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Maria Laura Bolognesi

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHEM-07/A Chimica farmaceutica

Coordinatrice del Corso di Dottorato in Drug discovery and development

Pubblicazioni

Uliassi, Elisa; Fiorani, Giulia; Krauth-Siegel, R. Luise; Bergamini, Christian; Fato, Romana; Bianchini, Giulia; Carlos Menéndez, J.; Molina, Maria Teresa; López-Montero, Eulogio; Falchi, Federico; Cavalli, Andrea; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura*, Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activity, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 141, pp. 138 - 148 [articolo]

Gandini, Annachiara; Prati, Federica; Uliassi, Elisa; Bolognesi, Maria L., Drug Discovery Strategies for the Generation of Multitarget Ligands against Neglected Tropical Diseases, in: Drug Selectivity: An Evolving Concept in Medicinal Chemistry, Weinheim, Wiley‐VCH Verlag GmbH & Co. KGaA, 2017, pp. 135 - 159 (METHODS AND PRINCIPLES IN MEDICINAL CHEMISTRY) [capitolo di libro]

Bolognesi, M.L.*, From Imaging Agents to Theranostic Drugs in Alzheimer's Disease, in: Bolognesi, M.L.*, Comprehensive Medicinal Chemistry III, Amsterdam, Elsevier Inc., 2017, pp. 74 - 106 [capitolo di libro]

Uliassi, Elisa*; Prati, Federica; Bongarzone, Salvatore; Bolognesi, Maria Laura, Medicinal Chemistry of Hybrids for Neurodegenerative Diseases, in: Uliassi, Elisa*, Design of Hybrid Molecules for Drug Development, oxford, Elsevier Inc., 2017, pp. 259 - 277 [capitolo di libro]

Huryn, Donna M.*; Bolognesi, Maria Laura; Young, Wendy B., Medicinal Chemistry: Where Are All the Women?, «ACS MEDICINAL CHEMISTRY LETTERS», 2017, 8, pp. 900 - 902 [articolo]

Bruno, Stefano; Uliassi, Elisa; Zaffagnini, Mirko; Prati, Federica; Bergamini, Christian; Amorati, Riccardo; Paredi, Gianluca; Margiotta, Marilena; Conti, Paola; Costi, Maria Paola; Kaiser, Marcel; Cavalli, Andrea; Fato, Romana; Bolognesi, Maria Laura, Molecular basis for covalent inhibition of glyceraldehyde-3-phosphate dehydrogenase by a 2-phenoxy-1,4-naphthoquinone small molecule, «CHEMICAL BIOLOGY & DRUG DESIGN», 2017, 89, pp. 1 - 11 [articolo]

Bolognesi, Maria Laura*, Neurodegenerative drug discovery: Building on the past, looking to the future, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 707 - 709 [replica/breve intervento]

Uliassi, Elisa; Gandini, Annachiara; Perone, Rosaria Carmela; Bolognesi, Maria Laura*, Neuroregeneration versus neurodegeneration: Toward a paradigm shift in Alzheimer's disease drug discovery, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 995 - 1013 [articolo]

Roldán-Peña, Jesús M.; Alejandre-Ramos, Daniel; López, O scar; Maya, Inés; Lagunes, Irene; Padrón, José M.; Peña-Altamira, Luis Emiliano; Bartolini, Manuela; Monti, Barbara; Bolognesi, Maria L.; Fernández-Bolaños, José G., New tacrine dimers with antioxidant linkers as dual drugs: Anti-Alzheimer's and antiproliferative agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 138, pp. 761 - 773 [articolo]Open Access

Peña-Altamira, E; Petralla, S; Massenzio, F; Virgili, M; Bolognesi, Ml; Monti, B., Nutritional and Pharmacological Strategies to Regulate Microglial Polarization in Cognitive Aging and Alzheimer's Disease., «FRONTIERS IN AGING NEUROSCIENCE», 2017, 9, pp. 1 - 15 [articolo]

Maria Laura Bolognesi, Sustainable Multi-Target Drugs for Neglected Tropical Diseases Caused by Trypanosomatids: Dream or Reality?, «PROCEEDINGS», 2017, 1, pp. 664 - 665 [abstract]Open Access

Jeřábek, Jakub; Uliassi, Elisa; Guidotti, Laura; Korábečný, Jan; Soukup, Ondřej; Sepsova, Vendula; Hrabinova, Martina; Kuča, Kamil; Bartolini, Manuela; Peña-Altamira, Luis Emiliano; Petralla, Sabrina; Monti, Barbara; Roberti, Marinella; Bolognesi, Maria Laura, Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 127, pp. 250 - 262 [articolo]

Gandini, Annachiara; Bolognesi, Maria Laura*, Therapeutic Approaches to Prion Diseases, in: Gandini, Annachiara, Progress in Molecular Biology and Translational Science, Cambridge, Elsevier B.V., 2017, pp. 433 - 453 [capitolo di libro]

Chacón-Vargas, Karla Fabiola; Nogueda-Torres, Benjamin; Sánchez-Torres, Luvia E.; Suarez-Contreras, Erick; Villalobos-Rocha, Juan Carlos; Torres-Martinez, Yuridia; Lara-Ramirez, Edgar E.; Fiorani, Giulia; Krauth-Siegel, R Luise; Bolognesi, Maria Laura; Monge, Antonio; Rivera, Gildardo, Trypanocidal activity of quinoxaline 1,4 Di-N-oxide derivatives as trypanothione reductase inhibitors, «MOLECULES», 2017, 22, Article number: 220, pp. 1 - 18 [articolo]Open Access

Lemes, Laís Flávia Nunes; De Andrade Ramos, Giselle; De Oliveira, Andressa Souza; Da Silva, Fernanda Motta R.; De Castro Couto, Gina; Da Silva Boni, Marina; Guimarães, Marcos Jorge R.; Souza, Isis Nem O.; Bartolini, Manuela; Andrisano, Vincenza; Do Nascimento Nogueira, Patrícia Coelho; Silveira, Edilberto Rocha; Brand, Guilherme D.; Soukup, Ondřej; Korábečný, Jan; Romeiro, Nelilma C.; Castro, Newton G.; Bolognesi, Maria Laura; Romeiro, Luiz Antonio Soares, Cardanol-derived AChE inhibitors: Towards the development of dual binding derivatives for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 108, pp. 687 - 700 [articolo]