Foto del docente

Alessandra Bisi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela, Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 6387 - 6406 [Scientific article]Open Access

Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [Scientific article]Open Access

Rampa, Angela; Tarozzi, Andrea; Mancini, Francesca; Pruccoli, Letizia; Di Martino, Rita Maria Concetta; Gobbi, Silvia; Bisi, Alessandra; De Simone, Angela; Palomba, Francesco; Zaccheroni, Nelsi; Belluti, Federica, Naturally inspired molecules as multifunctional agents for Alzheimer's disease treatment, «MOLECULES», 2016, 21, Article number: 643 , pp. 1 - 16 [Scientific article]Open Access

Gobbi, S; Hu, Q; Zimmer, C; Belluti, F; Rampa, A; Hartmann, Rw; Bisi, A., Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones, «CHEMMEDCHEM», 2016, 11, pp. 1770 - 1777 [Scientific article]

Di Martino, Rita Maria Concetta; De Simone, Angela; Andrisano, Vincenza; Bisignano, Paola; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Fato, Romana; Bergamini, Christian; Perez, Daniel I.; Martinez, Ana; Bottegoni, Giovanni; Cavalli, Andrea; Belluti, Federica, Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 531 - 544 [Scientific article]Open Access

Alessandra, Bisi; Silvia, Gobbi; Lucia, Merolle; Giovanna, Farruggia; Federica, Belluti; Angela, Rampa; Joseph, Molnar; Emil, Malucelli; Concettina, Cappadone, Design, synthesis and biological profile of new inhibitors of multidrug resistance associated proteins carrying a polycyclic scaffold, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2015, 92, pp. 471 - 480 [Scientific article]Open Access

Bisi Alessandra, Farmaci cardiaci, in: Chimica Farmaceutica, Milano, Casa Editrice Ambrosiana, 2015, pp. 404 - 424 [Chapter or essay]

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Gobbi S;Rampa A;Belluti F;Bisi A, Nonsteroidal aromatase inhibitors for the treatment of breast cancer: an update., «ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY», 2014, 14, pp. 54 - 65 [Scientific article]

A. Bisi;S. Gobbi;F. Belluti;A. Rampa, Design of Multifunctional Compounds for Cardiovascular Disease: From Natural Scaffolds to “Classical” Multitarget Approach, «CURRENT MEDICINAL CHEMISTRY», 2013, 20, pp. 1759 - 1782 [Scientific article]

Federica Belluti;Remo Perozzo;Leonardo Lauciello;Francesco Colizzi;Dirk Kostrewa;Alessandra Bisi;Silvia Gobbi;Angela Rampa;Maria Laura Bolognesi;Maurizio Recanatini;Reto Brun;Leonardo Scapozza;Andrea Cavalli, Design, Synthesis, and Biological and Crystallographic Evaluation of Novel Inhibitors ofPlasmodium falciparumEnoyl-ACP-reductase (PfFabI), «JOURNAL OF MEDICINAL CHEMISTRY», 2013, 56, pp. 7516 - 7526 [Scientific article]

Rampa A;Gobbi S;Belluti F;Bisi A, Emerging targets in neurodegeneration: new opportunities for Alzheimer's disease treatment?, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2013, 13, pp. 1879 - 1904 [Scientific article]

Silvia Gobbi;Qingzhong Hu;Matthias Negri;Christina Zimmer;Federica Belluti;Angela Rampa;Rolf W. Hartmann;Alessandra Bisi, Modulation of Cytochromes P450 with Xanthone-Based Molecules: From Aromatase to Aldosterone Synthase and Steroid 11β-Hydroxylase Inhibition, «JOURNAL OF MEDICINAL CHEMISTRY», 2013, 56, pp. 1723 - 1729 [Scientific article]

Rampa A; Bisi A, New approaches to the treatment of Alzheimer's disease., «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2013, 13, pp. 1743 - 1744 [Comment or similar]

Federica Belluti;Angela Rampa;Silvia Gobbi;Alessandra Bisi, Small-molecule inhibitors/modulators of amyloid-β peptide aggregation and toxicity for the treatment of Alzheimer's disease: a patent review (2010 – 2012), «EXPERT OPINION ON THERAPEUTIC PATENTS», 2013, 23, pp. 581 - 596 [Scientific article]