Foto del docente

Giuseppina Di Stefano

Associate Professor

Department of Medical and Surgical Sciences

Academic discipline: MEDS-02/A Experimental Medicine and Pathophysiology

Publications

Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; DI IANNI, Lorenza; Giacomini, Elisa; Falchi, Federico; DI STEFANO, Giuseppina; Roberti, Marinella; Recanatini, Maurizio, Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2016, 14, pp. 10981 - 10987 [Scientific article]

Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini, Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2015, 101, pp. 63 - 70 [Scientific article]

M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano, Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes., «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2015, 74, pp. 95 - 102 [Scientific article]Open Access

Fiume L;Manerba M;Di Stefano G, Albumin-drug conjugates in the treatment of hepatic disorders., «EXPERT OPINION ON DRUG DELIVERY», 2014, 11, pp. 1203 - 1217 [Scientific article]

Luigi FIUME; Marcella MANERBA; Marina VETTRAINO; Giuseppina DI STEFANO, Inhibition of lactate dehydrogenase activity as an approach to cancer therapy, «FUTURE MEDICINAL CHEMISTRY», 2014, 6, pp. 429 - 445 [Scientific article]

Fiume L.; Vettraino M.; Carnicelli D.; Arfilli V.; Di Stefano G.; Brigotti M., Galloflavin prevents the binding of lactate dehydrogenase A to single stranded DNA and inhibits RNA synthesis in cultured cells., «BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS», 2013, 430, pp. 466 - 469 [Scientific article]

Vettraino M; Manerba M; Govoni M; Di Stefano G., Galloflavin suppresses lactate dehydrogenase activity and causes MYC downregulationin Burkitt lymphoma cells via NAD/NADH-dependent inhibition of sirtuin-1, «ANTI-CANCER DRUGS», 2013, 24, pp. 862 - 870 [Scientific article]

Di Stefano G; Manerba M; Vettraino M, NAD metabolism and functions: a common therapeutic target for neoplastic, metabolic and neurodegenerative diseases, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2013, 13, pp. 2918 - 2929 [Scientific article]

Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G., Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways., «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2012, 47, pp. 729 - 738 [Scientific article]

Manerba M.; Vettraino M.; Fiume L.; Di Stefano G.; Sartini A.; Giacomini E.; Buonfiglio R.; Roberti M.; Recanatini M., Galloflavin (CAS 568-80-9), a novel inhibitor of lactate dehydrogenase., «CHEMMEDCHEM», 2012, 7, pp. 311 - 317 [Scientific article]

Fiume L.; Manerba M.; Vettraino M.; Di Stefano G., Effect of sorafenib on the energy metabolism of hepatocellular carcinoma cells., «EUROPEAN JOURNAL OF PHARMACOLOGY», 2011, 670, pp. 39 - 43 [Scientific article]

Fiume L.; Vettraino M.; Manerba M.; Di Stefano G., Inhibition of lactic dehydrogenase as a way to increase the anti-proliferative effect of multi-targeted kinase inhibitors., «PHARMACOLOGICAL RESEARCH», 2011, 63, pp. 328 - 334 [Scientific article]

Ianni M; Manerba M; Di Stefano G; Porcellini E; Chiappelli M; Carbone I; Licastro F., Altered glycosylation profile of purified plasma ACT from Alzheimer's disease., «IMMUNITY & AGEING», 2010, 7, Article number: 56 , pp. 1 - 8 [Scientific article]Open Access

Fiume L; Manerba M; Vettraino M; Di Stefano G, Impairment of aerobic glycolysis by inhibitors of lactic dehydrogenase hinders the growth of human hepatocellular carcinoma cell lines., «PHARMACOLOGY», 2010, 86, pp. 157 - 162 [Scientific article]

Fiume L.; Di Stefano G., Lactosaminated human albumin: a hepatotropic carrier of drugs., «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2010, 40, pp. 253 - 262 [Scientific article]

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