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Vincenzo Tumiatti

Professore ordinario

Dipartimento di Scienze per la Qualità della Vita

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Coordinatore del Corso di Laurea Magistrale a ciclo unico in Pharmacy

Pubblicazioni

Bolognesi M.L.; Marucci G.; Angeli P.; Buccioni M.; Minarini A.; Rosini M.; Tumiatti V.; Melchiorre C., Analogues of prazosin that bear a benextramine-related polyamine backbone exhibit different antagonism toward α1-adrenoreceptor subtypes, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 362 - 371 [articolo]

Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C., Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines, «BRITISH JOURNAL OF PHARMACOLOGY», 2001, 132, pp. 1009 - 1016 [articolo]Open Access

Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J., Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 4035 - 4038 [articolo]

Tumiatti V.; Wehrle J.; Hildebrandt C.; Moser U.; Dannhardt G.; Mutschler E.; Lambrecht G., Muscarinic properties of compounds related to arecaidine propargyl ester, «ARZNEIMITTEL-FORSCHUNG», 2000, 50, pp. 11 - 15 [articolo]

Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Marucci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V., α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety, «PHARMACEUTICA ACTA HELVETIAE», 2000, 74, pp. 181 - 190 [articolo]

Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C., Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 5212 - 5223 [articolo]

Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 4214 - 4224 [articolo]

Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Maggio R., Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor, «EUROPEAN JOURNAL OF PHARMACOLOGY», 1998, 355, pp. 267 - 274 [articolo]

Bolognesi M.L.; Minarini A.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Spampinato S.; Tumiatti V.; Melchiorre C., Universal template approach to drug design: Polyamines as selective muscarinic receptor antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4150 - 4160 [articolo]

Melchiorre C.; Angeli P.; Bolognesi M.L.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Crucianelli M.; Giardina D.; Gulini U.; Marucci G.; Minarini A.; Spampinato S.; Tumiatti V., Tetraamines as lead compounds for the design of neurotransmitter receptor ligands:Focus on α-adrenergic and muscarinic receptors recognition, «perspective in receptor research», 1996, 24, pp. 321 - 336 [articolo]

Melchiorre C.; Minarini A.; Spampinato S.; Tumiatti V., Design, synthesis and biological activity of some tetraamines related to methoctramine and 4-DAMP, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 785 - 790 [articolo]

Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R., Design, synthesis and biological activity of some 4-DAMP- related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 2325 - 2330 [articolo]

Recanatini M.; Tumiatti V.; Budriesi R.; Chiarini A.; Sabatino P.; Bolognesi M.L.; Melchiorre C., Synthesis, muscarinic blocking activity and molecular modeling studies of 4-DAMP-related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY», 1995, 3, pp. 267 - 277 [articolo]

Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V., The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists, «LIFE SCIENCES», 1995, 56, pp. 837 - 844 [articolo]

Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L., Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP, «IL FARMACO», 1992, 47, pp. 1133 - 1147 [articolo]