Linciano, Antonio Quotadamo, Stefania Ferrari, Matteo Santucci, Chiara Borsari, Maria Paola Costi, Sheraz Gul, Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform, «SLAS DISCOVERY», 2019, 24, pp. 346 - 361 [articolo]

Cerone M.; Uliassi E.; Prati F.; Ebiloma G.U.; Lemgruber L.; Bergamini C.; Watson D.G.; de A. M. Ferreira T.; Roth Cardoso G.S.H.; Soares Romeiro L.A.; de Koning H.P.; Bolognesi M.L., Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)-Based Hybrids Target Mitochondrial Function and ATP Production in Trypanosoma brucei, «CHEMMEDCHEM», 2019, 14, pp. 621 - 635 [articolo]

Alcaro S.; Bolognesi M.; Garcia-Sosa A.T.; Rapposelli S., Editorial: Multi-target-directed ligands (MTDL) as challenging research tools in drug discovery: From design to pharmacological evaluation, «FRONTIERS IN CHEMISTRY», 2019, 7, pp. 71 - 72 [replica/breve intervento]Open Access