De Marco, Rossella; Bedini, Andrea; Spampinato, Santi*; Comellini, Lorenzo; Zhao, Junwei; Artali, Roberto; Gentilucci, Luca, Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 5751 - 5757 [Scientific article]Open Access
Dattoli, Samantha Deianira; Baiula, Monica; De Marco, Rossella; Bedini, Andrea; Anselmi, Michele; Gentilucci, Luca; Spampinato, Santi*, DS-70, a novel and potent α4 integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs, «BRITISH JOURNAL OF PHARMACOLOGY», 2018, 175, pp. 3891 - 3910 [Scientific article]Open Access
De Marco, Rossella; Greco, Arianna; Calonghi, Natalia; Dattoli, Samantha D.; Baiula, Monica; Spampinato, Santi; Picchetti, Pierre; De Cola, Luisa; Anselmi, Michele; Cipriani, Francesca; Gentilucci, Luca*, Selective detection of alfa4beta1 integrin (VLA-4)-expressing cells using peptide-functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites, «PEPTIDE SCIENCE», 2018, 110, Article number: e23081 , pp. 1 - 10 [Scientific article]
Adamska-Bartłomiejczyk, Anna; De Marco, Rossella; Gentilucci, Luca; Kluczyk, Alicja; Janecka, Anna, Design and characterization of opioid ligands based on cycle-in-macrocycle scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY», 2017, 25, pp. 2399 - 2405 [Scientific article]
Zanna, Nicola; Focaroli, Stefano; Merlettini, Andrea; Gentilucci, Luca; Teti, Gabriella; Falconi, Mirella; Tomasini, Claudia, Thixotropic peptide-based physical hydrogels applied to three-dimensional cell culture, «ACS OMEGA», 2017, 2, pp. 2374 - 2381 [Scientific article]Open Access
Marco, Rossella De; Gentilucci, Luca*, Tryptophan-Containing Non-Cationizable Opioid Peptides - A new chemotype with unusual structure and in vivo activity, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 2099 - 2115 [Scientific article]
Gentilucci, Luca; Gallo, Francesca; Meloni, Fernanda; Mastandrea, Marco; Del Secco, Benedetta; de Marco, Rossella, Controlling Cyclopeptide Backbone Conformation with β/α-Hybrid Peptide–Heterocycle Scaffolds, «EUROPEAN JOURNAL OF ORGANIC CHEMISTRY», 2016, 2016, pp. 3243 - 3251 [Scientific article]
De Marco, Rossella; Mazzotti, Giacomo; Greco, Arianna; Gentilucci, Luca, Heterocyclic Scaffolds in the Design of Peptidomimetic Integrin Ligands: Synthetic Strategies, Structural Aspects, and Biological Activity, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2016, 16, pp. 343 - 359 [Scientific article]
De Marco, Rossella; Tolomelli, Alessandra; Juaristi, Eusebio; Gentilucci, Luca, Integrin Ligands with α/β-Hybrid Peptide Structure: Design, Bioactivity, and Conformational Aspects, «MEDICINAL RESEARCH REVIEWS», 2016, 36, pp. 389 - 424 [Scientific article]Open Access
Gentilucci, Luca; Tosi, Pierluigi; Bauer, Adriano; De Marco, Rossella, Modern tools for the chemical ligation and synthesis of modified peptides and proteins, «FUTURE MEDICINAL CHEMISTRY», 2016, 8, pp. 2287 - 2304 [Scientific article]
Piekielna, Justyna; De Marco, Rossella; Gentilucci, Luca; Cerlesi, Maria Camilla; Calo', Girolamo; Tömböly, Csaba; Artali, Roberto; Janecka, Anna, Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic, «BIOPOLYMERS», 2016, 106, pp. 309 - 317 [Scientific article]
Gentilucci, L, Synthesis and biomedical appications of tumor targeting peptidomimetics, «LA CHIMICA E L'INDUSTRIA WEB», 2016, 3, pp. 1 - 1 [Scientific article]
Gentilucci, L, Synthesis and Biomedical Applications of Tumor-Targeting Peptidomimetics.
Book of Abstracts., in: Gentilucci, L, Synthesis and Biomedical Applications of Tumor-Targeting Peptidomimetics. Book of Abstracts., 2016, pp. 1 - 87 (atti di: Synthesis and Biomedical Applications of Tumor-Targeting Peptidomimetics., Bologna, 14-16 Febbraio 2016,) [Contribution to conference proceedings]
Perlikowska, Renata; Piekielna, Justyna; Gentilucci, Luca; De Marco, Rossella; Cerlesi, Maria Camilla; Calo, Girolamo; Artali, Roberto; Tömböly, Csaba; Kluczyk, Alicja; Janecka, Anna, Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 109, pp. 276 - 286 [Scientific article]Open Access
DE MARCO, Rossella; Bedini, Andrea; Spampinato, SANTI MARIO; Cavina, Lorenzo; Pirazzoli, Edoardo; Gentilucci, Luca, Versatile Picklocks to Access All Opioid Receptors: Tuning the Selectivity and Functional Profile of the Cyclotetrapeptide c[Phe- d -Pro-Phe-Trp] (CJ-15,208), «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 9255 - 9261 [Scientific article]
