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Rita Morigi

Professoressa associata

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

Marzano S.; Miglietta G.; Morigi R.; Marinello J.; Arleo A.; Procacci M.; Locatelli A.; Leoni A.; Pagano B.; Randazzo A.; Amato J.; Capranico G., Balancing Affinity, Selectivity, and Cytotoxicity of Hydrazone-Based G-Quadruplex Ligands for Activation of Interferon β Genes in Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 12055 - 12067 [articolo]Open Access

Francesca Bonvicini, Alessandra Locatelli, Rita Morigi, Alberto Leoni, Giovanna Angela Gentilomi, Isatin Bis-Indole and Bis-Imidazothiazole Hybrids: Synthesis and Antimicrobial Activity, «MOLECULES», 2022, 27, pp. 5781 - 5792 [articolo]Open Access

Das A.; Greco G.; Kumar S.; Catanzaro E.; Morigi R.; Locatelli A.; Schols D.; Alici H.; Tahtaci H.; Ravindran F.; Fimognari C.; Karki S.S., Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives, «COMPUTATIONAL BIOLOGY AND CHEMISTRY», 2022, 97, Article number: 107641, pp. 1 - 18 [articolo]Open Access

Morigi R.; Catanzaro E.; Locatelli A.; Calcabrini C.; Pellicioni V.; Leoni A.; Fimognari C., Synthesis and biological evaluation of new bis-indolinone derivatives endowed with cytotoxic activity, «MOLECULES», 2021, 26, Article number: 6277, pp. 1 - 15 [articolo]Open Access

Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N., Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth, «MOLECULES», 2020, 25, Article number: 4438, pp. 1 - 15 [articolo]Open Access

Amato J.; Miglietta G.; Morigi R.; Iaccarino N.; Locatelli A.; Leoni A.; Novellino E.; Pagano B.; Capranico G.; Randazzo A., Monohydrazone Based G-Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 3090 - 3103 [articolo]Open Access

Emanuela Pesce, Nicoletta Pedemonte, Alberto Leoni, Alessandra Locatelli, Rita Morigi, Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis., «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2020, 30, Article number: 127473, pp. 1 - 7 [articolo]Open Access

Rita Morigi, Capitolo 7 - Titolazioni Complessometriche, in: Manuale di Analisi Quantitativa dei Medicinali, Napoli, EdiSES, 2019, pp. 163 - 180 [capitolo di libro]

De Magis, Alessio; Manzo, Stefano G.; Russo, Marco; Marinello, Jessica; Morigi, Rita; Sordet, Olivier; Capranico, Giovanni*, DNA damage and genome instability by G-quadruplex ligands are mediated by R loops in human cancer cells, «PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA», 2019, 116, pp. 816 - 825 [articolo]

Morigi, R., Locatelli, A., Leoni, A., Rambaldi, M., Bortolozzi, R., Mattiuzzo, E., Ronca, R., Maccarinelli, F., Hamel, E., Bai, R., Brancale, A., Viola, G., Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 166, pp. 514 - 530 [articolo]Open Access

Conti, Ilaria; Morigi, Rita; Locatelli, Alessandra*; Rambaldi, Mirella; Bua, Gloria; Gallinella, Giorgio; Leoni, Alberto, Synthesis of 3-(Imidazo[2,1-b]thiazol-6-yl)-2H-chromen-2-one derivatives and study of their antiviral activity against parvovirus B19, «MOLECULES», 2019, 24, Article number: 1037, pp. 1 - 15 [articolo]Open Access

Alessio De Magis, Stefano G. Manzo, Jessica Marinello, Marco Russo, Olivier Sordet, Rita Morigi, Giovanni Capranico, Genome instability by G-quadruplex ligands are mediated by R-loops in human cancer cells, in: BIONIC 2018 - Biology of non-canonical nucleic acids: from humans to pathogens - International Symposium - Abstract Book, 2018, pp. 24 - 24 (atti di: BIONIC 2018 - Biology of non-canonical nucleic acids: from humans to pathogens - International Symposium, Padova, 26-28 settembre 2018) [atti di convegno-abstract]

Morigi, Rita; Vitali, Beatrice; Prata, Cecilia; Palomino, Rogers A. A; Graziadio, Alessandra; Locatelli, Alessandra; Rambaldi, Mirella; Leoni, Alberto, Investigation on the effects of antimicrobial imidazo[2,1-b]thiazole derivatives on the genitourinary microflora, «MEDICINAL CHEMISTRY», 2018, 14, pp. 311 - 319 [articolo]

A. De Magis, S. G. Manzo, M. Russo, J. Marinello, O. Sordet, R. Morigi, G. Capranico., R loop-driven genome instability by G-quadruplex binders in BRCA2-silenced human cancer cells., in: AACR Annual Meeting 2018. Chicago, April 14 - 18, 2018. Abstract Book, «CANCER RESEARCH», 2018, 78, pp. 4838 - 4838 (atti di: AACR Annual Meeting 2018., Chicago, USA, April 14 - 18, 2018) [atti di convegno-poster]

R. Morigi, J. Amato, N. Iaccarino, B. Pagano, A. Locatelli, A. Leoni, M. Rambaldi, G. Miglietta, J. Marinello, G. Capranico, E. Novellino, A. Randazzo, Targeting human telomeric and promoter G-quardruplexes: synthesis, biophysical and biological studies of new guanylhydrazones as potential antitumor agents, in: BIONIC 2018: Biology of non-canonical nucleic acids: from humans to pathogens. 26th - 28th September 2018 - Padova, Italy - Abstract Book, Padova, 2018, pp. 126 - 126 (atti di: BIONIC 2018: Biology of non-canonical nucleic acids: from humans to pathogens., Padova, 26-28 settembre 2018) [atti di convegno-abstract]

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