Foto del docente

Luca Gentilucci

Associate Professor

Department of Chemistry "Giacomo Ciamician"

Academic discipline: CHIM/06 Organic Chemistry


He, Tingting; Giacomini, Daria; Tolomelli, Alessandra; Baiula, Monica; Gentilucci, Luca, Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic Applications, «BIOMEDICINES», 2024, 12, pp. 1 - 22 [Scientific article]

He T.; Valagussa B.; Boanini E.; Gentilucci L., Expedient recycling of peptide organocatalysts using a nanocrystalline hydroxyapatite catching system, «SUSTAINABLE CHEMISTRY AND PHARMACY», 2024, 37, pp. 1 - 10 [Scientific article]

Anselmi, Michele; Baiula, Monica; Spampinato, Santi; Artali, Roberto; He, Tingting; Gentilucci, Luca, Design and Pharmacological Characterization of α4β1 Integrin Cyclopeptide Agonists: Computational Investigation of Ligand Determinants for Agonism versus Antagonism, «JOURNAL OF MEDICINAL CHEMISTRY», 2023, 66, pp. 5021 - 5040 [Scientific article]Open Access

Santino, Federica; Gentilucci, Luca, Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects, «MOLECULES», 2023, 28, pp. 1 - 22 [Scientific article]Open Access

Baiula, Monica; Anselmi, Michele; Musiani, Francesco; Ghidini, Alessia; Carbone, Jacopo; Caligiana, Alberto; Maurizio, Andrea; Spampinato, Santi; Gentilucci, Luca, Design, Pharmacological Characterization, and Molecular Docking of Minimalist Peptidomimetic Antagonists of α4β1 Integrin, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2023, 24, pp. 1 - 22 [Scientific article]Open Access

Zhao, Junwei; Carbone, Jacopo; Farruggia, Giovanna; Janecka, Anna; Gentilucci, Luca; Calonghi, Natalia, Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives, «MOLECULES», 2023, 28, pp. 1 - 17 [Scientific article]Open Access

Carbone, Jacopo; Ghidini, Alessia; Romano, Antonio; Gentilucci, Luca; Musiani, Francesco, PacDOCK: A Web Server for Positional Distance-Based and Interaction-Based Analysis of Docking Results, «MOLECULES», 2022, 27, Article number: 6884 , pp. 1 - 12 [Scientific article]Open Access

Federica Santino; Pasquale Stavole; Tingting He; Silvia Pieraccini; Mayra Paolillo; Luca Prodi; Enrico Rampazzo; Luca Gentilucci, Preparation of Non-Toxic Fluorescent Peptide-Coated Silica/PEG Nanoparticles from Peptide-Block Copolymer Conjugates, «MICRO», 2022, 2, pp. 240 - 256 [Scientific article]Open Access

Wtorek, Karol; Ghidini, Alessia; Gentilucci, Luca; Adamska-Bartłomiejczyk, Anna; Piekielna-Ciesielska, Justyna; Ruzza, Chiara; Sturaro, Chiara; Calò, Girolamo; Pieretti, Stefano; Kluczyk, Alicja; McDonald, John; Lambert, David G; Janecka, Anna, Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2022, 23, pp. 12700 - 12718 [Scientific article]Open Access

Anselmi M.; Baiula M.; Santino F.; Zhao J.; Spampinato S.; Calonghi N.; Gentilucci L., Design of α/β-hybrid peptide ligands of α4β1 integrin equipped with a linkable side chain for chemoselective biofunctionalization of microstructured materials, «BIOMEDICINES», 2021, 9, Article number: 1737 , pp. 1 - 21 [Scientific article]Open Access

Baiula, Monica; Caligiana, Alberto; Bedini, Andrea; Zhao, Junwei; Santino, Federica; Cirillo, Martina; Gentilucci, Luca; Giacomini, Daria; Spampinato, Santi, Leukocyte Integrin Antagonists as a Novel Option to Treat Dry Age-Related Macular Degeneration, «FRONTIERS IN PHARMACOLOGY», 2021, 11, Article number: 617836 , pp. 1 - 13 [Scientific article]Open Access

Anselmi M.; Borbely A.; Figueras E.; Michalek C.; Kemker I.; Gentilucci L.; Sewald N., Linker Hydrophilicity Modulates the Anticancer Activity of RGD–Cryptophycin Conjugates, «CHEMISTRY-A EUROPEAN JOURNAL», 2021, 27, Article number: 3471 , pp. 1015 - 1022 [Scientific article]Open Access

Santino F.; Petruzzelli R.; Zhao J.; Boanini E.; Gentilucci L., Peptide bond formation using unprotected N-carboxyanhydrides under green chemistry conditions, «SUSTAINABLE CHEMISTRY AND PHARMACY», 2021, 24, Article number: 100540 , pp. 1 - 8 [Scientific article]Open Access

Piekielna-Ciesielska, Justyna; Artali, Roberto; Azzam, Ammar A H; Lambert, David G; Kluczyk, Alicja; Gentilucci, Luca; Janecka, Anna, Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation, «MOLECULES», 2021, 26, Article number: 13 , pp. 1 - 20 [Scientific article]Open Access

Bedini A.; Di Cesare Mannelli L.; Micheli L.; Baiula M.; Vaca G.; De Marco R.; Gentilucci L.; Ghelardini C.; Spampinato S., Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist, «FRONTIERS IN PHARMACOLOGY», 2020, 11, Article number: 188 , pp. 1 - 22 [Scientific article]Open Access