Foto del docente

Maria Laura Bolognesi

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Coordinatrice del Corso di Dottorato in Scienze biotecnologiche, biocomputazionali, farmaceutiche e farmacologiche

Pubblicazioni

Bolognesi M.L., Harnessing Polypharmacology with Medicinal Chemistry, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 273 - 275 [articolo]

Ivasiv V.; Albertini C.; Goncalves A.E.; Rossi M.; Bolognesi M., Molecular hybridization as a tool for designing multitarget drug candidates for complex diseases, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2019, 19, pp. 1694 - 1711 [articolo]

Romeiro L.A.S.; Da Costa Nunes J.L.; De Oliveira Miranda C.; Simoies Heyn Roth Cardoso G.; De Oliveira A.S.; Gandini A.; Kobrlova T.; Soukup O.; Rossi Michele.; Senger J.; Jung M.; Gervasoni S.; Vistoli G.; Petralla S.; Massenzio F.; Monti B.; Bolognesi M.L., Novel Sustainable-by-Design HDAC Inhibitors for the Treatment of Alzheimer's Disease, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 671 - 676 [articolo]

Lanthier, Caroline; Payan, Hugo; Liparulo, Irene; Hatat, Bérénice; Lecoutey, Cédric; Since, Marc; Davis, Audrey; Bergamini, Christian; Claeysen, Sylvie; Dallemagne, Patrick; Bolognesi, Maria-Laura; Rochais, Christophe, Novel multi target-directed ligands targeting 5-HT4 receptors with in cellulo antioxidant properties as promising leads in Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 182, pp. 111596 - 111607 [articolo]

Moda F.; Bolognesi M.L.; Legname G., Novel screening approaches for human prion diseases drug discovery, «EXPERT OPINION ON DRUG DISCOVERY», 2019, 14, pp. 983 - 993 [articolo]

Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.-J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K., Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 168, pp. 491 - 514 [articolo]

Michela Freschi, Cristina Angeloni, Michele Rossi, Marco Malaguti, Luiz Antonio Soares Romeiro, Luciana de Camargo Nascente, Maria Laura Bolognesi, Silvana Hrelia, STUDY OF THE ANTI-INFLAMMATORY ACTIVITY OF NOVEL TACRINE DERIVATIVES WITH LIPIDS EXTRACTED FROM CASHEW NUT SHELL LIQUID, in: Comitato scientifico, 1st International Conference on Neuroprotection by Drugs, Nutraceuticals and Physical Activity, 2019, pp. 66 - 66 (atti di: 1st International Conference on Neuroprotection by Drugs, Nutraceuticals and Physical Activity, Rimini, 6-7 giugno) [atti di convegno-abstract]

Staderini M.; Piquero M.; Abengozar M.A.; Nacher-Vazquez M.; Romanelli G.; Lopez-Alvarado P.; Rivas L.; Bolognesi M.L.; Menendez J.C., Structure-activity relationships and mechanistic studies of novel mitochondria-targeted, leishmanicidal derivatives of the 4-aminostyrylquinoline scaffold, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 171, pp. 38 - 53 [articolo]

Bolognesi M.L., Sustainable anti-trypanosomatid drugs: An aspirational goal for medicinal chemistry, in: Annual Reports in Medicinal Chemistry, 525 B STREET, SUITE 1900, SAN DIEGO, CA 92101-4495 USA, Academic Press Inc., 2019, pp. 153 - 176 [capitolo di libro]

Roldan-Pena J.M.; Romero-Real V.; Hicke J.; Maya I.; Franconetti A.; Lagunes I.; Padron J.M.; Petralla S.; Poeta E.; Naldi M.; Bartolini M.; Monti B.; Bolognesi M.; Lopez O.; Fernandez-Bolanos J.G., Tacrine-O-protected phenolics heterodimers as multitarget-directed ligands against Alzheimer's disease: Selective subnanomolar BuChE inhibitors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 181, Article number: 111550, pp. 111550 - 111565 [articolo]

Bolognesi M.L.; Ganamet K.L.; Liu H.; Poulsen S.-A.; Georg G.I.; Wang S., Women in Medicinal Chemistry Special Issue Call for Papers, «JOURNAL OF MEDICINAL CHEMISTRY», 2019, 62, pp. 3783 - 3783 [replica/breve intervento]

Ramsay, Rona R; Popovic-Nikolic, Marija R; Nikolic, Katarina; Uliassi, Elisa; Bolognesi, Maria Laura, A perspective on multi-target drug discovery and design for complex diseases, «CLINICAL AND TRANSLATIONAL MEDICINE», 2018, 7, Article number: 3, pp. 1 - 14 [articolo]Open Access

Prati, Federica; Bottegoni, Giovanni; Bolognesi, Maria Laura; Cavalli, Andrea, BACE-1 Inhibitors: From Recent Single-Target Molecules to Multitarget Compounds for Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 619 - 637 [articolo]

Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura*, Development of a Focused Library of Triazole-Linked Privileged-Structure-Based Conjugates Leading to the Discovery of Novel Phenotypic Hits against Protozoan Parasitic Infections, «CHEMMEDCHEM», 2018, 13, pp. 678 - 683 [articolo]

Brevetto n. PCT/IT2018/000084, Electrospun fibers for a local release of an anti-inflammatory and a promyelinating drug. Open Access