Foto del docente

Rita Morigi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Germoglio, Marcello; D'Aria, Federica; Cortone, Giuseppe; Prodomo, Antonello; Mahtab, Mohammad; Morigi, Rita; Amato, Jussara; Pisani, Francesca M; Giancola, Concetta, Effects of hydrazone-based G-quadruplex ligands on FANCJ/BRIP1-depleted cancer cells and a Caenorhabditis elegans dog-1-/- strain, «NAR CANCER», 2025, 7, Article number: zcaf004 , pp. 1 - 15 [Scientific article]

Morigi R.; Zalambani C.; Farruggia G.; Verardi L.; Esposito D.; Leoni A.; Borsetti F.; Voltattorni M.; Zambonin L.; Pincigher L.; Calonghi N.; Locatelli A., Identification of a new bisindolinone arresting IGROV1 cells proliferation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2024, 271, pp. 1 - 19 [Scientific article]Open Access

Morigi, Rita; Esposito, Daniele; Calvaresi, Matteo; Marforio, TAINAH DORINA; Gentilomi, GIOVANNA ANGELA; Bonvicini, Francesca; Locatelli, Alessandra, Isatin Bis-Imidathiazole Hybrids Identified as FtsZ Inhibitors with On-Target Activity Against Staphylococcus aureus, «ANTIBIOTICS», 2024, 13, pp. 1 - 17 [Scientific article]Open Access

Marzano S.; Miglietta G.; Morigi R.; Marinello J.; Arleo A.; Procacci M.; Locatelli A.; Leoni A.; Pagano B.; Randazzo A.; Amato J.; Capranico G., Balancing Affinity, Selectivity, and Cytotoxicity of Hydrazone-Based G-Quadruplex Ligands for Activation of Interferon β Genes in Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 12055 - 12067 [Scientific article]Open Access

Francesca Bonvicini, Alessandra Locatelli, Rita Morigi, Alberto Leoni, Giovanna Angela Gentilomi, Isatin Bis-Indole and Bis-Imidazothiazole Hybrids: Synthesis and Antimicrobial Activity, «MOLECULES», 2022, 27, pp. 5781 - 5792 [Scientific article]Open Access

Das A.; Greco G.; Kumar S.; Catanzaro E.; Morigi R.; Locatelli A.; Schols D.; Alici H.; Tahtaci H.; Ravindran F.; Fimognari C.; Karki S.S., Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives, «COMPUTATIONAL BIOLOGY AND CHEMISTRY», 2022, 97, Article number: 107641 , pp. 1 - 18 [Scientific article]Open Access

Morigi R.; Catanzaro E.; Locatelli A.; Calcabrini C.; Pellicioni V.; Leoni A.; Fimognari C., Synthesis and biological evaluation of new bis-indolinone derivatives endowed with cytotoxic activity, «MOLECULES», 2021, 26, Article number: 6277 , pp. 1 - 15 [Scientific article]Open Access

Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N., Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth, «MOLECULES», 2020, 25, Article number: 4438 , pp. 1 - 15 [Scientific article]Open Access

Amato J.; Miglietta G.; Morigi R.; Iaccarino N.; Locatelli A.; Leoni A.; Novellino E.; Pagano B.; Capranico G.; Randazzo A., Monohydrazone Based G-Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 3090 - 3103 [Scientific article]Open Access

Emanuela Pesce, Nicoletta Pedemonte, Alberto Leoni, Alessandra Locatelli, Rita Morigi, Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis., «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2020, 30, Article number: 127473 , pp. 1 - 7 [Scientific article]Open Access

Rita Morigi, Capitolo 7 - Titolazioni Complessometriche, in: Manuale di Analisi Quantitativa dei Medicinali, Napoli, EdiSES, 2019, pp. 163 - 180 [Chapter or essay]

De Magis, Alessio; Manzo, Stefano G.; Russo, Marco; Marinello, Jessica; Morigi, Rita; Sordet, Olivier; Capranico, Giovanni*, DNA damage and genome instability by G-quadruplex ligands are mediated by R loops in human cancer cells, «PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA», 2019, 116, pp. 816 - 825 [Scientific article]

Conti, Ilaria; Morigi, Rita; Locatelli, Alessandra*; Rambaldi, Mirella; Bua, Gloria; Gallinella, Giorgio; Leoni, Alberto, Synthesis of 3-(Imidazo[2,1-b]thiazol-6-yl)-2H-chromen-2-one derivatives and study of their antiviral activity against parvovirus B19, «MOLECULES», 2019, 24, Article number: 1037 , pp. 1 - 15 [Scientific article]Open Access

Morigi, R., Locatelli, A., Leoni, A., Rambaldi, M., Bortolozzi, R., Mattiuzzo, E., Ronca, R., Maccarinelli, F., Hamel, E., Bai, R., Brancale, A., Viola, G., Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 166, pp. 514 - 530 [Scientific article]Open Access

Alessio De Magis, Stefano G. Manzo, Jessica Marinello, Marco Russo, Olivier Sordet, Rita Morigi, Giovanni Capranico, Genome instability by G-quadruplex ligands are mediated by R-loops in human cancer cells, in: BIONIC 2018 - Biology of non-canonical nucleic acids: from humans to pathogens - International Symposium - Abstract Book, 2018, pp. 24 - 24 (atti di: BIONIC 2018 - Biology of non-canonical nucleic acids: from humans to pathogens - International Symposium, Padova, 26-28 settembre 2018) [Abstract]

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