Foto del docente

Silvia Gobbi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti, Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease, «ACS CHEMICAL NEUROSCIENCE», 2020, 11, pp. 2728 - 2740 [Scientific article]Open Access

Caciolla J.; Bisi A.; Belluti F.; Rampa A.; Gobbi S., Reconsidering Aromatase for Breast Cancer Treatment: New Roles for an Old Target, «MOLECULES», 2020, 25, pp. 5351 - 5351 [Scientific article]Open Access

Caciolla J.; Spinello A.; Martini S.; Bisi A.; Zaffaroni N.; Gobbi S.; Magistrato A., Targeting Orthosteric and Allosteric Pockets of Aromatase via Dual-Mode Novel Azole Inhibitors, «ACS MEDICINAL CHEMISTRY LETTERS», 2020, 11, pp. 732 - 739 [Scientific article]

Gobbi S.; Hu Q.; Foschi G.; Catanzaro E.; Belluti F.; Rampa A.; Fimognari C.; Hartmann R.W.; Bisi A., Benzophenones as xanthone-open model CYP11B1 inhibitors potentially useful for promoting wound healing, «BIOORGANIC CHEMISTRY», 2019, 86, pp. 401 - 409 [Scientific article]

Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolini M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A., Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 178, pp. 243 - 258 [Scientific article]Open Access

Bonvicini F.; Gentilomi G.A.; Bressan F.; Gobbi S.; Rampa A.; Bisi A.; Belluti F., Functionalization of the chalcone scaffold for the discovery of novel lead compounds targeting fungal infections, «MOLECULES», 2019, 24, Article number: 372 , pp. 372 - 397 [Scientific article]Open Access

Catanzaro E.; Seghetti F.; Calcabrini C.; Rampa A.; Gobbi S.; Sestili P.; Turrini E.; Maffei F.; Hrelia P.; Bisi A.; Belluti F.; Fimognari C., Identification of a new tamoxifen-xanthene hybrid as pro-apoptotic anticancer agent, «BIOORGANIC CHEMISTRY», 2019, 86, pp. 538 - 549 [Scientific article]

Bisi, Alessandra; Arribas, Raquel L.; Micucci, Matteo; Budriesi, Roberta; Feoli, Alessandra; Castellano, Sabrina; Belluti, Federica; Gobbi, Silvia; de los Rios, Cristobal; Rampa, Angela*, Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 163, pp. 394 - 402 [Scientific article]

Bisi A.; Mokhtar Mahmoud A.; Allara M.; Naldi M.; Belluti F.; Gobbi S.; Ligresti A.; Rampa A., Polycyclic Maleimide-based Scaffold as New Privileged Structure for Navigating the Cannabinoid System Opportunities, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 596 - 600 [Scientific article]

Bonvicini F.; Manet I.; Belluti F.; Gobbi S.; Rampa A.; Gentilomi G.A.; Bisi A., Targeting the Bacterial Membrane with a New Polycyclic Privileged Structure: A Powerful Tool To Face Staphylococcus aureus Infections, «ACS INFECTIOUS DISEASES», 2019, 5, pp. 1524 - 1534 [Scientific article]

Pavlin, Matic; Spinello, Angelo; Pennati, Marzia; Zaffaroni, Nadia; Gobbi, Silvia; Bisi, Alessandra; Colombo, Giorgio; Magistrato, Alessandra, A Computational Assay of Estrogen Receptor α Antagonists Reveals the Key Common Structural Traits of Drugs Effectively Fighting Refractory Breast Cancers, «SCIENTIFIC REPORTS», 2018, 8, Article number: 649 , pp. 1 - 11 [Scientific article]Open Access

Bisi, Alessandra*; Micucci, Matteo; Gobbi, Silvia; Belluti, Federica; Budriesi, Roberta; Rampa, Angela, Cardiovascular profile of xanthone-based 1,4 dihydropyridines bearing a lidoflazine pharmacophore fragment, «MOLECULES», 2018, 23, Article number: 3088 , pp. 1 - 14 [Scientific article]Open Access

Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease, «MOLECULES», 2018, 23, Article number: 1902 , pp. 1 - 22 [Scientific article]Open Access

Ortalli, Margherita; Ilari, Andrea; Colotti, Gianni; De Ionna, Ilenia; Battista, Theo; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Di Martino, Rita M.C.; Gentilomi, Giovanna A.; Varani, Stefania; Belluti, Federica*, Identification of chalcone-based antileishmanial agents targeting trypanothione reductase, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2018, 152, pp. 527 - 541 [Scientific article]Open Access

Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli, Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Chalcone-based carbamates for Alzheimer's disease treatment, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 749 - 764 [Scientific article]