Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J., Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 4035 - 4038 [articolo]
Bixel M.G.; Weise C.; Bolognesi M.L.; Rosini M.; Brierly M.J.; Mellor I.R.; Usherwood P.N.R.; Melchiorre C.; Hucho F., Location of the Polyamine Binding Site in the Vestibule of the Nicotinic Acetylcholine Receptor Ion Channel, «THE JOURNAL OF BIOLOGICAL CHEMISTRY», 2001, 276, pp. 6151 - 6160 [articolo]
D'Agostino G.; Bolognesi M.L.; Lucchelli A.; Vicini D.; Balestra B.; Spelta V.; Melchiorre C.; Tonini M., Prejunctional muscarinic inhibitory control of acetylcholine release in the human isolated detrusor: Involvement of the M4 receptor subtype, «BRITISH JOURNAL OF PHARMACOLOGY», 2000, 129, pp. 493 - 500 [articolo]
Bixel M.G.; Krauss M.; Liu Y.; Bolognesi M.L.; Rosini M.; Mellor I.S.; Usherwood P.N.R.; Melchiorre C.; Koji N.; Hucho F., Structure-activity relationship and site of binding of polyamine derivatives at the nicotinic acetylcholine receptor, «EUROPEAN JOURNAL OF BIOCHEMISTRY», 2000, 267, pp. 110 - 120 [articolo]
Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Marucci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V., α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety, «PHARMACEUTICA ACTA HELVETIAE», 2000, 74, pp. 181 - 190 [articolo]
Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C., Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 5212 - 5223 [articolo]
Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 4214 - 4224 [articolo]
Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Maggio R., Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor, «EUROPEAN JOURNAL OF PHARMACOLOGY», 1998, 355, pp. 267 - 274 [articolo]
Bolognesi M.L.; Budriesi R.; Chiarini A.; Poggesi E.; Leonardi A.; Melchiorre C., Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for α1-adrenoreceptor subtypes, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4844 - 4853 [articolo]
Melchiorre C.; Bolognesi M.L.; Budriesi R.; Chiarini A.; Giardina D.; Minarini A.; Quaglia W.; Leonardi A., Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?, «IL FARMACO», 1998, 53, pp. 278 - 286 [articolo]
Bolognesi M.L.; Minarini A.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Spampinato S.; Tumiatti V.; Melchiorre C., Universal template approach to drug design: Polyamines as selective muscarinic receptor antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4150 - 4160 [articolo]
Bolognesi M.; Ojala W.H.; Gleason W.B.; Griffin J.F.; Farouz-Grant F.; Larson D.L.; Takemori A.E.; Portoghese P.S., Opioid antagonist activity of naltrexone-derived bivalent ligands: Importance of a properly oriented molecular scaffold to guide "address" recognition at κ opioid receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1996, 39, pp. 1816 - 1822 [articolo]
Melchiorre C.; Angeli P.; Bolognesi M.L.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Crucianelli M.; Giardina D.; Gulini U.; Marucci G.; Minarini A.; Spampinato S.; Tumiatti V., Tetraamines as lead compounds for the design of neurotransmitter receptor ligands:Focus on α-adrenergic and muscarinic receptors recognition, «perspective in receptor research», 1996, 24, pp. 321 - 336 [articolo]
Chiarini A.; Budriesi R.; Bolognesi M.L.; Minarini A.; Melchiorre C., In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors, «BRITISH JOURNAL OF PHARMACOLOGY», 1995, 114, pp. 1507 - 1517 [articolo]
Recanatini M.; Tumiatti V.; Budriesi R.; Chiarini A.; Sabatino P.; Bolognesi M.L.; Melchiorre C., Synthesis, muscarinic blocking activity and molecular modeling studies of 4-DAMP-related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY», 1995, 3, pp. 267 - 277 [articolo]
