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Publications prior to 2004
1) Andreani A., Rambaldi M., Locatelli A., Bossa R., Galatulas
I., Ninci M.:Synthesis and cardiotonic activity of
2-indolinones
Eur.J.Med.Chem. 25, 187-190 (1990)
2) Andreani A., Rambaldi M., Locatelli A., Aresca P., Bossa R.,
Galatulas I.:Potential antitumor agents XVIII. Synthesis and
cytotoxic activity of phenothiazine derivatives
Eur.J.Med.Chem. 26, 113-116 (1991)
3) Andreani A., Rambaldi M., Locatelli A., Andreani F., Aresca
P., Bossa R., Galatulas I.: Potential antitumor agents XVII.
Cytotoxic agents from indole derivatives and their
intermediates
Acta Pharm.Nord. 2, 407-414 (1990)
4) Andreani A., Rambaldi M., Locatelli A., Isetta A.M.:
Synthesis and mitogenic activity of new imidazo[2,1-b]thiazoles
Eur.J.Med.Chem. 26, 335-337 (1991)
5) Andreani A., Rambaldi M., Locatelli A., Conti M., Malandrino
S.: Synthesis and antiinflammatory activity of indole carboxylic
acids and esters
Acta Pharm.Nord. 3, 5-8 (1991)
6) Andreani A., Rambaldi M., Locatelli A., Andreani F.:
5-Formylimidazo[2,1-b]thiazoles and derivatives with herbicidal
activity
Collect.Czech.Chem.Comm. 56, 2436-2447 (1991)
7) Andreani A., Rambaldi M., Locatelli A.: Herbicidal activity
of 5-haloimidazo[2,1-b]thiazoles
Collect.Czech.Chem.Comm. 56, 2430-2435 (1991)
8) Andreani A., Rambaldi M., Locatelli A., Andreani F., Bossa
R., Galatulas I., Ninci M.: Synthesis and analgesic activity of
1-(N-methylanilinoethyl)indoles
Acta Pharm.Nord. 3, 125-129 (1991)
9) Andreani A., Rambaldi M., Locatelli A., Bongini A., Bossa R.,
Galatulas I., Ninci M.: Synthesis and cardiotonic activity of
pyridylmethylene-2-indolinones
Eur.J.Med.Chem. 27, 167-170 (1992)
10) Andreani A., Rambaldi M., Locatelli A., Cristoni A.,
Malandrino S., Pifferi G.: Synthesis and antihypertensive activity
of imidazo[2,1-b]thiazoles bearing a 2,6-dichlorophenyl group
Acta Pharm.Nord. 4, 93-96 (1992)
11) Andreani A., Rambaldi M., Locatelli A., Bossa R., Galatulas
I., Ninci M.: Synthesis and cardiotonic activity of
2,5-dimethoxyphenylimidazo[2,1-b]thiazoles
Eur.J.Med.Chem. 27, 431-433 (1992)
12) Andreani A., Rambaldi M., Locatelli A., Fraccari A., Bossa
R., Galatulas I.: Potential antitumor agents. XIX. Synthesis and
antitumor activity of tricyclic compounds related to lotifazole
Pharm.Acta Helv. 67, 234-236 (1992)
13) Andreani A., Rambaldi M., Locatelli A., Pifferi G.,
Malandrino S.: Synthesis and pharmacological activity of
imidazo[2,1-b]thiazole nitriles, amides and
p-sulfamido-phenylhydrazones
Pharm.Acta Helv. 67, 195-197 (1992)
14) Andreani A., Rambaldi M., Locatelli A., Malandrino S.,
Pifferi G.: Synthesis and diuretic activity of
(E)-2-methyl-6-phenylimidazo[2,1-b]-1,3,4-thiadiazole-5-carboxaldehyde
dimethyl-aminoacetohydrazone
Arzneim.Forsch. 44, 618-619 (1994)
15) Andreani A., Rambaldi M., Locatelli A., Andreani F.,
Poglayen G., Degli Esposti M.: 3-(2-Thienylvinyl)indoles as
potential specific inhibitors of the energy metabolism in
helminthic parasites
Eur.J.Med.Chem. 27, 729-734 (1992)
16) Andreani A., Rambaldi M., Locatelli A., Bossa R., Fraccari
A., Galatulas I.: Potential antitumor agents XX.
6-Anilinoimidazo[2,1-b]thiazoles
Pharm.Acta Helv. 68, 21-24 (1993)
17) Andreani A., Rambaldi M., Locatelli A., Bossa R., Fraccari
A., Galatulas I.: Potential antitumor agents. XXI. Structure
determination and antitumor activity of imidazo[2,1-b]thiazole
guanylhydrazones
J.Med.Chem. 35, 4634-4637 (1992)
18) Andreani A., Rambaldi M., Leoni A., Locatelli A., Bossa R.,
Chiericozzi M., Dambrosio M., Galatulas I.: Synthesis and
cardiotonic activity of 2-indolinones bearing pyridyl groups
Eur.J.Med.Chem. 28, 653-657 (1993)
19) Andreani A., Rambaldi M., Locatelli A., Leoni A., Bossa R.,
Chiericozzi M., Galatulas I., Salvatore G.: Synthesis of lactams
with potential cardiotonic activity
Eur.J.Med.Chem. 28, 825-829 (1993)
20) Andreani A., Rambaldi M., Locatelli A., Bossa R., Fraccari
A., Galatulas I.: Potential antitumor agents XXII. Synthesis and
cytotoxic activity of imidazo[2,1-b]thiazole
adamanthylthioureas
J.Pharm.Belg. 48, 378-382 (1993)
21) Andreani A., Rambaldi M.,Locatelli A., Leoni A., Ghelli A.,
Degli Esposti M.: Thienylvinylindoles as inhibitors of
mitochondrial NADH dehydrogenase
Pharm.Acta Helv. 69, 15-20 (1994)
22) Andreani A., Rambaldi M., Locatelli A., Andreani F., Lollini
P.L., Nanni P., Bossa R., Galatulas I.: Potential antitumor agents
XXIII. Cytotoxic and differentiating activity of compounds related
to hexamethylenebisacetamide
Il Farmaco 48, 1503-1513 (1993)
23) Andreani A., Rambaldi M., Leoni A., Locatelli A., Pifferi
G.: Synthesis of imidazo[2,1-b]thiazoles as potential antiulcer
agents
J.Pharm.Belg. 49, 308-314 (1994)
24) Andreani A., Rambaldi M., Locatelli A., Bossa R., Salvatore
G., Galatulas I: Synthesis and cardiotonic activity of aryl- or
pyridyl-substituted fused imidazoles
Eur.J.Med.Chem. 29, 339-342 (1994)
25) Andreani A., Rambaldi M., Leoni A., Locatelli A., Ghelli A.,
Ratta M., Benelli B., Degli Esposti M.:
Thienylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH
dehydrogenase
J.Med.Chem. 38, 1090-1097 (1995)
26) Andreani A., Locatelli A., Rambaldi M.: Synthesis and
herbicidal properties of
3-(2-oxo-1-imidazolidinyliminomethyl)indoles
J.Heterocyclic Chem. 32, 49-51 (1995)
27) Andreani A., Rambaldi M., Locatelli A., Bossa R., Galatulas
I., Salvatore G.: Antitumor and cardiotonic activity of
imidazo[2,1-b]thiazole guanylhydrazones
In vivo 8, 1031-1032 (1994)
28) Andreani A., Rambaldi M., Locatelli A., Pifferi G.:
Synthesis and antiinflammatory activity of indolylacrylic and
methylacrylic acids
Eur.J.Med.Chem. 29, 903-906 (1994)
29) Andreani A., Rambaldi M., Locatelli A.: Synthesis and
fungicide activity of
2,3-dihydoimidazo[2,1-b]thiazole-5-carboxamides
Pharm.Acta Helv. 70, 325-328 (1995)
30) Andreani A., Rambaldi M., Leoni A., Locatelli A.,
Andreani F., Gehret J.C.: Synthesis of imidazo[2,1-b]thiazoles as
herbicides
Pharm.Acta Helv. 71, 247-252 (1996)
31) Andreani A., Rambaldi M., Leoni A., Locatelli A., Bossa R.,
Chiericozzi M., Galatulas I., Salvatore G.: Synthesis and
cardiotonic activity of imidazo[2,1-b]thiazoles bearing a lactam
ring
Eur.J.Med.Chem. 31, 383-387 (1996)
32) Andreani A., Rambaldi M., Leoni A., Locatelli A., Bossa R.,
Fraccari A., Galatulas I., Salvatore G.: Potential antitumor
agents. 24. Synthesis and pharmacological behavior of
imidazo[2,1-b]thiazole guanylhydrazones bearing at least one
chlorine
J.Med.Chem. 39, 2852-2855 (1996)
33) Andreani A., Rambaldi M., Leoni A., Locatelli A., Andreani
F., Bossa R., Chiericozzi M., Cozzi R., Galatulas I: Synthesis of
6-methylimidazo[2,1-b]thiazole derivatives acting on neuromuscular
transmission
Eur.J.Med.Chem. 31, 741-744 (1996)
34) Andreani A., Locatelli A., Rambaldi M., Leoni A., Bossa R.,
Fraccari A., Galatulas I.: Potential antitumor agents. 25.
Synthesis and cytotoxic activity of
3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones
Anticancer Res. 16, 3585-3588 (1996)
35) Andreani A., Leoni A., Rambaldi M., Locatelli A., Bossa R.,
Galatulas I., Chiericozzi M., Cozzi R.: Dihydropyridines bearing an
imidazo[2,1-b]thiazole system
Eur.J.Med.Chem. 32, 151-157 (1997)
36) Andreani A., Locatelli A., Leoni A., Rambaldi M., Morigi R.,
Bossa R., Chiericozzi M., Fraccari A., Galatulas I.: Synthesis and
potential coanthracyclinic activity of substituted
3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones
Eur.J.Med.Chem. 32, 919-924 (1997)
37) Andreani A., Leoni A., Locatelli A., Morigi R., Rambaldi M.,
Gehret J.C., Traniello S., Cariani A., Spisani S.: Ring opened
analogs of indomethacin affecting human neutrophil functions
Collect.Czech.Chem.Comm. 64, 299-312 (1999)
38) Andreani A., Locatelli A., Morigi R., Leoni A., Bossa R.,
Chiericozzi M., Galatulas I.: In vivo cardiotonic activity of
pyridylmethylene-2-indolinones
Arzneim.Forsch. 48, 727-729 (1998)
39) Andreani A., Locatelli A., Leoni A., Morigi R., Chiericozzi
M., Fraccari A., Galatulas I., Salvatore G.: Synthesis and
potential coanthracyclinic activity of pyridylmethylene and
indolylmethylene lactams
Eur.J.Med.Chem. 33, 905-909 (1998)
40) Andreani A., Leoni A., Locatelli A., Morigi R., Chiericozzi
M., Fraccari A., Galatulas I.: Potential coanthracyclinic activity
of pyridylmethylene-2-indolinones
Anticancer Res. 18, 3407-3410 (1998)
41) Andreani A., Rambaldi M., Leoni A., Locatelli A., Morigi R.,
Traniello S., Cariani A., Rizzuti O. Spisani S.:
Hydroxyphenylimidazo[2,1-b]thiazoles as potential antiinflammatory
agents: effects on human neutrophil functions
Collect.Czech.Chem.Comm. 65, 267-279 (2000)
42) Andreani A., Rambaldi M., Leoni A., Morigi R., Locatelli A.,
Giorgi G., Lenaz G., Ghelli A., Degli Esposti M.: 6-Thienyl and
6-phenylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH
dehydrogenase
Eur.J.Med.Chem. 34, 883-889 (1999)
43) Andreani A., Leoni A., Locatelli A., Morigi R., Rambaldi M.,
Simon W.A., Senn-Bilfinger J.: Synthesis and antisecretory activity
of 6-substituted 5-cyanomethylimidazo[2,1-b]thiazoles and
2,6-dimethyl-5-hydroxymethylimidazo[2,1-b][1,3,4]thiadiazole
Arzneim. Forsch. 50, 550-553 (2000)
44) Giorgi G., Salvini L., Andreani A., Locatelli A., Leoni A.:
Molecular structure, characterization and stereochemical properties
of new biologically interesting
3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones
J.Mol.Struct. 524, 189-199 (2000)
45) Andreani A., Leoni A., Locatelli A., Morigi R., Rambaldi M.,
Pietra C., Villetti G.: 4-Aminopyridine derivatives with
antiamnesic activity
Eur.J.Med.Chem. 35, 77-82 (2000)
46) Andreani A., Leoni A., Locatelli A., Morigi R., Rambaldi M.,
Recanatini M., Garaliene V.: Potential antitumor agents. 29.
Synthesis and potential coanthracyclinic activity of
imidazo[2,1-b]thiazole guanylhydrazones
Bioorg.Med.Chem. 8, 2359-2366 (2000)
47) Andreani A., Cavalli A., Granaiola M., Leoni A., Locatelli
A., Morigi R., Rambaldi M., Recanatini M., Garnier M., Meijer L.:
Imidazo[2,1-b]thiazolylmethylene- and
Indolylmethylene-2-indolinones: a New Class of Cyclin-Dependent
Kinase Inhibitors. Design, Synthesis, and CDK1/Cyclin B
Inhibition
Anticancer Drug Design 15, 447-452 (2000)
48) Andreani A., Cavalli A., Granaiola M., Guardigli M., Leoni
A., Locatelli A., Morigi R., Rambaldi M., Recanatini M., Roda A.:
Synthesis and screening for antiacetylcholinesterase activity of
(1-benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles
related to donepezil
J.Med.Chem. 44, 4011-4014 (2001)
49) Andreani A., Granaiola M., Leoni A., Locatelli A., Morigi
R., Rambaldi M.: Synthesis and antitubercular activity of
imidazo[2,1-b]thiazoles
Eur.J.Med.Chem. 36, 743-746 (2001)
50) Andreani A., Granaiola M., Leoni A., Locatelli A., Morigi
R., Rambaldi M., Giorgi G., Salvini L., Garaliene V.
Synthesis and antitumor activity of substituted
3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones
Anticancer Drug Design 16, 167-174 (2001)
51) Andreani A., Granaiola M., Leoni A., Locatelli A., Morigi
R., Rambaldi M., Garaliene V.: Synthesis and antitumor activity of
1,5,6-substituted
3-(2-chloro-3-indolylmethylene)1,3-dihydroindol-2-ones
J.Med.Chem. 45, 2666-2669 (2002)
52) Andreani A., Granaiola M., Leoni A., Locatelli A., Morigi
R., Rambaldi M., Giorgi G., Salvini L.: Cancer fighting cancer:
synthesis of the new heterocyclic system
diimidazo-[1,2-a:1,2-c]-pyrimidine
Arkivoc 2002, Part XI (Commemorative Issue in Honor of Prof.
Domenico Spinelli), 32-38. Received Sep. 25, 2002; published Nov.
11, 2002
http://www.arkat-usa.org/ark/journal/2002/I11_Spinelli/MS-561H/561H.pdf