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Giuseppina Di Stefano

Associate Professor

Department of Medical and Surgical Sciences

Academic discipline: MED/04 Experimental Medicine and Pathophysiology

Publications

Marinella Roberti, Fabrizio Schipani, Greta Bagnolini, Domenico Milano, Elisa Giacomini, Federico Falchi, Andrea Balboni, Marcella Manerba, Fulvia Farabegoli, Francesca De Franco, Janet Robertson, Saverio Minucci, Isabella Pallavicini, Giuseppina Di Stefano, Stefania Girotto, Roberto Pellicciari, and Andrea Cavalli, Rad51/Brca2 Disruptors Inhibit Homologous Recombination and Synergize with Olaparib in Pancreatic Cancer Cells, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 165, pp. 80 - 92 [Scientific article]

Manerba M, Di Ianni L, Govoni M, Comparone A, Di Stefano G., The activation of lactate dehydrogenase induced by mTOR drives neoplastic change in breast epithelial cells, «PLOS ONE», 2018, 13, Article number: e0202588 , pp. 1 - 17 [Scientific article]Open Access

Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina, Lactate dehydrogenase inhibitors can reverse inflammation induced changes in colon cancer cells, «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2017, 96, pp. 37 - 44 [Scientific article]Open Access

Manerba, Marcella; Di Ianni, Lorenza; Govoni, Marzia; Roberti, Marinella; Recanatini, Maurizio; Di Stefano, Giuseppina, LDH inhibition impacts on heat shock response and induces senescence of hepatocellular carcinoma cells, «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2017, 105, pp. 91 - 98 [Scientific article]Open Access

Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba, Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea, Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors, «ACS CHEMICAL BIOLOGY», 2017, 12, pp. 2491 - 2497 [Scientific article]

Di Stefano, Giuseppina; Manerba, Marcella; Di Ianni, Lorenza; Fiume, Luigi, Lactate dehydrogenase inhibition: Exploring possible applications beyond cancer treatment, «FUTURE MEDICINAL CHEMISTRY», 2016, 8, pp. 713 - 725 [Scientific article]

Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Falchi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio, Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2016, 14, pp. 10981 - 10987 [Scientific article]

Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini, Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2015, 101, pp. 63 - 70 [Scientific article]

M. Manerba; L. Di Ianni; L. Fiume; M. Roberti; M. Recanatini; G. Di Stefano, Lactate dehydrogenase inhibitors sensitize lymphoma cells to cisplatin without enhancing the drug effects on immortalized normal lymphocytes., «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2015, 74, pp. 95 - 102 [Scientific article]Open Access

Fiume L;Manerba M;Di Stefano G, Albumin-drug conjugates in the treatment of hepatic disorders., «EXPERT OPINION ON DRUG DELIVERY», 2014, 11, pp. 1203 - 1217 [Scientific article]

Luigi FIUME; Marcella MANERBA; Marina VETTRAINO; Giuseppina DI STEFANO, Inhibition of lactate dehydrogenase activity as an approach to cancer therapy, «FUTURE MEDICINAL CHEMISTRY», 2014, 6, pp. 429 - 445 [Scientific article]

Fiume L.; Vettraino M.; Carnicelli D.; Arfilli V.; Di Stefano G.; Brigotti M., Galloflavin prevents the binding of lactate dehydrogenase A to single stranded DNA and inhibits RNA synthesis in cultured cells., «BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS», 2013, 430, pp. 466 - 469 [Scientific article]

Vettraino M; Manerba M; Govoni M; Di Stefano G., Galloflavin suppresses lactate dehydrogenase activity and causes MYC downregulationin Burkitt lymphoma cells via NAD/NADH-dependent inhibition of sirtuin-1, «ANTI-CANCER DRUGS», 2013, 24, pp. 862 - 870 [Scientific article]

Di Stefano G; Manerba M; Vettraino M, NAD metabolism and functions: a common therapeutic target for neoplastic, metabolic and neurodegenerative diseases, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2013, 13, pp. 2918 - 2929 [Scientific article]

Farabegoli F.; Vettraino M.; Manerba M.; Fiume L.; Roberti M.; Di Stefano G., Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways., «EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES», 2012, 47, pp. 729 - 738 [Scientific article]

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