Foto del docente

Alessandra Locatelli

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Andreani A.; Burnelli S.; Granaiola M.; Leoni A.; Locatelli A.; Morigi R.; Rambaldi M.; Varoli L.; Calonghi N.; Cappadone C.; Farruggia G.; Zini M.; Stefanelli C.; Masotti L., Substituted E-3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity. Effect on the cell cycle and apoptosis., «JOURNAL OF MEDICINAL CHEMISTRY», 2007, 50, pp. 3167 - 3172 [Scientific article]

A. Andreani; S. Burnelli; M. Granaiola; A. Leoni; A. Locatelli; R. Morigi; M. Rambaldi; L. Varoli; M.W. Kunkel, Antitumor Activity of Substituted E-3-(3,4,5-Trimethoxybenzylidene)-1,3-dihydroindol-2-ones, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 6922 - 6924 [Scientific article]

A. Andreani; S. Burnelli; M. Granaiola; A. Leoni; A. Locatelli; R. Morigi; M. Rambaldi; L. Varoli; G. Farruggia; C. Stefanelli; L. Masotti; M.W. Kunkel, Synthesis and antitumor activity of Guanylhydrazones from 6-(2,4-dichloro-5-nitrophenyl)imidazo[2,1-b]thiazoles and 6-pyridylimidazo[2,1-b]thiazoles, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 7897 - 7901 [Scientific article]

A. Andreani; M. Granaiola; A. Leoni; A. Locatelli; R. Morigi; M. Rambaldi; V. Garaliene; W. Welsh; S. Arora; G. Farruggia;| L. Masotti, Antitumor Activity of New Substituted 3-(5-Imidazo[2,1-b]thiazolylmethylene)-2-indolinones and Study of Their Effect on the Cell Cycle, «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48, pp. 5604 - 5607 [Scientific article]

Patent n. Brev. Ital. BO2005 A 000476, Composti organici ad attività antitumorale.

A. Andreani; M. Granaiola; A. Leoni; A. Locatelli; R. Morigi; M. Rambaldi; G. Lenaz; R. Fato; C. Bergamini; G. Farruggia, Potential Antitumor Agents. 37. Synthesis and Antitumor Activity of Guanylhydrazones from Imidazo[2,1-b]thiazoles and from the New Heterocyclic System Thiazolo[2',3':2,3]imidazo[4,5-c]quinoline, «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48, pp. 3085 - 3089 [Scientific article]

ALDO ANDREANI; MASSIMILIANO GRANAIOLA; MASSIMO GUARDIGLI; ALBERTO LEONI; ALESSANDRA LOCATELLI; RITA MORIGI; MIRELLA RAMBALDI; ALDO RODA, Synthesis and chemiluminescent high throughput screening for inhibition of acetylcholinesterase activity by imidazo[2,1-b]thiazole derivatives, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2005, 40, pp. 1331 - 1334 [Scientific article]

ANDREANI A.; GRANAIOLA M.; LEONI A.; LOCATELLI A.; MORIGI R.; RAMBALDI M.; RECANATINI M.; LENAZ G.; FATO R.; BERGAMINI C., Effect of new ubiquinone-imidazo[2,1-b] thiazoles on mitochondrial Complex I (NADH ubiquinone reductase) and on mitochondrial permeability transition pore., «BIOORGANIC & MEDICINAL CHEMISTRY», 2004, 12, pp. 5525 - 5532 [Scientific article]

A. Andreani; M. Granaiola; A. Leoni; A. Locatelli; R. Morigi; M. Rambaldi; A. Roda; M. Guardigli; S. Traniello; S. Spisani, N-Benzyl-2-chloroindole-3-carboxylic acids as potential anti-inflammatory agents. Synthesis and screening for the effects on human neutrophil functions and on COX1/COX2 activity, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2004, 39, pp. 785 - 791 [Scientific article]

ANDREANI A.; GRANAIOLA M.; LEONI A.; LOCATELLI A.; MORIGI R.; RAMBALDI M.; GIORGI G.; GARALIENE V., Potential antitumor agents. 34.(1)Synthesis and antitumor activity of guanylhydrazones from imidazo[2,1-b]thiazoles and from diimidazo[1,2-a:1,2-c]pyrimidine, «ANTICANCER RESEARCH», 2004, 24, pp. 203 - 212 [Scientific article]

Andreani A.; Granaiola M.; Leoni A.; Locatelli A.; Morigi R.; Rambaldi M.; Garaliene V.; Farruggia G.; Masotti L., Substituted E-3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones with antitumor activity, «BIOORGANIC & MEDICINAL CHEMISTRY», 2004, 12, pp. 1121 - 1128 [Scientific article]

ALDO ANDREANI; MASSIMILIANO GRANAIOLA; ALBERTO LEONI; ALESSANDRA LOCATELLI; RITA MORIGI; MIRELLA RAMBALDI; GIORGIO LENAZ; ROMANA FATO; CHRISTIAN BERGAMINI, 2-[(E)-3-(6-chloroimidazo[2,1-b]thiazol-5-ylprop-2-enyl]5,6-dimethoxy-3-methyl-1,4-benzo quinone: a new inhibitor of NADH dehydrogenase with antitumor activity, «ARKIVOC», 2004, V, pp. 76 - 84 [Scientific article]