35805 - Molecular Design Strategies with lab

Academic Year 2010/2011

  • Docente: Maurizio Recanatini
  • Credits: 5
  • SSD: CHIM/08
  • Language: Italian
  • Moduli: Maurizio Recanatini (Modulo 1) Marinella Roberti (Modulo 2)
  • Teaching Mode: Traditional lectures (Modulo 1) Traditional lectures (Modulo 2)
  • Campus: Bologna
  • Corso: Second cycle degree programme (LM) in Pharmaceutical Biotecnology (cod. 8180)

Course contents

1) Drugs, discovery,and design
- Drugs and biologically active compounds
- Drug discovery: the classical paradigm in the post-genomic era
- Rational drug design

2) Molecular modeling (basic concepts)

3) Pharmacophore-based drug design

4) Target-based drug design

5) Combinatorial chemistry: a tool for drug discovery

Office hours

See the website of Maurizio Recanatini

See the website of Marinella Roberti