Foto del docente

Maria Laura Bolognesi

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Coordinatrice del Corso di Dottorato in Scienze biotecnologiche, biocomputazionali, farmaceutiche e farmacologiche

Pubblicazioni

Staderini, Matteo; Martín, María Antonia; Bolognesi, Maria Laura; Menéndez, J. Carlos, Imaging of β-amyloid plaques by near infrared fluorescent tracers: A new frontier for chemical neuroscience, «CHEMICAL SOCIETY REVIEWS», 2015, 44, pp. 1807 - 1819 [articolo]

Matteo Staderini;Maria Laura Bolognesi;J. Carlos Menéndez, Lewis Acid-Catalyzed Generation of CC and CN Bonds on π-Deficient Heterocyclic Substrates, «ADVANCED SYNTHESIS & CATALYSIS», 2015, 357, pp. 185 - 195 [articolo]

Maria Bolognesi, Recensione a: Meet the Editorial Board:, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2015, 15, pp. 197 - 197 [recensione]

Prati F;De Simone A;Bisignano P;Armirotti A;Summa M;Pizzirani D;Scarpelli R;Perez DI;Andrisano V;Perez-Castillo A;Monti B;Massenzio F;Polito L;Racchi M;Favia AD;Bottegoni G;Martinez A;Bolognesi ML;Cavalli A, Multitarget drug discovery for Alzheimer's disease: triazinones as BACE-1 and GSK-3β inhibitors., «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2015, 54, pp. 1578 - 1582 [articolo]

Benchekroun, M.; Bartolini, M.; Egea, J.; Romero, A.; Soriano, E.; Pudlo, M.; Luzet, V.; Andrisano, V.; Jimeno, M.-L.; Lopez, M.G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; De Andres, L.; Herrera-Arozamena, C.; Monti, B.; Bolognesi, M.L.; Rodriguez-Franco, M.I.; Decker, M.; Marco-Contelles, J.; Ismaili, L., Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids, «CHEMMEDCHEM», 2015, 10, pp. 523 - 539 [articolo]

De Vin, Filip; Choi, Sze Men; Bolognesi, Maria L.; Lefebvre, Romain A, Presynaptic M3 muscarinic cholinoceptors mediate inhibition of excitatory synaptic transmission in area CA1 of rat hippocampus, «BRAIN RESEARCH», 2015, 1629, pp. 260 - 269 [articolo]

Bolognesi, Maria Laura; Bongarzone, Salvatore; Aulic, Suzana; Ai Tran, Hoang Ngoc; Prati, Federica; Carloni, Paolo; Legname, Giuseppe, Rational approach to an antiprion compound with a multiple mechanism of action, «FUTURE MEDICINAL CHEMISTRY», 2015, 7, pp. 2113 - 2120 [articolo]

Prati, F.; Bolognesi, M. L, Tackling neurodegeneration with multi-target and theranostic small molecules, in: 2015 Medicinal Chemistry Reviews, Washington,, ACS Division of Medicinal Chemistry, 2015, pp. 347 - 356 [capitolo di libro]

Santucci, Matteo; Vignudelli, Tatiana; Ferrari, Stefania; Mor, Marco; Scalvini, Laura; Bolognesi, Maria Laura; Uliassi, Elisa; Costi, Maria Paola, The Hippo Pathway and YAP/TAZ-TEAD Protein-Protein Interaction as Targets for Regenerative Medicine and Cancer Treatment, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 4857 - 4873 [articolo]

Prati, Federica; Bergamini, Christian; Molina, Maria Teresa; Falchi, Federico; Cavalli, Andrea; Kaiser, Marcel; Brun, Reto; Fato, Romana; Bolognesi, Maria Laura, 2-Phenoxy-1,4-naphthoquinones: From a Multitarget Antitrypanosomal to a Potential Antitumor Profile, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 6422 - 6434 [articolo]

Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpelli, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L., 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2015, 6, pp. 1665 - 1682 [articolo]Open Access

Maria, Bolognesi, Biotecnologie e scoperta dei farmaci, in: Chimica organica medica e farmaceutica, Rozzano Milano, Zanichelli Editore spa, 2014, pp. 119 - 154 . Opera originale: Autore: John M. Beale, Jr. - Titolo: Biotechnology and drug discovery [contributo in volume (traduzione)]

Eugenie Nepovimova;Elisa Uliassi;Jan Korabecny;Luis Emiliano Peña-Altamira;Sarah Samez;Alessandro Pesaresi;Gregory E. Garcia;Manuela Bartolini;Vincenza Andrisano;Christian Bergamini;Romana Fato;Doriano Lamba;Marinella Roberti;Kamil Kuca;Barbara Monti;Maria Laura Bolognesi, Multitarget Drug Design Strategy: Quinone–Tacrine Hybrids Designed To Block Amyloid-β Aggregation and To Exert Anticholinesterase and Antioxidant Effects, «JOURNAL OF MEDICINAL CHEMISTRY», 2014, 57, pp. 8576 - 8589 [articolo]

Salvatore Bongarzone;Matteo Staderini;Maria Laura Bolognesi, Multitarget ligands and theranostics: sharpening the medicinal chemistry sword against prion diseases, «FUTURE MEDICINAL CHEMISTRY», 2014, 6, pp. 1017 - 1029 [articolo]

Federica Prati; Maria Laura Bolognesi, PHENOTYPIC HITS IN ANTI-TRYPANOSOMA DRUG DISCOVERY, «LA CHIMICA E L'INDUSTRIA», 2014, XCVI, pp. 46 - 47 [articolo]