Foto del docente

Roberta Budriesi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/10 Food Chemistry

Publications

Bisi A.; Budriesi R.; Rampa A.; Fabbri G.; Chiarini A.; Valenti P., Synthesis and pharmacological profile of some chloroxanthone-1,4-dihydropyridine derivatives, «ARZNEIMITTEL-FORSCHUNG», 1996, 46, pp. 848 - 851 [Scientific article]

Melchiorre C.; Angeli P.; Bolognesi M.L.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Crucianelli M.; Giardina D.; Gulini U.; Marucci G.; Minarini A.; Spampinato S.; Tumiatti V., Tetraamines as lead compounds for the design of neurotransmitter receptor ligands:Focus on α-adrenergic and muscarinic receptors recognition, «perspective in receptor research», 1996, 24, pp. 321 - 336 [Scientific article]

Chiarini A.; Rampa A.; Budriesi R.; Bisi A.; Fabbri G.; Valenti P., 1,4-Dihydropyridine bearing a pharmacophoric fragment of lidoflazine, «BIOORGANIC & MEDICINAL CHEMISTRY», 1996, 4, pp. 1629 - 1635 [Scientific article]

Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R., Design, synthesis and biological activity of some 4-DAMP- related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 2325 - 2330 [Scientific article]

Chiarini A.; Budriesi R.; Bolognesi M.L.; Minarini A.; Melchiorre C., In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors, «BRITISH JOURNAL OF PHARMACOLOGY», 1995, 114, pp. 1507 - 1517 [Scientific article]

Campiani G.; Garofalo A.; Fiorini I.; Botta M.; Nacci V.; Tafi A.; Chiarini A.; Budriesi R.; Bruni G.; Romeo M.R., Pyrrolo[2,1-c][1,4]benzothiazines: Synthesis, Structure-Activity Relationships, Molecular Modeling Studies, and Cardiovascular Activity, «JOURNAL OF MEDICINAL CHEMISTRY», 1995, 38, pp. 4393 - 4410 [Scientific article]

Rampa A.; Budriesi R.; Bisi A.; Fabbri G.; Barili P.L.; Chiarini A.; Valenti P., Structure-activity relationship studies in the field of calcium antagonists. Xanthone 1,4-dihydropyridines bearing a 2,3-lactone ring, «ARZNEIMITTEL-FORSCHUNG», 1995, 45, pp. 957 - 962 [Scientific article]

Budriesi R.; Rampa A.; Bisi A.; Fabbri G.; Chiarini A.; Valenti P., Synthesis and pharmacological characterization of some benzazepinone derivatives, «ARZNEIMITTEL-FORSCHUNG», 1995, 45, pp. 234 - 239 [Scientific article]

Recanatini M.; Tumiatti V.; Budriesi R.; Chiarini A.; Sabatino P.; Bolognesi M.L.; Melchiorre C., Synthesis, muscarinic blocking activity and molecular modeling studies of 4-DAMP-related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY», 1995, 3, pp. 267 - 277 [Scientific article]

Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V., The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists, «LIFE SCIENCES», 1995, 56, pp. 837 - 844 [Scientific article]

Gasco A.M.; Ermondi G.; Gasco A.; Budriesi R.; Chiarini A., 1,4-Dihydropyridines containing R-NNO-azoxy moieties, «IL FARMACO», 1995, 50, pp. 61 - 64 [Scientific article]

Minarini A.; Bolognesi M.L.; Budriesi R.; Canossa M.; Chiarini A.; Spampinato S.; Melchiorre C., Design, Synthesis, and Biological Activity of Methoctramine-Related Tetraamines Bearing an 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Moiety: Structural Requirements for Optimum Occupancy of Muscarinic Receptor Subtypes As Revealed by Symmetrical and Unsymmetrical Polyamines, «JOURNAL OF MEDICINAL CHEMISTRY», 1994, 37, pp. 3363 - 3372 [Scientific article]

Romanelli M.N.; Dei S.; Scapecchi S.; Teodori E.; Gualtieri F.; Budriesi R.; Mannhold R., Semi-rigid analogues of the calcium antagonist verapamil: A molecular modelling study, «JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN», 1994, 8, pp. 123 - 134 [Scientific article]

Campiani G.; Garofalo A.; Fiorini I.; Nacci V.; Botta M.; Tafi A.; Chiarini A.; Budriesi R.; Bruni G.; Romeo M.R., Synthesis and "in vitro" cardiovascular activity of 4-aryl-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,4]benzothiazin-1-ones and 7-acetoxy-6-phenyl-7a,8,9,10-tetrahydropyrrolo [2,1,-d][1,5]benzothiazepin-10-one, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1994, 4, pp. 1235 - 1240 [Scientific article]

Teodori E.; Dei S.; Romanelli M.; Scapecchi S.; Gualtieri F.; Budriesi R.; Chiarini A.; Lemoine H.; Mannhold R., Synthesis and pharmacological evaluation of verapamil analogs with restricted molecular flexibility, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 1994, 29, pp. 139 - 148 [Scientific article]

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