De Simone, A; Milelli, A; Naldi, M; Andrisano, V., Application of an ESI-MS method enabling the discovery of new non-ATP competitive GSK-3beta inhibitors., in: XXIV National Meeting in Medicinal Chemistry., 2016(atti di: XXIV National Meeting in Medicinal Chemistry., Perugia, Italia., 11-14 Settembre 2016.) [atti di convegno-poster]
Chlebek, Jakub; De Simone, Angela; Hoš͗álková, Anna; Opletal, Lubomír; Pérez, Concepción; Pérez, Daniel I.; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenza, Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targets, «FITOTERAPIA», 2016, 109, pp. 241 - 247 [articolo]
De Simone, A; Naldi, M; Milelli, A; Andrisano, V, Application of ESI-MS method for detailed characterization of GSK-3β inhibitors by monitoring GSM peptide phosphorylation.Angelini Farmaceutici., in: 9° MS-PHARMA DAY, 2016, pp. 35 - 37 (atti di: 9° MS-PHARMA DAY., S. Palomba. Roma, 25-27 Maggio 2016.) [Contributo in Atti di convegno]
Lemes, Laís Flávia Nunes; De Andrade Ramos, Giselle; De Oliveira, Andressa Souza; Da Silva, Fernanda Motta R.; De Castro Couto, Gina; Da Silva Boni, Marina; Guimarães, Marcos Jorge R.; Souza, Isis Nem O.; Bartolini, Manuela; Andrisano, Vincenza; Do Nascimento Nogueira, Patrícia Coelho; Silveira, Edilberto Rocha; Brand, Guilherme D.; Soukup, Ondřej; Korábečný, Jan; Romeiro, Nelilma C.; Castro, Newton G.; Bolognesi, Maria Laura; Romeiro, Luiz Antonio Soares, Cardanol-derived AChE inhibitors: Towards the development of dual binding derivatives for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 108, pp. 687 - 700 [articolo]
Pérez-Areales JF; Bartolini M; De Simone A; Espergaro A; Sabaté R; Pérez B; Andrisano V; Luque FJ; Messeguer A; Munoz-Torrero D., Design, Synthesis and Biological profiling of a promising new family of multitarget directed ligands for the treatment of Alzheimer Disease., in: III Symposium of Young Researchers of the Spanish Society of Medicinal Chemistry., 2016(atti di: III Symposium of Young Researchers of the Spanish Society of Medicinal Chemistry., Barcellona, Spagna., 17 Giugno) [atti di convegno-poster]
D'Urzo, Annalisa; DE SIMONE, Angela; Fiori, Jessica; Naldi, Marina; Milelli, Andrea; Andrisano, Vincenza, Direct determination of GSK-3β activity and inhibition by UHPLC-UV-vis diode arrays detector (DAD), «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2016, 124, pp. 104 - 111 [articolo]
Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela, Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 6387 - 6406 [articolo]Open Access
Boulebd, Houssem; Ismaili, Lhassane; Bartolini, Manuela; Bouraiou, Abdelmalek; Andrisano, Vincenza; Martin, Helene; Bonet, Alexandre; Moraleda, Ignacio; Iriepa, Isabel; Chioua, Mourad; Belfaitah, Ali; Marco-Contelles, José, Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease Therapy, «MOLECULES», 2016, 21, Article number: 400, pp. 1 - 16 [articolo]Open Access
Chlebek, J; De Simone, A; Pérez, Di; Pérez, C; Havlíková, L; Hošťálková, A; Opletal, L; Cahlíková, L; Andrisano, V, Multifunctional activity of some isoquinoline alkaloids from Corydalis cava tubers on Alzheimer's disease targets, «PLANTA MEDICA», 2016, 81, pp. S1 - S381 [articolo]
Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [articolo]Open Access
Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela, Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease, «CHEMMEDCHEM», 2016, 11, pp. 1309 - 1317 [articolo]Open Access
Wang, C.H.; Alluri, S.; Nikogosyan, G.; Decarlo, C.; Monteiro, C.; Mabagos, G.; Feng, H.H.; White, A.R.; Bartolini, M.; Andrisano, V.; Zhang, L.K.; Ganguly, A.K, Novel synthesis of physovenine and physostigmine analogs, «TETRAHEDRON LETTERS», 2016, 57, pp. 3046 - 3049 [articolo]
Zha, Xiaoming; Lamba, Doriano; Zhang, Lili; Lou, Yinghan; Xu, Changxu; Kang, Di; Chen, Li; Xu, Yungen; Zhang, Luyong; De Simone, Angela; Samez, Sarah; Pesaresi, Alessandro; Stojan, Jure; Lopez, Manuela G.; Egea, Javier; Andrisano, Vincenza; Bartolini, Manuela, Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimers Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 114 - 131 [articolo]Open Access
Prati, Federica; Bergamini, Christian; Fato, Romana; Soukup, Ondrej; Korabecny, Jan; Andrisano, Vincenza; Bartolini, Manuela; Bolognesi, Maria Laura, Novel 8-Hydroxyquinoline Derivatives as Multitarget Compounds for the Treatment of Alzheimer's Disease, «CHEMMEDCHEM», 2016, 11, pp. 1284 - 1295 [articolo]
Simoni, Elena; Caporaso, Roberta; Bergamini, Christian; Fiori, Jessica; Fato, Romana; Miszta, Przemyslaw; Filipek, Sławomir; Caraci, Filippo; Giuffrida, Maria Laura; Andrisano, Vincenza; Minarini, Anna; Bartolini, Manuela; Rosini, Michela, Polyamine Conjugation as a Promising Strategy To Target Amyloid Aggregation in the Framework of Alzheimer’s Disease, «ACS MEDICINAL CHEMISTRY LETTERS», 2016, 7, pp. 1145 - 1150 [articolo]