Budriesi R.; Cacciaguerra S.; Di Toro R.; Bolognesi M.L.; Chiarini A.; Minarini A.; Rosini M.; Spampinato S.; Tumiatti V.; Melchiorre C., Analysis of the muscarinic receptor subtype mediating inhibition of the neurogenic contractions in rabbit isolated vas deferens by a series of polymethylene tetra-amines, «BRITISH JOURNAL OF PHARMACOLOGY», 2001, 132, pp. 1009 - 1016 [Scientific article]Open Access
Melchiorre C.; Bolognesi M.L.; Budriesi R.; Ghelardini C.; Chiarini A.; Minarini A.; Rosini M.; Tumiatti V.; Wade E.J., Design, synthesis, and biological activity of methoctramine-related polyamines as putative Gi protein activators, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 4035 - 4038 [Scientific article]
Teodori E.; Dei S.; Garnier-Suillerot A.; Quidu P.; Scapecchi S.; Budriesi R., Structure-activity relationship studies on the potent multidrug resistance (MDR) modulator 2-(3,4-dimethoxyphenyl)-2-(methylethyl)-5[(anthr-9-yl) methylamino]pentanenitrile (MM 36), «MEDICINAL CHEMISTRY RESEARCH», 2001, 10, pp. 563 - 576 [Scientific article]
Dei S.; Teodori E.; Garnier-Suillerot A.; Gualtieri F.; Scapecchi S.; Budriesi R.; Chiarini A., Structure-activity relationships and optimisation of the selective MDR modulator 2-(3,4-dimethoxyphenyl)-5-(9-fluorenylamino)-2-(methylethyl) pentanenitrile and its N-methyl derivative, «BIOORGANIC & MEDICINAL CHEMISTRY», 2001, 9, pp. 2673 - 2682 [Scientific article]
Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C., Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 5212 - 5223 [Scientific article]
Teodori E.; Dei S.; Quidu P.; Budriesi R.; Chiarini A.; Garnier-Suillerot A.; Gualtieri F.; Manetti D.; Romanelli M.N.; Scapecchi S., Design, synthesis, and in vitro activity of catamphiphilic reverters of multidrug resistance: Discovery of a selective, highly efficacious chemosensitizer with potency in the nanomolar range, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 1687 - 1697 [Scientific article]
Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 4214 - 4224 [Scientific article]
Valenti P.; Rampa A.; Budriesi R.; Bisi A.; Chiarini A., Coumarin 1,4-dihydropyridine derivatives, «BIOORGANIC & MEDICINAL CHEMISTRY», 1998, 6, pp. 803 - 810 [Scientific article]
Bolognesi M.L.; Budriesi R.; Chiarini A.; Poggesi E.; Leonardi A.; Melchiorre C., Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for α1-adrenoreceptor subtypes, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4844 - 4853 [Scientific article]
Melchiorre C.; Bolognesi M.L.; Budriesi R.; Chiarini A.; Giardina D.; Minarini A.; Quaglia W.; Leonardi A., Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?, «IL FARMACO», 1998, 53, pp. 278 - 286 [Scientific article]
Minarini A.; Budriesi R.; Chiarini A.; Leonardi A.; Melchiorre C., Search for α1-adrenoceptor subtypes selective antagonists: Design, synthesis and biological activity of cystazosin, an α(1D)-adrenoceptor antagonist, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1998, 8, pp. 1353 - 1358 [Scientific article]
Bolognesi M.L.; Minarini A.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Spampinato S.; Tumiatti V.; Melchiorre C., Universal template approach to drug design: Polyamines as selective muscarinic receptor antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4150 - 4160 [Scientific article]
Campiani G.; Fiorini I.; De Filippis M.P.; Ciani S.M.; Garofalo A.; Nacci V.; Giorgi G.; Sega A.; Botta M.; Chiarini A.; Budriesi R.; Bruni G.; Romeo M.R.; Manzoni C.; Mennini T., Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepine derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): From dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers, «JOURNAL OF MEDICINAL CHEMISTRY», 1996, 39, pp. 2922 - 2938 [Scientific article]
Budriesi R.; Rampa A.; Bisi A.; Fabbri G.; Chiarini A.; Valenti P., Structure-activity relationship studies of xanthone and fluorenone-1,4-dihydropyridine-5-phosphonates, «ARZNEIMITTEL-FORSCHUNG», 1996, 46, pp. 374 - 377 [Scientific article]
Varoli L.; Burnelli S.; Budriesi R.; Guarnieri A.; Chiarini A.; Recanatini M., Synthesis and biological profile at muscarinic M2 and M3 receptor subtypes of some analogs of diphenidol, «MEDICINAL CHEMISTRY RESEARCH», 1996, 6, pp. 571 - 580 [Scientific article]
