Foto del docente

Vincenza Andrisano

Full Professor

Department for Life Quality Studies

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Director of Single Cycle Degree in Pharmacy

Publications

Ismaili L.; Monnin J.; Etievant A.; Arribas R.L.; Viejo L.; Refouvelet B.; Soukup O.; Janockova J.; Hepnarova V.; Korabecny J.; Kucera T.; Jun D.; Andrys R.; Musilek K.; Baguet A.; Garcia-Frutos E.M.; De Simone A.; Andrisano V.; Bartolini M.; De Los Rios C.; Marco-Contelles J.; Haffen E., (±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2021, 12, pp. 1328 - 1342 [Scientific article]

Naldi M.; Brusotti G.; Massolini G.; Andrisano V.; Temporini C.; Bartolini M., Bio-guided fractionation of stem bark extracts from phyllanthus muellarianus: Identification of phytocomponents with anti-cholinesterase activity, «MOLECULES», 2021, 26, Article number: 4376 , pp. 4376-1 - 4376-14 [Scientific article]Open Access

De Simone A.; Davani L.; Montanari S.; Tumiatti V.; Avanessian S.; Testi F.; Andrisano V., Combined Methodologies for Determining In Vitro Bioavailability of Drugs and Prediction of In Vivo Bioequivalence From Pharmaceutical Oral Formulations, «FRONTIERS IN CHEMISTRY», 2021, 9, Article number: 741876 , pp. 1 - 13 [Scientific article]

Montanari S.; Davani L.; Tumiatti V.; Dimilta M.; Gaddi A.V.; De Simone A.; Andrisano V., Development of an UHPLC-diode arrays detector (DAD) method for the analysis of polydatin in human plasma, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2021, 198, Article number: 113985 , pp. 1 - 7 [Scientific article]

Viayna, Elisabet; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Cisternas, Pedro; Oliva, Carolina A.; Sánchez-López, Elena; Ettcheto, Miren; Bartolini, Manuela; De Simone, Angela; Ricchini, Mattia; Rendina, Marisa; Pons, Mégane; Firuzi, Omidreza; Pérez, Belén; Saso, Luciano; Andrisano, Vincenza; Nachon, Florian; Brazzolotto, Xavier; García, Maria Luisa; Camins, Antoni; Silman, Israel; Jean, Ludovic; Inestrosa, Nibaldo C.; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero, Diego, Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 Mice, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 812 - 839 [Scientific article]

Pont C.; Ginex T.; Grinan-Ferre C.; Scheiner M.; Mattellone A.; Martinez N.; Arce E.M.; Soriano-Fernandez Y.; Naldi M.; De Simone A.; Barenys M.; Gomez-Catalan J.; Perez B.; Sabate R.; Andrisano V.; Loza M.I.; Brea J.; Bartolini M.; Bolognesi M.L.; Decker M.; Pallas M.; Luque F.J.; Munoz-Torrero D., From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2021, 225, Article number: 113779 , pp. 1 - 25 [Scientific article]

Angela De Simone, Vincenzo Tumiatti, VIncenza Andrisano, Andrea Milelli, Glycogen Synthase Kinase 3β: A New Gold Rush in Anti-Alzheimer’s Disease Multitarget Drug Discovery?, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 26 - 41 [Scientific article]Open Access

Glicerina V, Siroli L, Ticchi N, Capelli F, Accorsi R, Gherardi M, Fiorini M, Andrisano V, Colombo V, Manzini R, Lanciotti R, Romani S, INFLUENCE OF AN INNOVATIVE, BIODEGRADABLE MULTILAYER ACTIVE PACKAGING ON “PESTO” SAUCE CHARACTERISTICS DURING STORAGE, in: Giancarlo Colelli E Milena Corredig, FIRST CIRCUL-A-BILITY CONFERENCE Re-thinking Packaging for Circular & Sustainable Food Supply Chains of the Future-Book of Abstract, 2021, pp. 1 - 63 (atti di: FIRST CIRCUL-A-BILITY CONFERENCE Re-thinking Packaging for Circular & Sustainable Food Supply Chains of the Future, Online, 26-29 Settembre 2021) [Contribution to conference proceedings]

De Simone A.; Naldi M.; Tedesco D.; Bartolini M.; Davani L.; Andrisano V., Advanced analytical methodologies in Alzheimer's disease drug discovery, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2020, 178, Article number: 112899 , pp. 1 - 25 [Scientific article]

Pérez-Areales, F Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer, Angel; Muñoz-Torrero, Diego, Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 9360 - 9390 [Scientific article]

Rozálie Peřinová , Negar Maafia , Jan Korábečný, , Eliška Kohelová , Angela De Simone , Abdullah Al Mamuna , Daniela Hulcováa, , Jana Markováa , Tomáš Kučera , Daniel Jun, Marcela Šafratová , Jana Maříková, Vincenza Andrisano, , Jaroslav Jenčoa , Jiří Kunešf , Ana Martinezg , Lucie Novákováh , Lucie Cahlíkováa,, Functionalized aromatic esters of the Amaryllidaceae alkaloid haemanthamine and their in vitro and in silico biological activity connected to Alzheimer's disease, «BIOORGANIC CHEMISTRY», 2020, 100, Article number: 103928 , pp. 1 - 10 [Scientific article]

Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N., Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth, «MOLECULES», 2020, 25, Article number: 4438 , pp. 1 - 15 [Scientific article]Open Access

Catanzaro E.; Betari N.; Arencibia J.M.; Montanari S.; Sissi C.; De Simone A.; Vassura I.; Santini A.; Andrisano V.; Tumiatti V.; De Vivo M.; Krysko D.V.; Rocchi M.B.L.; Fimognari C.; Milelli A., Targeting topoisomerase II with trypthantrin derivatives: Discovery of 7-((2-(dimethylamino)ethyl)amino)indolo[2,1-b]quinazoline-6,12-dione as an antiproliferative agent and to treat cancer, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2020, 202, Article number: 112504 , pp. 112504 - 112504 [Scientific article]

Perez-Areales F.J.; Turcu A.L.; Barniol-Xicota M.; Pont C.; Pivetta D.; Espargaro A.; Bartolini M.; De Simone A.; Andrisano V.; Perez B.; Sabate R.; Sureda F.X.; Vazquez S.; Munoz-Torrero D., A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 180, pp. 613 - 626 [Scientific article]

Hulcova D.; Marikova J.; Korabecny J.; Hostalkova A.; Jun D.; Kunes J.; Chlebek J.; Opletal L.; De Simone A.; Novakova L.; Andrisano V.; Ruzicka A.; Cahlikova L., Amaryllidaceae alkaloids from Narcissus pseudonarcissus L. cv. Dutch Master as potential drugs in treatment of Alzheimer's disease, «PHYTOCHEMISTRY», 2019, 165, Article number: 112055 , pp. 112055 - 112063 [Scientific article]