Foto del docente

Vincenza Andrisano

Full Professor

Department for Life Quality Studies

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Director of Single Cycle Degree in Pharmacy

Publications

Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [Scientific article]Open Access

Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela, Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease, «CHEMMEDCHEM», 2016, 11, pp. 1309 - 1317 [Scientific article]Open Access

Wang, C.H.; Alluri, S.; Nikogosyan, G.; Decarlo, C.; Monteiro, C.; Mabagos, G.; Feng, H.H.; White, A.R.; Bartolini, M.; Andrisano, V.; Zhang, L.K.; Ganguly, A.K, Novel synthesis of physovenine and physostigmine analogs, «TETRAHEDRON LETTERS», 2016, 57, pp. 3046 - 3049 [Scientific article]

Zha, Xiaoming; Lamba, Doriano; Zhang, Lili; Lou, Yinghan; Xu, Changxu; Kang, Di; Chen, Li; Xu, Yungen; Zhang, Luyong; De Simone, Angela; Samez, Sarah; Pesaresi, Alessandro; Stojan, Jure; Lopez, Manuela G.; Egea, Javier; Andrisano, Vincenza; Bartolini, Manuela, Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimers Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 114 - 131 [Scientific article]Open Access

Prati, Federica; Bergamini, Christian; Fato, Romana; Soukup, Ondrej; Korabecny, Jan; Andrisano, Vincenza; Bartolini, Manuela; Bolognesi, Maria Laura, Novel 8-Hydroxyquinoline Derivatives as Multitarget Compounds for the Treatment of Alzheimer's Disease, «CHEMMEDCHEM», 2016, 11, pp. 1284 - 1295 [Scientific article]

Simoni, Elena; Caporaso, Roberta; Bergamini, Christian; Fiori, Jessica; Fato, Romana; Miszta, Przemyslaw; Filipek, Sławomir; Caraci, Filippo; Giuffrida, Maria Laura; Andrisano, Vincenza; Minarini, Anna; Bartolini, Manuela; Rosini, Michela, Polyamine Conjugation as a Promising Strategy To Target Amyloid Aggregation in the Framework of Alzheimer’s Disease, «ACS MEDICINAL CHEMISTRY LETTERS», 2016, 7, pp. 1145 - 1150 [Scientific article]

D'Urzo, A; Boichenko, Ap; van den Bosch, T; Hermans, J; Dekker, F; Andrisano, V; Bischoff, R., Site-specific quantification of lysine acetylation in the N-terminal tail of histone H4 using a double-labelling, targeted UHPLC MS/MS approach., «ANALYTICAL AND BIOANALYTICAL CHEMISTRY», 2016, 408, pp. 3547 - 3553 [Scientific article]

Fiori, J; De Simone, A; Naldi, M; Andrisano, V, The role of Chromatography in Alzheimer’s Disease Drug Discovery., in: Advances in Chromatography, United Kingdom, Taylor & Francis Group, 2016, pp. 75 - 107 (ADVANCES IN CHROMATOGRAPHY) [Chapter or essay]

Di Martino, Rita Maria Concetta; De Simone, Angela; Andrisano, Vincenza; Bisignano, Paola; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Fato, Romana; Bergamini, Christian; Perez, Daniel I.; Martinez, Ana; Bottegoni, Giovanni; Cavalli, Andrea; Belluti, Federica, Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 531 - 544 [Scientific article]Open Access

De Simone, Angela; Bartolini, Manuela; Fiori, Jessica; D’Urzo, Annalisa; Naldi, Marina.; Andrisano, Vincenza, Analytical approaches in Alzheimer’s disease Drug Discovery, in: SIMCC 2015 - Spanish-Italian Medicinal Chemistry Congress - Book of Abstracts, 2015, pp. 35 - 35 (atti di: SIMCC 2015 - Spanish-Italian Medicinal Chemistry Congress, BARCELONA (SPAIN), JULY 12-15, 2015) [Contribution to conference proceedings]

De Simone, A.; Andrisano, V., Characterization of essential oil components in cosmetic products by GC-MS., in: 8°MS PHARMA DAY, 2015(atti di: 8°MS PHARMA DAY, San Sepolcro (AR), 11-13 Giugno) [Poster]

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Prati F;De Simone A;Bisignano P;Armirotti A;Summa M;Pizzirani D;Scarpelli R;Perez DI;Andrisano V;Perez-Castillo A;Monti B;Massenzio F;Polito L;Racchi M;Favia AD;Bottegoni G;Martinez A;Bolognesi ML;Cavalli A, Multitarget drug discovery for Alzheimer's disease: triazinones as BACE-1 and GSK-3β inhibitors., «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2015, 54, pp. 1578 - 1582 [Scientific article]

Bartolini, Manuela; Naldi, Marina; Andrisano, Vincenza, New analytical tools to investigate the role of protein glycosylation in Alzheimer’s disease, in: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, 2015, pp. 167 - 167 (atti di: SIMCC 2015 - Spanish - Italian medicinal chemistry congress, Barcelona Biomedical Research Park, Barcellona, Spagna, July 12-15 2015) [Poster]

Benchekroun, M.; Bartolini, M.; Egea, J.; Romero, A.; Soriano, E.; Pudlo, M.; Luzet, V.; Andrisano, V.; Jimeno, M.-L.; Lopez, M.G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; De Andres, L.; Herrera-Arozamena, C.; Monti, B.; Bolognesi, M.L.; Rodriguez-Franco, M.I.; Decker, M.; Marco-Contelles, J.; Ismaili, L., Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids, «CHEMMEDCHEM», 2015, 10, pp. 523 - 539 [Scientific article]