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Federico Falchi

Senior assistant professor (fixed-term)

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Falchi, Federico; Giacomini, Elisa; Masini, Tiziana; Boutard, Nicolas; Di Ianni, Lorenza; Manerba, Marcella; Farabegoli, Fulvia; Rossini, Lara; Robertson, Janet; Minucci, Saverio; Pallavicini, Isabella; Di Stefano, Giuseppina; Roberti, Marinella; Pellicciari, Roberto; Cavalli, Andrea, Synthetic Lethality Triggered by Combining Olaparib with BRCA2-Rad51 Disruptors, «ACS CHEMICAL BIOLOGY», 2017, 12, pp. 2491 - 2497 [Scientific article]

Falchi, Federico; Bertozzi, Sine Mandrup; Ottonello, Giuliana; Ruda, Gian Filippo; Colombano, Giampiero; Fiorelli, Claudio; Martucci, Cataldo; Bertorelli, Rosalia; Scarpelli, Rita; Cavalli, Andrea; Bandiera, Tiziano; Armirotti, Andrea, Kernel-Based, Partial Least Squares Quantitative Structure-Retention Relationship Model for UPLC Retention Time Prediction: A Useful Tool for Metabolite Identification, «ANALYTICAL CHEMISTRY», 2016, 88, pp. 9510 - 9517 [Scientific article]

Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [Scientific article]Open Access

Rupiani, Sebastiano; Guidotti, Laura; Manerba, Marcella; Di Ianni, Lorenza; Giacomini, Elisa; Falchi, Federico; Di Stefano, Giuseppina; Roberti, Marinella; Recanatini, Maurizio, Synthesis of natural urolithin M6, a galloflavin mimetic, as a potential inhibitor of lactate dehydrogenase A, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2016, 14, pp. 10981 - 10987 [Scientific article]

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Sebastiano Rupiani; Rosa Buonfiglio; Marcella Manerba; Lorenza Di Ianni; Marina Vettraino; Elisa Giacomini; Matteo Masetti; Federico Falchi; Giuseppina Di Stefano; Marinella Roberti; Maurizio Recanatini, Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitors, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2015, 101, pp. 63 - 70 [Scientific article]

Tintori C.; La Sala G.; Vignaroli G.; Botta L.; Fallacara A.L.; Falchi F.; Radi M.; Zamperini C.; Dreassi E.; Dello Iacono L.; Orioli D.; Biamonti G.; Garbelli M.; Lossani A.; Gasparrini F.; Tuccinardi T.; Laurenzana I.; Angelucci A.; Maga G.; Schenone S.; Brullo C.; Musumeci F.; Desogus A.; Crespan E.; Botta M., Studies on the ATP Binding Site of Fyn Kinase for the Identification of New Inhibitors and Their Evaluation as Potential Agents against Tauopathies and Tumors, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 4590 - 4609 [Scientific article]

Prati, Federica; Bergamini, Christian; Molina, Maria Teresa; Falchi, Federico; Cavalli, Andrea; Kaiser, Marcel; Brun, Reto; Fato, Romana; Bolognesi, Maria Laura, 2-Phenoxy-1,4-naphthoquinones: From a Multitarget Antitrypanosomal to a Potential Antitumor Profile, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 6422 - 6434 [Scientific article]

Giacomini E;Nebbioso A;Ciotta A;Ianni C;Falchi F;Roberti M;Tolomeo M;Grimaudo S;Cristina AD;Pipitone RM;Altucci L;Recanatini M, Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity., «ACS MEDICINAL CHEMISTRY LETTERS», 2014, 5, pp. 973 - 978 [Scientific article]

Patent n. WO/2014/187777, NOVEL INHIBITORS OF PVHL-ELONGIN C BINDING.

Matteo Masetti;Federico Falchi;Maurizio Recanatini, Protein Dynamics of the HIF-2α PAS-B Domain upon Heterodimerization and Ligand Binding, «PLOS ONE», 2014, 9, pp. e94986 - e94986 [Scientific article]Open Access

Federico Falchi;Fabiana Caporuscio;Maurizio Recanatini, Structure-based design of small-molecule protein–protein interaction modulators: the story so far, «FUTURE MEDICINAL CHEMISTRY», 2014, 6, pp. 343 - 357 [Scientific article]

R. Buonfiglio; M. Ferraro; F. Falchi; A. Cavalli; M. Masetti; M. Recanatini, Collecting and assessing human lactate dehydrogenase-A conformations for structure-based virtual screening, «JOURNAL OF CHEMICAL INFORMATION AND MODELING», 2013, 53, pp. 2792 - 2797 [Scientific article]

Tintori C.; Laurenzana I.; LaRocca F.; Falchi F.; Carraro F.; Ruiz A.; Este J.A.; Kissova M.; Crespan E.; Maga G.; Biava M.; Brullo C.; Schenone S.; Botta M., Identification of Hck Inhibitors As Hits for the Development of Antileukemia and Anti-HIV Agents, «CHEMMEDCHEM», 2013, 8, pp. 1353 - 1360 [Scientific article]

Radi M.; Evensen L.; Dreassi E.; Zamperini C.; Caporicci M.; Falchi F.; Musumeci F.; Schenone S.; Lorens J.B.; Botta M., A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: From in silico screening to cyclodextrin formulation, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2012, 22, pp. 5579 - 5583 [Scientific article]

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