Nordio G.; Piazzola F.; Cozza G.; Rossetto M.; Cervelli M.; Minarini A.; Basagni F.; Tassinari E.; Dalla Via L.; Milelli A.; Di Paolo M.L., From Monoamine Oxidase Inhibition to Antiproliferative Activity: New Biological Perspectives for Polyamine Analogs, «MOLECULES», 2023, 28, Article number: 6329 , pp. 1 - 18 [Scientific article]Open Access
Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A., PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease, «ACS CHEMICAL NEUROSCIENCE», 2023, 14, pp. 1963 - 1970 [Scientific article]Open Access
Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi M.L., Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery, «ACS BIO & MED CHEM AU», 2023, 3, pp. 32 - 45 [Scientific article]Open Access
EFRAIM REYES; Liher Prieto; ANDREA MILELLI, Asymmetric Organocatalysis: A Survival Guide to Medicinal Chemists, «MOLECULES», 2022, 28, Article number: 271 , pp. 1 - 24 [Scientific article]Open Access
Ragno, Rino; Minarini, Anna; Proia, Eleonora; Lorenzo, Antonini; Milelli, Andrea; Tumiatti, Vincenzo; Fiore, Marco; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Di Paolo, Maria Luisa; Agostinelli, Enzo, Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies, «JOURNAL OF CHEMICAL INFORMATION AND MODELING», 2022, 62, pp. 3910 - 3927 [Scientific article]Open Access
Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Guardigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura, Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 9507 - 9530 [Scientific article]Open Access
Angela De Simone,
Vincenzo Tumiatti,
VIncenza Andrisano,
Andrea Milelli, Glycogen Synthase Kinase 3β: A New Gold Rush in Anti-Alzheimer’s Disease Multitarget Drug Discovery?, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 26 - 41 [Scientific article]Open Access
Loi, Manuela; Gennaccaro, Laura; Fuchs, Claudia; Trazzi, Stefania; Medici, Giorgio; Galvani, Giuseppe; Mottolese, Nicola; Tassinari, Marianna; Giorgini, Roberto Rimondini; Milelli, Andrea; Ciani, Elisabetta, Treatment with a GSK-3β/HDAC Dual Inhibitor Restores Neuronal Survival and Maturation in an In Vitro and In Vivo Model of CDKL5 Deficiency Disorder, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2021, 22, Article number: 5950 , pp. 1 - 24 [Scientific article]Open Access
Catanzaro E.; Betari N.; Arencibia J.M.; Montanari S.; Sissi C.; De Simone A.; Vassura I.; Santini A.; Andrisano V.; Tumiatti V.; De Vivo M.; Krysko D.V.; Rocchi M.B.L.; Fimognari C.; Milelli A., Targeting topoisomerase II with trypthantrin derivatives: Discovery of 7-((2-(dimethylamino)ethyl)amino)indolo[2,1-b]quinazoline-6,12-dione as an antiproliferative agent and to treat cancer, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2020, 202, Article number: 112504 , pp. 112504 - 112504 [Scientific article]Open Access
Di Paolo, Maria Luisa; Cozza, Giorgio; Milelli, Andrea; Zonta, Francesca; Sarno, Stefania; Minniti, Elirosa; Ursini, Fulvio; Rosini, Michela; Minarini, Anna, Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach, «THE FEBS JOURNAL», 2019, 286, pp. 4995 - 5015 [Scientific article]
Patent n. 102019000025840, COMPOSTI ISOTIOCIANATI E ISOSELENCIANATI.
Sestili P.; Brigotti M.; Calcabrini C.; Turrini E.; Arfilli V.; Carnicelli D.; Lucarini M.; Mazzanti A.; Milelli A.; Righi V.; Fimognari C., Deuterium Incorporation Protects Cells from Oxidative Damage, «OXIDATIVE MEDICINE AND CELLULAR LONGEVITY», 2019, 2019, Article number: 6528106 , pp. 1 - 13 [Scientific article]Open Access
De Simone A, La Pietra V, Betari N, Petragnani N, Conte M, Daniele S, Pietrobono D, Martini C, Petralla S, Casadei R, Davani L, Frabetti F, Russomanno P, Novellino E, Montanari S, Tumiatti V, Ballerini P, Sarno F, Nebbioso A, Altucci L, Monti B, Andrisano V, Milelli A., Discovery of the First-in-Class GSK-3β/HDAC Dual Inhibitor as Disease-Modifying Agent To Combat Alzheimer's Disease., «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 469 - 474 [Scientific article]Open Access
Recagni M.; Greco M.L.; Milelli A.; Minarini A.; Zaffaroni N.; Folini M.; Sissi C., Distinct biological responses of metastatic castration resistant prostate cancer cells upon exposure to G-quadruplex interacting naphthalenediimide derivatives, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 177, pp. 401 - 413 [Scientific article]
Di Paolo, Maria Luisa; Cervelli, Manuela; Mariottini, Paolo; Leonetti, Alessia; Polticelli, Fabio; Rosini, Michela; Milelli, Andrea; Basagni, Filippo; Venerando, Rina; Agostinelli, Enzo; Minarini, Anna, Exploring the activity of polyamine analogues on polyamine and spermine oxidase: methoctramine, a potent and selective inhibitor of polyamine oxidase, «JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY», 2019, 34, pp. 740 - 752 [Scientific article]Open Access
