Foto del docente

Vincenza Andrisano

Full Professor

Department for Life Quality Studies

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

A. Rampa; M. Bartolini; A. Bisi; F. Belluti; S. Gobbi; V. Andrisano; A. Ligresti; V. Di Marzo, The first dual ChE/FAAH inhibitors: new perspectives for Alzheimer's disease?, «ACS MEDICINAL CHEMISTRY LETTERS», 2012, 3, pp. 182 - 186 [Scientific article]

Pulawski W; Ghoshdastider U; Andrisano V; Filipek S, Ubiquitous amyloids, «APPLIED BIOCHEMISTRY AND BIOTECHNOLOGY», 2012, 166, pp. 1626 - 1643 [Scientific article]

V. González-Ruiz; M. Staderini; M. Bartolini; V. Andrisano; M. L. Bolognesi; N. Cabezas; J. C. Menéndez; A. I. Olives; M. A. Martína, XV International Symposium on Luminescence Spectrometry - Biophysical and Analytical Aspects, Extended Abstracts, 19-22 June 2012, Barcelona,Spain - (ISLS 2012), «LUMINESCENCE», 2012, 27, pp. 534 - 572 [Abstract]

F. Belluti; M. Bartolini; G. Bottegoni; A. Bisi; A. Cavalli; V. Andrisano; A. Rampa, Benzophenone-based derivatives: A novel series of potent and selective dual inhibitors of acetylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 1682 - 1693 [Scientific article]

F. Mancini; A. De Simone; V. Andrisano, Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors., «ANALYTICAL AND BIOANALYTICAL CHEMISTRY», 2011, 400, pp. 1979 - 1996 [Scientific article]

Bartolini M.; Pistolozzi M.; Andrisano V.; Egea J.; Lopez M.G.; Iriepa I.; Moraleda I.; Galvez E.; Marco-Contelles J.; Samadi A., Chemical and Pharmacological Studies on Enantiomerically Pure p-Methoxytacripyrines, Promising Multi-Target-Directed Ligands for the Treatment of Alzheimer's Disease, «CHEMMEDCHEM», 2011, 6, pp. 1990 - 1997 [Scientific article]

A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre, Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment, in: Atti del XXIV Congresso Nazionale della Società Chimica Italiana, LECCE, 2011 Università del Salento – Coordinamento SIBA-, 2011, pp. 434 - 435 (atti di: XXIV Congresso Nazionale della Società Chimica Italiana, Lecce, 11-16 settembre 2011) [Abstract]

M. Rosini; E. Simoni; M. Bartolini; A. Tarozzi; R. Matera; A. Milelli; P. Hrelia; V. Andrisano; M.L. Bolognesi; C. Melchiorre, Exploiting the lipoic acid structure in the search for novel multitarget ligands against Alzheimer's disease., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 5435 - 5442 [Scientific article]

M. Bartolini; M. Naldi; J. Fiori; F. Valle; F. Biscarini; D.V. Nicolau; V. Andrisano, Kinetic characterization of amyloid-beta 1-42 aggregation with a multimethodological approach., «ANALYTICAL BIOCHEMISTRY», 2011, 414, pp. 215 - 225 [Scientific article]

S. Rizzo; A. Bisi; M. Bartolini; F. Mancini; F. Belluti; S. Gobbi; V. Andrisano; A. Rampa, Multi-target strategy to address Alzheimer’s disease: Design, synthesis and biological evaluation of new tacrine-based dimers, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 4336 - 4343 [Scientific article]

Bolognesi M.L.; Bartolini M. ; Tarozzi A.; Morroni F. ; Lizzi F. ; Milelli A. ; Minarini A. ; Rosini M.; Hrelia P.; Andrisano V.; Melchiorre C., Multitargeted drugs discovery: Balancing anti-amyloid and anticholinesterase capacity in a single chemical entity, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2011, 21, pp. 2655 - 2658 [Scientific article]

Chiriano G.; Sartini A.; Mancini F.; Andrisano V.; Bolognesi M. L.; Roberti M.; Recanatini M.; Carloni P.; Cavalli A., Sequential Virtual Screening Approach to the Identification of Small Organic Molecules as Potential BACE-1 Inhibitors, «CHEMICAL BIOLOGY & DRUG DESIGN», 2011, 77, pp. 268 - 271 [Scientific article]

Martins C.; Carreiras M. C.; Leon R.; de Los Rios C.; Bartolini M.; Andrisano V.; Iriepa I.; Moraleda I.; Galvez E.; Garcia M.; Egea J.; Samadi A.; Chioua M.; Marco-Contelles J., Synthesis and biological assessment of diversely substituted furo[2,3-b]quinolin-4-amine and pyrrolo[2,3-b]quinolin-4-amine derivatives, as novel tacrine analogues, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2011, 46, pp. 6119 - 6130 [Scientific article]

Bolognesi ML; Chiriano G; Bartolini M; Mancini F; Bottegoni G; Maestri V; Czvitkovich S; Windisch M; Cavalli A; Minarini A; Rosini M; Tumiatti V; Andrisano V; Melchiorre C., Synthesis of Monomeric Derivatives To Probe Memoquin's Bivalent Interactions, «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 8299 - 82304 [Scientific article]

Vincenza Andrisano; Manuela Bartolini, 'Enzymes' immobilization on monolithic matrices: applications in drug discovery', in: PERRY G. WANG, Monolithic chromatography and its modern applications, ST ALBANS, HERTFORDSHIRE, UK, ILM Publications, 2010, pp. 403 - 425 [Chapter or essay]