Foto del docente

Alessandra Locatelli

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Delegate of Department of Pharmacy and Biotechnology

Publications

Ravegnini, Gloria; Esposito, Daniele; Gorini, Francesca; Marforio, Tainah Dorina; Coschina, Emma; Benuzzi, Eva; Simone, Antonella; Samaha, Ahmed; Di Vito, Aldo; Rossi, Martina; Hrelia, Patrizia; Locatelli, Alessandra; Calvaresi, Matteo; Facchinello, Nicola; Morigi, Rita; Angelini, Sabrina, Identification of MBT3T as a new effective therapeutic option in imatinib-resistant gastrointestinal stromal tumors (GISTs), «JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH», 2026, 45, pp. 1 - 15 [Scientific article]

Esposito, Daniele; Locatelli, Alessandra; Morigi, Rita, Molecular Tools for Precision Targeting and Detection of G-Quadruplex Structures, «MOLECULES», 2025, 30, Article number: 4099 , pp. 1 - 44 [Scientific article]Open Access

Camarda, Luca; Corazza, Ivan; Locatelli, Alessandra; Leoni, Alberto; Frosini, Maria; Budriesi, Roberta; Carosati, Emanuele; Santini, Alberto; Montagnani, Marco; Marzetti, Carla; Mattioli, Laura Beatrice, Repurposing 1,4-Dihydropyridine Scaffold: 4-Imidazo[2,1-b]thiazole-Derivatives from Calcium Entry Blockers to a New Approach for Gut Dysfunctional Motility, «PHARMACEUTICALS», 2025, 18, Article number: 1476 , pp. 1 - 41 [Scientific article]Open Access

Morigi R.; Zalambani C.; Farruggia G.; Verardi L.; Esposito D.; Leoni A.; Borsetti F.; Voltattorni M.; Zambonin L.; Pincigher L.; Calonghi N.; Locatelli A., Identification of a new bisindolinone arresting IGROV1 cells proliferation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2024, 271, pp. 1 - 19 [Scientific article]Open Access

Morigi, Rita; Esposito, Daniele; Calvaresi, Matteo; Marforio, TAINAH DORINA; Gentilomi, GIOVANNA ANGELA; Bonvicini, Francesca; Locatelli, Alessandra, Isatin Bis-Imidathiazole Hybrids Identified as FtsZ Inhibitors with On-Target Activity Against Staphylococcus aureus, «ANTIBIOTICS», 2024, 13, pp. 1 - 17 [Scientific article]Open Access

Marzano S.; Miglietta G.; Morigi R.; Marinello J.; Arleo A.; Procacci M.; Locatelli A.; Leoni A.; Pagano B.; Randazzo A.; Amato J.; Capranico G., Balancing Affinity, Selectivity, and Cytotoxicity of Hydrazone-Based G-Quadruplex Ligands for Activation of Interferon β Genes in Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 12055 - 12067 [Scientific article]Open Access

Francesca Bonvicini, Alessandra Locatelli, Rita Morigi, Alberto Leoni, Giovanna Angela Gentilomi, Isatin Bis-Indole and Bis-Imidazothiazole Hybrids: Synthesis and Antimicrobial Activity, «MOLECULES», 2022, 27, pp. 5781 - 5792 [Scientific article]Open Access

Das A.; Greco G.; Kumar S.; Catanzaro E.; Morigi R.; Locatelli A.; Schols D.; Alici H.; Tahtaci H.; Ravindran F.; Fimognari C.; Karki S.S., Synthesis, in vitro cytotoxicity, molecular docking and ADME study of some indolin-2-one linked 1,2,3-triazole derivatives, «COMPUTATIONAL BIOLOGY AND CHEMISTRY», 2022, 97, Article number: 107641 , pp. 1 - 18 [Scientific article]Open Access

Morigi R.; Catanzaro E.; Locatelli A.; Calcabrini C.; Pellicioni V.; Leoni A.; Fimognari C., Synthesis and biological evaluation of new bis-indolinone derivatives endowed with cytotoxic activity, «MOLECULES», 2021, 26, Article number: 6277 , pp. 1 - 15 [Scientific article]Open Access

Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N., Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth, «MOLECULES», 2020, 25, Article number: 4438 , pp. 1 - 15 [Scientific article]Open Access

Amato J.; Miglietta G.; Morigi R.; Iaccarino N.; Locatelli A.; Leoni A.; Novellino E.; Pagano B.; Capranico G.; Randazzo A., Monohydrazone Based G-Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 3090 - 3103 [Scientific article]Open Access

Pesce, Emanuela; Pedemonte, Nicoletta; Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita, Synthesis and biological evaluation of thiazole derivatives on basic defects underlying cystic fibrosis., «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2020, 30, Article number: 127473 , pp. 1 - 7 [Scientific article]Open Access

Leoni, Alberto; Frosini, Maria; Locatelli, Alessandra; Micucci, Matteo; Carotenuto, Claudio; Durante, Miriam; Cosconati, Sandro; Budriesi, Roberta*, 4-Imidazo[2,1-b]thiazole-1,4-DHPs and neuroprotection: preliminary study in hits searching, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 169, pp. 89 - 102 [Scientific article]Open Access

Alessandra Locatelli, Luisa Iommarini, Alessandra Graziadio, Alberto Leoni, Anna Maria Porcelli, Stefano Iotti, Emil Malucelli, Francesco Francia, Giovanni Venturoli, Giovanna Farruggia, Dansyl acetyl trehalose: a novel tool to investigate the cellular fate of trehalose, «RSC ADVANCES», 2019, 9, pp. 15350 - 15356 [Scientific article]Open Access

Conti, Ilaria; Morigi, Rita; Locatelli, Alessandra*; Rambaldi, Mirella; Bua, Gloria; Gallinella, Giorgio; Leoni, Alberto, Synthesis of 3-(Imidazo[2,1-b]thiazol-6-yl)-2H-chromen-2-one derivatives and study of their antiviral activity against parvovirus B19, «MOLECULES», 2019, 24, Article number: 1037 , pp. 1 - 15 [Scientific article]Open Access