Viayna, E.; Sola, I.; Bartolini, M.; De Simone, A.; Tapia-Rojas, C.; Carvajal, F. J.; Serrano, F. G.; Sabate, R.; Juárez, J.; Pérez, B.; Badia, A.; Luque, F. J.; Andrisano, V.; Clos, M. V.; Inestrosa, N. C.; Muñoz-Torrero, D. ., Synthesis, molecular modelling, in vitro biological profiling, and in vivo efficacy studies of a novel family of huprine-based multi-target anti-alzheimer compounds., in: XVII National Meeting of the Spanish Society of Medicinal Chemistry., 2013(atti di: XVII National Meeting of the Spanish Society of Medicinal Chemistry., Madrid, Spagna, 2-4 Ottobre 2013) [atti di convegno-poster]
M. Bartolini; V. Andrisano; A. De Simone; L. Zhang; Y. Lou; X. Zha, Tacrine-benzofunan hybrids as multi-target directed ligands for Alzheimer´s disease treatment, in: 11th International Conference on Alzheimer's and Parkinson's Diseases AD/PD 2013, 2013(atti di: 11th International Conference on Alzheimer's and Parkinson's Diseases (AD/PD), Firenze, 6-10 marzo 2013) [atti di convegno-poster]
Michela Rosini; Elena Simoni; Manuela Bartolini; Elena Soriano; José Marco-Contelles; Vincenza Andrisano; Barbara Monti; Manfred Windisch; Birgit Hutter-Paier; David W. McClymont; Ian R. Mellor; Maria Laura Bolognesi, The bivalent ligand approach as a tool for improving the in vitro anti-Alzheimer multitarget profile of dimebon, «CHEMMEDCHEM», 2013, 8, pp. 1276 - 1281 [articolo]
M. Bartolini; I. W. Wainer; C. Bertucci; V. Andrisano, The rapid and direct determination of ATPase activity by ion exchange chromatography and the application to the activity of heat shock protein-90, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2013, 73, pp. 77 - 81 [articolo]
Andrisano, V.; Seidl, C.; Santos, C.; De Simone, A.; Bartolini, M. ., Uleine an indole alkaloid from Himatanthus lancifolius as acetylcholinesterase, butyrylcholinesterase, beta-secretase and beta-amyloid(1-42) spontaneous aggregation inhibitor., in: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, 2013(atti di: 11th International Conference on Alzheimer's and Parkinson's Diseases, AD/ PD™ 2013, Florence, 6-10 Marzo 2013 .) [atti di convegno-poster]
G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A. Martinez; V. Andrisano; P. Carloni; M. Roberti, A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2012, 48, pp. 206 - 213 [articolo]
M. Bartolini; M. Naldi; D.V. Nicolau; F.C.M.J.M. van Delft; J. van Zijl; J. Snijder; F.C. van den Heuvel; V. Andrisano, ACETYLCHOLINESTERASE-BASED ANALYTICAL TOOLS FOR
DRUG SCREENING, in: Vth Conversatory on Medicinal Chemistry, LUBLIN, bestprint, 2012, pp. L-5 - L-5 (atti di: Vth Conversatory on Medicinal Chemistry - Book of Abstract, Lublin, 13-15 September 2012) [atti di convegno-abstract]
Naldi M.; Fiori J.; Pistolozzi M.; Drake A.F.; Bertucci C.; Wu R.; Mlynarczyk K.; Filipek S.; De Simone A.; Andrisano V., Amyloid beta-Peptide 25-35 Self Assembly and Its Inhibition: A Model Undecapeptide System to Gain Atomistic and Secondary Structure Details of the Alzheimer's Disease Process and Treatment, «ACS CHEMICAL NEUROSCIENCE», 2012, 3, pp. 952 - 962 [articolo]
Chlebek, Jakub; De Simone, Angela; Mancini, Francesca; Andrisano, Vincenza, An immobilized enzyme reactor based on human recombinant betasecretase (hrBACE-1-IMER) for the fast processing of substrates and screening of inhibitors, in: 21st National Meeting on Medicinal Chemistry NMMC 2012, 2012(atti di: 21st National Meeting on Medicinal Chemistry NMMC 2012, Palermo, 17-20 Luglio) [atti di convegno-poster]
Bartolini M.; Andrisano V, CHOLINESTERASE INHIBITION AS STARTING POINT FOR A MORE EFFECTIVE TREATMENT OF ALZHEIMER’S DISEASE, in: SINS 2012 - XIV Congress of the Italian Society for Neuroscience - 1st joint meeting with the Israel Society for Neuroscience - Program and abstract book, CATANIA, s.n, 2012, pp. 110 - 110 (atti di: SINS 2012 - XIV Congress of the Italian Society for Neuroscience - 1st joint meeting with the Israel Society for Neuroscience, Monastero dei Benedettini, Catania Italy, April 19th - 22nd, 2012) [atti di convegno-abstract]
De Simone, A; Mancini, F; Belluti, F; Bartolini, M; Bottegoni, G.; Rampa, A.; Cavalli, A.; Andrisano, V., Curcumin derivatives as beta-secretase (BACE1) inhibitors., in: Nuove Prospettive in Chimica Farmaceutica 6, 2012(atti di: Nuove Prospettive in Chimica Farmaceutica 6, Riccione, 11-13 Aprile) [atti di convegno-poster]
Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S., Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment., «NEUROPHARMACOLOGY», 2012, 62, pp. 997 - 1003 [articolo]
J. Fiori; M. Naldi; M. Bartolini; V. Andrisano, Disclosure of a fundamental clue for the elucidation of the myricetin mechanism of action as amyloid aggregation inhibitor by mass spectrometry, «ELECTROPHORESIS», 2012, 33, pp. 1 - 7 [articolo]
Galdeano C.; Viayna E.; Sola I.; Formosa X.; Camps P. Badia A.; Clos M.V.; Relat J.; Ratia M.; Bartolini M.; Mancini F.; Andrisano V.; Salmona M.; Minguillon C.; Gonzalez-Munoz G. C.; Rodriguez-Franco M. I.; Bidon-Chanal A.; Luque F. J.; Munoz-Torrero D., Huprine-tacrine heterodimers as anti-amyloidogenic compounds of potential interest against Alzheimer's and prion diseases, «JOURNAL OF MEDICINAL CHEMISTRY», 2012, 55, pp. 661 - 669 [articolo]
Kacker, Puneet; De Simone, Angela; Masetti, Matteo; Bottegoni, Giovanni; Andrisano, Vincenza; Cavalli, Andrea, Identification of Novel BACE-1 Inhibitors through an Advanced Structure-Based Virtual Screening Protocol., in: Structural & Computational Chemistry Congress, 2012(atti di: Structural & Computational Chemistry Congress, Munich, Germany, 13-14 March 2012) [atti di convegno-poster]
