Foto del docente

Andrea Milelli

Professore associato

Dipartimento di Scienze per la Qualità della Vita

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minniti, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna, Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach, «THE FEBS JOURNAL», 2019, 286, pp. 4995 - 5015 [articolo]

Brevetto n. 102019000025840, COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI.

Sestili P.; Brigotti M.; Calcabrini C.; Turrini E.; Arfilli V.; Carnicelli D.; Lucarini M.; Mazzanti A.; Milelli A.; Righi V.; Fimognari C., Deuterium Incorporation Protects Cells from Oxidative Damage, «OXIDATIVE MEDICINE AND CELLULAR LONGEVITY», 2019, 2019, pp. 1 - 13 [articolo]

De Simone A, La Pietra V, Betari N, Petragnani N, Conte M, Daniele S, Pietrobono D, Martini C, Petralla S, Casadei R, Davani L, Frabetti F, Russomanno P, Novellino E, Montanari S, Tumiatti V, Ballerini P, Sarno F, Nebbioso A, Altucci L, Monti B, Andrisano V, Milelli A., Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent To Combat Alzheimer's Disease., «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 469 - 474 [articolo]

Recagni M.; Greco M.L.; Milelli A.; Minarini A.; Zaffaroni N.; Folini M.; Sissi C., Distinct biological responses of metastatic castration resistant prostate cancer cells upon exposure to G-quadruplex interacting naphthalenediimide derivatives, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 177, pp. 401 - 413 [articolo]

Di Paolo, Maria Luisa; Cervelli, Manuela; Mariottini, Paolo; Leonetti, Alessia; Polticelli, Fabio; Rosini, Michela; Milelli, Andrea; Basagni, Filippo; Venerando, Rina; Agostinelli, Enzo; Minarini, Anna, Exploring the activity of polyamine analogues on polyamine and spermine oxidase: methoctramine, a potent and selective inhibitor of polyamine oxidase, «JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY», 2019, 34, pp. 740 - 752 [articolo]

De Simone Angela; Milelli Andrea, Histone Deacetylase Inhibitors as Multitarget Ligands: New Players in Alzheimer's Disease Drug Discovery?, «CHEMMEDCHEM», 2019, 14, pp. 1067 - 1073 [articolo]

De Simone A.; Naldi M.; Tedesco D.; Milelli A.; Bartolini M.; Davani L.; Widera D.; Dallas M.L.; Andrisano V., Investigating in vitro amyloid peptide 1−42 aggregation: Impact of higher molecular weight stable adducts, «ACS OMEGA», 2019, 4, pp. 12308 - 12318 [articolo]

Turrini E, Maffei F, Milelli A, Calcabrini C, Fimognari C, Overview of the Anticancer Profile of Avenanthramides from Oat, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2019, 20, pp. 1 - 23 [articolo]

Basso M.; Milelli A., Transglutaminases, neuronal cell death and neural repair: Implications for traumatic brain injury and therapeutics, «CURRENT OPINION IN NEUROLOGY», 2019, 32, pp. 796 - 801 [articolo]

Manuela Basso; Huan Huan Chen; Debasmita Tripathy; Mariarosaria Conte; Kim Y. P. Apperley; Angela De Simone; Jeffrey W. Keillor; Rajiv Ratan; Angela Nebbioso; Federica Sarno; Lucia Altucci; Andrea Milelli., Designing Dual Transglutaminase 2/Histone Deacetylase Inhibitors Effective at Halting Neuronal Death, «CHEMMEDCHEM», 2018, 13, pp. 227 - 230 [articolo]

Andrea Milelli, Chiara Marchetti, Eleonora Turrini, Elena Catanzaro, Roberta Mazzone, Daniela Tomaselli, Carmela FImognari, Vincenzo Tumiatti, Anna MInarini, Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2018, 28, pp. 1001 - 1004 [articolo]

De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, Andrea; Andrisano, Vincenza, Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2017, 144, pp. 159 - 166 [articolo]

De Simone, Angela; Bartolini, Manuela; Baschieri, Andrea; Apperley, Kim Y.P.; Chen, Huan Huan; Guardigni, Melissa; Montanari, Serena; Kobrlova, Tereza; Soukup, Ondrej; Valgimigli, Luca; Andrisano, Vincenza; Keillor, Jeffrey W.; Basso, Manuela; Milelli, Andrea, Hydroxy-substituted trans-cinnamoyl derivatives as multifunctional tools in the context of Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 139, pp. 378 - 389 [articolo]

Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini, Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna, Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 128, pp. 107 - 122 [articolo]