Foto del docente

Luca Gentilucci

Professore associato confermato

Dipartimento di Chimica "Giacomo Ciamician"

Settore scientifico disciplinare: CHIM/06 CHIMICA ORGANICA

Pubblicazioni

Bedini A.; Di Cesare Mannelli L.; Micheli L.; Baiula M.; Vaca G.; De Marco R.; Gentilucci L.; Ghelardini C.; Spampinato S., Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist, «FRONTIERS IN PHARMACOLOGY», 2020, 11, pp. 1 - 22 [articolo]Open Access

Anselmi M.; Stavole P.; Boanini E.; Bigi A.; Juaristi E.; Gentilucci L., Green synthesis of bioactive oligopeptides promoted by recyclable nanocrystalline hydroxyapatite, «FUTURE MEDICINAL CHEMISTRY», 2020, 12, pp. 479 - 491 [articolo]

Stefan A.; Gentilucci L.; Piaz F.D.; D'Alessio F.; Santino F.; Hochkoeppler A., Purification from Deinococcus radiodurans of a 66 kDa ABC transporter acting on peptides containing at least 3 amino acids, «BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS», 2020, 529, pp. 869 - 875 [articolo]

Martelli G.; Baiula M.; Caligiana A.; Galletti P.; Gentilucci L.; Artali R.; Spampinato S.; Giacomini D., Could Dissecting the Molecular Framework of β-Lactam Integrin Ligands Enhance Selectivity?, «JOURNAL OF MEDICINAL CHEMISTRY», 2019, 62, pp. 10156 - 10166 [articolo]

Wtorek K.; Artali R.; Piekielna-Ciesielska J.; Koszuk J.; Kluczyk A.; Gentilucci L.; Janecka A., Endomorphin-2 analogs containing modified tyrosines: Biological and theoretical investigation of the influence on conformation and pharmacological profile, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 179, pp. 527 - 536 [articolo]

De Marco R.; Zhao J.; Greco A.; Ioannone S.; Gentilucci L., In-Peptide Synthesis of Imidazolidin-2-one Scaffolds, Equippable with Proteinogenic or Taggable/Linkable Side Chains, General Promoters of Unusual Secondary Structures, «JOURNAL OF ORGANIC CHEMISTRY», 2019, 84, pp. 4992 - 5004 [articolo]

Baiula, M; Spampinato, S; Gentilucci, L ; Tolomelli, A, Novel Ligands Targeting alpha(4)beta(1) Integrin: Therapeutic Applications and Perspectives, «FRONTIERS IN CHEMISTRY», 2019, 7, pp. 1 - 12 [articolo]Open Access

De Marco, Rossella; Bedini, Andrea; Spampinato, Santi*; Comellini, Lorenzo; Zhao, Junwei; Artali, Roberto; Gentilucci, Luca, Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 5751 - 5757 [articolo]

Dattoli, Samantha Deianira; Baiula, Monica; De Marco, Rossella; Bedini, Andrea; Anselmi, Michele; Gentilucci, Luca; Spampinato, Santi*, DS-70, a novel and potent α4 integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs, «BRITISH JOURNAL OF PHARMACOLOGY», 2018, 175, pp. 3891 - 3910 [articolo]

De Marco, Rossella; Greco, Arianna; Calonghi, Natalia; Dattoli, Samantha D.; Baiula, Monica; Spampinato, Santi; Picchetti, Pierre; De Cola, Luisa; Anselmi, Michele; Cipriani, Francesca; Gentilucci, Luca*, Selective detection of alfa4beta1 integrin (VLA-4)-expressing cells using peptide-functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites, «PEPTIDE SCIENCE», 2018, 110, pp. 1 - 10 [articolo]

Adamska-Bartłomiejczyk, Anna; De Marco, Rossella; Gentilucci, Luca; Kluczyk, Alicja; Janecka, Anna, Design and characterization of opioid ligands based on cycle-in-macrocycle scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY», 2017, 25, pp. 2399 - 2405 [articolo]

Zanna, Nicola; Focaroli, Stefano; Merlettini, Andrea; Gentilucci, Luca; Teti, Gabriella; Falconi, Mirella; Tomasini, Claudia, Thixotropic peptide-based physical hydrogels applied to three-dimensional cell culture, «ACS OMEGA», 2017, 2, pp. 2374 - 2381 [articolo]Open Access

Marco, Rossella De; Gentilucci, Luca, Tryptophan-Containing Non-Cationizable Opioid Peptides - A new chemotype with unusual structure and in vivo activity, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 2099 - 2115 [articolo]

Gentilucci, Luca; Gallo, Francesca; Meloni, Fernanda; Mastandrea, Marco; Del Secco, Benedetta; de Marco, Rossella, Controlling Cyclopeptide Backbone Conformation with β/α-Hybrid Peptide–Heterocycle Scaffolds, «EUROPEAN JOURNAL OF ORGANIC CHEMISTRY», 2016, 2016, pp. 3243 - 3251 [articolo]

De Marco, Rossella; Mazzotti, Giacomo; Greco, Arianna; Gentilucci, Luca, Heterocyclic Scaffolds in the Design of Peptidomimetic Integrin Ligands: Synthetic Strategies, Structural Aspects, and Biological Activity, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2016, 16, pp. 343 - 359 [articolo]