Foto del docente

Alessandra Bisi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Alessandra Bisi; Concettina Cappadone; Rampa Angela; Farruggia Giovanna; Sargenti Azzurra; Belluti Federica; Rita M.C. Di Martino; Malucelli, Emil; Meluzzi Alessia; Iotti Stefano; Silvia Gobbi, Coumarin derivatives as potential antitumor agents: Growth inhibition, apoptosis induction and multidrug resistance reverting activity, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 127, pp. 577 - 585 [Scientific article]

Gobbi, Silvia; Qingzhong, Hu; Zimmer, Christina; Belluti, Federica; Rampa, Angela; Hartmann, Rolf W.; Bisi, Alessandra, Drifting of heme-coordinating group in imidazolylmethylxanthones leading to improved selective inhibition of CYP11B1, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 139, pp. 60 - 67 [Scientific article]

Rampa, Angela; Gobbi, Silvia; Concetta Di Martino, Rita Maria; Belluti, Federica; Bisi, Alessandra, Dual BACE-1/GSK-3β Inhibitors To Combat Alzheimer's Disease: A Focused Review, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2017, 17, pp. 3361 - 3369 [Scientific article]

Di Martino, Rita Maria Concetta; Luppi, Barbara; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Abruzzo, Angela; Belluti, Federica, Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part I: Curcumin, «EXPERT OPINION ON THERAPEUTIC PATENTS», 2017, 27, pp. 579 - 590 [Scientific article]

Di Martino, Rita Maria Concetta; Bisi, Alessandra; Rampa, Angela; Gobbi, Silvia; Belluti, Federica, Recent progress on curcumin-based therapeutics: a patent review (2012-2016). Part II: curcumin derivatives in cancer and neurodegeneration, «EXPERT OPINION ON THERAPEUTIC PATENTS», 2017, 27, pp. 953 - 965 [Scientific article]

Gobbi, Silvia; Hu, Qingzhong; Zimmer, Christina; Engel, Matthias; Belluti, Federica; Rampa, Angela; Hartmann, Rolf W.; Bisi, Alessandra, Exploiting the Chromone Scaffold for the Development of Inhibitors of Corticosteroid Biosynthesis, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 2468 - 2477 [Scientific article]

Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela, Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 6387 - 6406 [Scientific article]Open Access

Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [Scientific article]Open Access

Rampa, Angela; Tarozzi, Andrea; Mancini, Francesca; Pruccoli, Letizia; Di Martino, Rita Maria Concetta; Gobbi, Silvia; Bisi, Alessandra; De Simone, Angela; Palomba, Francesco; Zaccheroni, Nelsi; Belluti, Federica, Naturally inspired molecules as multifunctional agents for Alzheimer's disease treatment, «MOLECULES», 2016, 21, Article number: 643 , pp. 1 - 16 [Scientific article]Open Access

Gobbi, S; Hu, Q; Zimmer, C; Belluti, F; Rampa, A; Hartmann, Rw; Bisi, A., Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones, «CHEMMEDCHEM», 2016, 11, pp. 1770 - 1777 [Scientific article]

Di Martino, Rita Maria Concetta; De Simone, Angela; Andrisano, Vincenza; Bisignano, Paola; Bisi, Alessandra; Gobbi, Silvia; Rampa, Angela; Fato, Romana; Bergamini, Christian; Perez, Daniel I.; Martinez, Ana; Bottegoni, Giovanni; Cavalli, Andrea; Belluti, Federica, Versatility of the Curcumin Scaffold: Discovery of Potent and Balanced Dual BACE-1 and GSK-3β Inhibitors, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 531 - 544 [Scientific article]Open Access

Alessandra, Bisi; Silvia, Gobbi; Lucia, Merolle; Giovanna, Farruggia; Federica, Belluti; Angela, Rampa; Joseph, Molnar; Emil, Malucelli; Concettina, Cappadone, Design, synthesis and biological profile of new inhibitors of multidrug resistance associated proteins carrying a polycyclic scaffold, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2015, 92, pp. 471 - 480 [Scientific article]Open Access

Bisi Alessandra, Farmaci cardiaci, in: Chimica Farmaceutica, Milano, Casa Editrice Ambrosiana, 2015, pp. 404 - 424 [Chapter or essay]

Angela, Rampa; Francesca, Mancini; Angela, De Simone; Federico, Falchi; Federica, Belluti; Rita Maria, Concetta Di Martino; Silvia, Gobbi; Vincenza, Andrisano; Andrea, Tarozzi; Manuela, Bartolini; Andrea, Cavalli; Alessandra, Bisi, From AChE to BACE1 inhibitors: The role of the amine on the indanone scaffold, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 2804 - 2808 [Scientific article]

Gobbi S;Rampa A;Belluti F;Bisi A, Nonsteroidal aromatase inhibitors for the treatment of breast cancer: an update., «ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY», 2014, 14, pp. 54 - 65 [Scientific article]