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Andrea Milelli

Professore associato

Dipartimento di Scienze per la Qualità della Vita

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

De Simone Angela; Milelli Andrea, Histone Deacetylase Inhibitors as Multitarget Ligands: New Players in Alzheimer's Disease Drug Discovery?, «CHEMMEDCHEM», 2019, 14, pp. 1067 - 1073 [articolo]

De Simone A.; Naldi M.; Tedesco D.; Milelli A.; Bartolini M.; Davani L.; Widera D.; Dallas M.L.; Andrisano V., Investigating in vitro amyloid peptide 1−42 aggregation: Impact of higher molecular weight stable adducts, «ACS OMEGA», 2019, 4, pp. 12308 - 12318 [articolo]Open Access

Turrini E, Maffei F, Milelli A, Calcabrini C, Fimognari C, Overview of the Anticancer Profile of Avenanthramides from Oat, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2019, 20, Article number: 4536, pp. 1 - 23 [articolo]Open Access

Basso M.; Milelli A., Transglutaminases, neuronal cell death and neural repair: Implications for traumatic brain injury and therapeutics, «CURRENT OPINION IN NEUROLOGY», 2019, 32, pp. 796 - 801 [articolo]

Manuela Basso; Huan Huan Chen; Debasmita Tripathy; Mariarosaria Conte; Kim Y. P. Apperley; Angela De Simone; Jeffrey W. Keillor; Rajiv Ratan; Angela Nebbioso; Federica Sarno; Lucia Altucci; Andrea Milelli., Designing Dual Transglutaminase 2/Histone Deacetylase Inhibitors Effective at Halting Neuronal Death, «CHEMMEDCHEM», 2018, 13, pp. 227 - 230 [articolo]Open Access

Andrea Milelli, Chiara Marchetti, Eleonora Turrini, Elena Catanzaro, Roberta Mazzone, Daniela Tomaselli, Carmela FImognari, Vincenzo Tumiatti, Anna MInarini, Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2018, 28, pp. 1001 - 1004 [articolo]

De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, Andrea; Andrisano, Vincenza, Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2017, 144, pp. 159 - 166 [articolo]

De Simone, Angela; Bartolini, Manuela; Baschieri, Andrea; Apperley, Kim Y.P.; Chen, Huan Huan; Guardigni, Melissa; Montanari, Serena; Kobrlova, Tereza; Soukup, Ondrej; Valgimigli, Luca; Andrisano, Vincenza; Keillor, Jeffrey W.; Basso, Manuela; Milelli, Andrea, Hydroxy-substituted trans-cinnamoyl derivatives as multifunctional tools in the context of Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 139, pp. 378 - 389 [articolo]

Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini, Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna, Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 128, pp. 107 - 122 [articolo]

Alice, Pasini; Chiara, Marchetti; Claudia, Sissi; Marilisa, Cortesi; Emanuele, Giordano; Anna, Minarini; Andrea, Milelli, Novel Polyamine–Naphthalene Diimide Conjugates Targeting Histone Deacetylases and DNA for Cancer Phenotype Reprogramming, «ACS MEDICINAL CHEMISTRY LETTERS», 2017, 8, pp. 1218 - 1223 [articolo]Open Access

Milelli, Andrea; De Simone, Angela; Ticchi, Nicole; Chen, Huan Huan; Betari, Nibal; Andrisano, Vincenza; Tumiatti, Vincenzo, Tacrine-based Multifunctional Agents in Alzheimer's Disease: an Old Story in Continuous Development, «CURRENT MEDICINAL CHEMISTRY», 2017, 24, pp. 3522 - 3546 [articolo]

Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A., Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 117, pp. 283 - 291 [articolo]

D'Urzo, Annalisa; DE SIMONE, Angela; Fiori, Jessica; Naldi, Marina; Milelli, Andrea; Andrisano, Vincenza, Direct determination of GSK-3β activity and inhibition by UHPLC-UV-vis diode arrays detector (DAD), «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2016, 124, pp. 104 - 111 [articolo]

Milelli, Andrea; Turrini, Eleonora; Catanzaro, Elena; Maffei, Francesca; Fimognari, Carmela, Perspectives in Designing Multifunctional Molecules in Antipsychotic Drug Discovery, «DRUG DEVELOPMENT RESEARCH», 2016, 77, pp. 437 - 443 [articolo]

Tumiatti, Vincenzo; Milelli, Andrea, Farmaci Tiroidei, in: Chimica farmaceutica, Rozzano (MI), Casa Editrice Ambrosiana, 2015, pp. 583 - 594 [capitolo di libro]