Foto del docente

Vincenza Andrisano

Full Professor

Department for Life Quality Studies

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Director of Single Cycle Degree in Pharmacy

Publications

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Prati F;De Simone A;Bisignano P;Armirotti A;Summa M;Pizzirani D;Scarpelli R;Perez DI;Andrisano V;Perez-Castillo A;Monti B;Massenzio F;Polito L;Racchi M;Favia AD;Bottegoni G;Martinez A;Bolognesi ML;Cavalli A, Multitarget drug discovery for Alzheimer's disease: triazinones as BACE-1 and GSK-3β inhibitors., «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2015, 54, pp. 1578 - 1582 [Scientific article]

Bartolini, Manuela; Naldi, Marina; Andrisano, Vincenza, New analytical tools to investigate the role of protein glycosylation in Alzheimer’s disease, in: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, 2015, pp. 167 - 167 (atti di: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, Barcelona Biomedical Research Park, Barcellona, Spagna, July 12-15 2015) [Poster]

Benchekroun, M.; Bartolini, M.; Egea, J.; Romero, A.; Soriano, E.; Pudlo, M.; Luzet, V.; Andrisano, V.; Jimeno, M.-L.; Lopez, M.G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; De Andres, L.; Herrera-Arozamena, C.; Monti, B.; Bolognesi, M.L.; Rodriguez-Franco, M.I.; Decker, M.; Marco-Contelles, J.; Ismaili, L., Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids, «CHEMMEDCHEM», 2015, 10, pp. 523 - 539 [Scientific article]

Bartolini, M.; Naldi, M.; Andrisano, V., ON-LINE GLYCAN RELEASE AND ANALYSIS BY AN INTEGRATED PNGASE F-IMER LC-ESI-Q-TOF APPROACH, in: IMASS PHARMA NETWORK 2015 Book of Abstracts, 2015, pp. 10 - 10 (atti di: IMASS PHARMA NETWORK 2015, Verona, Italia, 26-28 ottobre 2015) [Contribution to conference proceedings]

Bartolini, M.; Naldi, M.; Andrisano, V., PROTEIN GLYCOSILATION ANALYSIS BY AN INTEGRATED PNGASE-F-IMER-LC-ESI-Q-TOF APPROACH, in: Abstract Book - RDPA 2015, 2015, pp. 26 - 26 (atti di: RDPA 2015 - Recent Developments in Pharmaceutical Analysis, Perugia, June 28 - July 1, 2015) [Contribution to conference proceedings]

Prati, Federica; De Simone, Angela; Armirotti, Andrea; Summa, Maria; Pizzirani, Daniela; Scarpelli, Rita; Bertozzi, Sine Mandrup; Perez, Daniel I.; Andrisano, Vincenza; Perez-Castillo, Ana; Monti, Barbara; Massenzio, Francesca; Polito, Letizia; Racchi, Marco; Sabatino, Piera; Bottegoni, Giovanni; Martinez, Ana; Cavalli, Andrea; Bolognesi, Maria L., 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the First Dual BACE-1/GSK-3β Fragment Hits against Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2015, 6, pp. 1665 - 1682 [Scientific article]Open Access

Gurjar AS; Andrisano V; De Simone A; Velingkar VS, Design, synthesis, in silico and in vitro screening of 1,2,4-thiadiazole analogues as non-peptide inhibitors of beta-secretase., «BIOORGANIC CHEMISTRY», 2014, 57, pp. 90 - 98 [Scientific article]

Carlo Bertucci; Daniele Tedesco; Edoardo Fabini; Anna Maria Di Pietra; Francesca Rossi; Marco Garagnani; Elia Del Borrello; Vincenza Andrisano, Determination of levamisole and tetramisole in seized cocaine samples by enantioselective high-performance liquid chromatography and circular dichroism detection, «JOURNAL OF CHROMATOGRAPHY A», 2014, 1363, pp. 150 - 154 [Scientific article]

Simone Brogi; Stefania Butini; Samuele Maramai; Raffaella Colombo; Laura Verga; Cristina Lanni; Ersilia De Lorenzi; Stefania Lamponi; Marco Andreassi; Manuela Bartolini; Vincenza Andrisano; Ettore Novellino; Giuseppe Campiani; Margherita Brindisi; Sandra Gemma, Disease-Modifying Anti-Alzheimer's Drugs: Inhibitors of Human Cholinesterases Interfering with β-Amyloid Aggregation, «CNS NEUROSCIENCE & THERAPEUTICS», 2014, 20, pp. 624 - 632 [Scientific article]

D’Urzo, A.; De Simone, A.; Fiori, J.; Andrisano, V., ESI-MS and UHPLC combined analytical approaches for determining the kinetics of Glycogen Synthase Kinase-3β, in: Nuove Prospettive in Chimica Farmaceutica 8, 2014(atti di: Nuove Prospettive in Chimica Farmaceutica 8, Parma, 9-11 Giugno) [Poster]

Belluti F.; De Simone A.; Tarozzi A.; Bartolini M.; Djemil A.; Bisi A.; Gobbi S.; Montanari S.; Cavalli A.; Andrisano V.; Bottegoni G.; Rampa A., Fluorinated benzophenone derivatives: balanced multipotent agents for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2014, 78, pp. 157 - 166 [Scientific article]

Tarozzi A.; Bartolini M.; Piazzi L.; Valgimigli L.; Amorati R.; Bolondi C.; Djemil A.; Mancini F.; Andrisano V.; Rampa A., From the dual function lead AP2238 to AP2469, a multi-target-directed ligand for the treatment of Alzheimer’s disease, «PHARMACOLOGY RESEARCH & PERSPECTIVES», 2014, 2, Article number: e00023 , pp. 1 - 14 [Scientific article]Open Access

Jessica Fiori; Vincenza andrisano, LC–MS method for the simultaneous determination of six glucocorticoids in pharmaceutical formulations and counterfeit cosmetic products, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2014, 91, pp. 185 - 192 [Scientific article]

Angela De Simone; Claudia Seidl; Cid A. Santos; Vincenza Andrisano, Liquid chromatographic enzymatic studies with on-line Beta-secretase immobilized enzyme reactor and 4-(4-dimethylaminophenylazo) benzoic acid/5-[(2-aminoethyl) amino] naphthalene-1-sulfonic acid as fluorogenic substrate, «JOURNAL OF CHROMATOGRAPHY B», 2014, 953-954, pp. 108 - 114 [Scientific article]