Foto del docente

Luca Gentilucci

Associate Professor

Department of Chemistry "Giacomo Ciamician"

Academic discipline: CHIM/06 Organic Chemistry

Publications

Piekielna, J.; Gentilucci, L.; De Marco, R.; Perlikowska, R.; Adamska, A.; Olczak, J.; Mazur, M.; Artali, R.; Modranka, J.; Janecki, T.; Tomboly, C.; Janecka, A., Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine, «BIOORGANIC & MEDICINAL CHEMISTRY», 2014, 22, pp. 6545 - 6551 [Scientific article]

Tolomelli, Alessandra; Gentilucci, Luca; Viola, Angelo; Dattoli, Samantha Deianira; Baiula, Monica; Spampinato, Santi; Petkau-Milroy, Katja; Brunsveld, Luc, Design and synthesis of Alpha-v-beta-3 and Alpha-5-beta-1 integrin ligands as delivery systems for fluorescent molecules, «LA CHIMICA E L'INDUSTRIA», 2014, 96, pp. 56 - 58 [Scientific article]

A. Tolomelli; L. Gentilucci; A. Viola; S. D. Dattoli; M. Baiula; S. Spampinato; L. Belvisi; M.Civera, Design, synthesis and in vitro evaluation of tumor homing agents by conjugation of integrin ligands to diagnostics and cytotoxic drugs, in: 15th Tetrahedron Symposium Book of abstract, London, Elsevier, 2014, /, pp. / - / (atti di: 15th Tetrahedron Symposium Chellenges in Bioorganic and Organic Medicinal Chemistry, Londra, 24-27 Giugno 2014) [Abstract]

De Marco, R.; Cavina, L.; Greco, A.; Gentilucci, L., Easy preparation of dehydroalanine building blocks equipped with oxazolidin-2-one chiral auxiliaries, and applications to the stereoselective synthesis of substituted tryptophans, «AMINO ACIDS», 2014, 46, pp. 2823 - 2839 [Scientific article]

R. De Marco; A. Greco; L. Gentilucci, Hybrid alfa/beta-dipeptide scaffolds as inductors of constrained conformations, in: Abstract Book, Paris, European Peptide Society, 2014, pp. 69 - 69 (atti di: PIPS 2014, Gennevilliers, 05 10 2014) [Contribution to conference proceedings]

De Marco, Rossella; Ricci, Giampaolo; Schinelli, Sergio; Cola, Luisa De; Prodi, Luca; Gentilucci, Luca, Nanostructured Materials for the Detection of Markers of Asthma and Other Correlated Inflammatory Diseases, «ERN. EUROPEAN RESPIRATORY NEWS», 2014, 22, pp. 142 - 143 [Scientific article]

Arianna Greco; Sara Tani; Rossella De Marco; Luca Gentilucci, Synthesis and Analysis of the Conformational Preferences of 5- Aminomethyloxazolidine-2,4-dione Scaffolds: First Examples of beta2- and beta2,2-Homo-Freidinger Lactam Analogues, «CHEMISTRY-A EUROPEAN JOURNAL», 2014, 20, pp. 13390 - 13404 [Scientific article]

S. D. Dattoli ; R. De Marco; M. Baiula; S. Spampinato; A. Greco; A. Tolomelli; L. Gentilucci, Synthesis and assay of retro-α4β1 integrin-targeting motifs, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2014, 73, pp. 225 - 232 [Scientific article]

R. De Marco; A. Greco; L. Comellini; L. Caliò; L. Gentilucci, Synthesis of beta2- and beta2,2-homo-Freidinger Lactam analogs, conformational analysis, and applications in Medicinal Chemistry, in: Conference Programme, Windsor, Royal Soc of Chemistry - SCI, 2014, pp. 44 - 44 (atti di: 14th Anglo Italian Meeting Heterocyclic Chemistry, Windsor, 29 06 2014) [Contribution to conference proceedings]

De Marco R; Bedini A; Spampinato S; Gentilucci L, Synthesis of tripeptides containing D-Trp substituted at indole ring, and assessment of MOR affinity and in vivo central antinociception., «JOURNAL OF MEDICINAL CHEMISTRY», 2014, 57, pp. 6861 - 6866 [Scientific article]

R. De Marco; R. Artali; S. Spampinato; A. Bedini; L. Gentilucci, TRYptophan-COntaining Non-Cationizable Opioid PeptideS (TRYCONCOPS): A new paradigm for opioid peptides, in: Abstract Book, Paris, Eupean peptide Society, 2014, pp. 26 - 26 (atti di: PIPS 2014, Gennevilliers, 05 10 2014) [Contribution to conference proceedings]

Paola Galletti;Roberto Soldati;Matteo Pori;Margherita Durso;Alessandra Tolomelli;Luca Gentilucci;Samantha Deianira Dattoli;Monica Baiula;Santi Spampinato;Daria Giacomini, Targeting integrins αvβ3 and α5β1 with new β-lactam derivatives, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2014, 83, pp. 284 - 293 [Scientific article]

De Marco R; Tolomelli A; Greco A; Gentilucci L, Controlled solid phase peptide bond formation using N-carboxyanhydrides and PEG resins in water., «ACS SUSTAINABLE CHEMISTRY & ENGINEERING», 2013, 1, pp. 566 - 569 [Scientific article]

De Marco R; Greco A; Rupiani S; Tolomelli A; Tomasini C; Pieraccini S; Gentilucci L, In-peptide synthesis of di-oxazolidinone and dehydroamino acid-oxazolidinone motifs as β-turn inducers, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2013, 11, pp. 4316 - 4326 [Scientific article]

Coordination of a Research Project: Inibitori dei processi infiammatori cronici connessi allo sviluppo di tumori (Inhibitors of the chronic inflammatory processes connected to tumor development).