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Rita Morigi

Professoressa associata

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

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Pubblicazioni antecedenti il 2004

Pubblicazioni antecedenti il 2004

1)                 A. Andreani, A. Locatelli, A. Leoni, M. Rambaldi, R. Morigi, R. Bossa, M. Chiericozzi, A. Fraccari, I. Galatulas.

Synthesis and potential coanthracyclinic activity of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones. Eur. J. Med. Chem. 32, 919-924 (1997).

 

2)                 A. Andreani, A. Leoni, R. Morigi, R. Bossa, M. Chiericozzi, I. Galatulas.

In vivo cardiotonic  activity of aryl- and pyridyl- substituted fused imidazoles. Arzneim.-Forsch./Drug Res. 48 (I), 3, 232-235 (1998).

 

3)         A. Andreani, A. Locatelli, R. Morigi, A. Leoni, R. Bossa, M. Chiericozzi, I. Galatulas.

In vivo cardiotonic activity of pyridylmethylene-2-indolinones. Arzneim.-Forsch./Drug Res. 48 (II), 7, 727-729 (1998).

 

4)         A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Chiericozzi, A. Fraccari, I. Galatulas.

Potential coanthracyclinic activity of pyridylmethylene-2-indolinones. Anticancer Res. 18, 3407-3410 (1998).

 

5)                 A. Andreani, A. Locatelli, A. Leoni, R. Morigi, M. Chiericozzi, A. Fraccari, I. Galatulas, G. Salvatore.

Synthesis and potential coanthracyclinic activity of pyridylmethylene and indolylmethylene lactams. Eur. J. Med. Chem. 33, 905-909, (1998).

 

6)                 A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, J.C. Gehret, S. Traniello, A. Cariani, S. Spisani.

Ring-opened analogs of indomethacin affecting human neutrophil functions. Collect. Czech. Chem. Commun. 64, 299-312, (1999).

 

7)                 A. Andreani, M. Rambaldi, A. Leoni, R. Morigi, A. Locatelli, G. Giorgi, G. Lenaz, A. Ghelli, M. Degli Esposti.

6-Thienyl and 6-phenylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH dehydrogenase. Eur. J. Med. Chem. 34, 883-889, (1999).

 

8)         A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, C. Pietra, G. Villetti.

4-Aminopyridine derivatives with antiamnesic activity. Eur. J. Med. Chem. 35, 77-82, (2000).

 

9)         A. Andreani, M. Rambaldi, A. Leoni, A. Locatelli, R. Morigi, S. Traniello, A. Cariani, O. Rizzuti, S. Spisani.

6-(Hydroxyphenyl)imidazo[2,1-b]thiazoles as potential antiinflammatory agents: effects on human neutrophil functions. Collect. Czech. Chem. Commun. 65, 267-279, (2000).

 

10)             A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, W.A. Simon, J. Senn-Bilfinger.

Synthesis and antisecretory activity of 6-substituted 5-cyanomethylimidazo[2,1-b]thiazoles and 2,6-dimethyl-5-hydroxymethylimidazo[2,1-b][1,3,4]thiadiazole. Arzneim.-Forsch./Drug Res. 50 (I), 6, 550-553, (2000).

 

11)             A. Andreani, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, M. Recanatini, V. Garaliene.

Potential antitumor agents. Part 29. Synthesis and potential coanthracyclinic activity of imidazo[2,1-b]thiazole guanylhydrazones. Bioorg. Med. Chem. 8, 2359-2366, (2000).

 

12)             A. Andreani, A. Cavalli, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, M. Recanatini, M. Garnier, L. Meijer.

Imidazo[2,1-b]thiazolylmethylene- and indolylmethylene-2-indolinones: a new class of cyclin-dependent kinase inhibitors. Design, synthesis and CDK1/cyclin B inhibition. Anti-Cancer Drug Design. 15, 447-452, (2000).

 

13)             A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi.

Synthesis and antitubercular activity of imidazo[2,1-b]thiazoles. Eur. J. Med. Chem. 36, 743-746 (2001).

 

14)             A. Andreani, A. Cavalli, M. Granaiola, M. Guardigli, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, M. Recanatini, A. Roda.

Synthesis and screening for antiacetylcholinesterase activity of (1-benzil-4-oxopiperidin-3-ylidene)methylindoles and –pyrroles related to donezepil. J. Med. Chem. 44, 4011-4014 (2001).

 

15)             A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, G. Giorgi, L. Salvini, V. Garaliene.

Synthesis and antitumor activity of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones. Anti-Cancer Drug Design 16, 167-174 (2001).

 

16)             A. Andreani, M. Granaiola, A. Leoni, A. Locatelli, R. Morigi, M. Rambaldi, V. Garaliene.

Synthesis and antitumor activity of 1,5,6-substituted E-3-(2-chloro-3-indolylmethylene)-1,3-dihydroindol-2-ones. J. Med. Chem. 45, 2666-2669 (2002).

 

17)             A. Andreani, M. Granaiola, A.  Leoni, A. Locatelli, R. Morigi, M. Rambaldi, G. Giorgi, L. Salvini.

Cancer fighting cancer: synthesis of the new heterocyclic system diimidazo[1,2-a:1,2-c]pyrimidine. Arkivoc (XI) 32-38 (2002) (Issue in Honor of Prof. Domenico Spinelli)

http://www.arkat-usa.org/ark/journal/2002/Spinelli/Spinelli_index.htm

 

 

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