Codony S.; Pont C.; Grinan-Ferre C.; Di Pede-Mattatelli A.; Calvo-Tusell C.; Feixas F.; Osuna S.; Jarne-Ferrer J.; Naldi M.; Bartolini M.; Loza M.I.; Brea J.; Perez B.; Bartra C.; Sanfeliu C.; Juarez-Jimenez J.; Morisseau C.; Hammock B.D.; Pallas M.; Vazquez S.; Munoz-Torrero D., Discovery and in Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 4909 - 4925 [Scientific article]Open Access
Parenti, Md; Naldi, M; Manoni, E; Fabini, E; Cederfelt, D; Talibov, Vo; Gressani, V; Guven, U; Grossi, V; Fasano, C; Sanese, P; De Marco, K; Shtil, Aa; Kurkin, Av; Altieri, A; Danielson, Uh; Caretti, G; Simone, C; Varchi, G; Bartolini, M; Del Rio, A, Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2022, 243, pp. 114683 - 114695 [Scientific article]Open Access
Rapozzi V.; Moret F.; Menilli L.; Guerrini A.; Tedesco D.; Naldi M.; Bartolini M.; Gani M.; Zorzet S.; Columbaro M.; Milani C.; Martini C.; Ferroni C.; Varchi G., HSA-Binding Prodrugs-Based Nanoparticles Endowed with Chemo and Photo-Toxicity against Breast Cancer, «CANCERS», 2022, 14, Article number: 877 , pp. 877 - 902 [Scientific article]Open Access
Basagni, Filippo; Naldi, Marina; Ginex, Tiziana; Luque, F Javier; Fagiani, Francesca; Lanni, Cristina; Iurlo, Matteo; Marcaccio, Massimo; Minarini, Anna; Bartolini, Manuela; Rosini, Michela, Inhibition of β-Amyloid Aggregation in Alzheimer's Disease: The Key Role of (Pro)electrophilic Warheads, «ACS MEDICINAL CHEMISTRY LETTERS», 2022, 13, pp. 1812 - 1818 [Scientific article]Open Access
Naldi M.; Brusotti G.; Massolini G.; Andrisano V.; Temporini C.; Bartolini M., Bio-guided fractionation of stem bark extracts from phyllanthus muellarianus: Identification of phytocomponents with anti-cholinesterase activity, «MOLECULES», 2021, 26, Article number: 4376 , pp. 4376-1 - 4376-14 [Scientific article]Open Access
Baldassarre M.; Naldi M.; Zaccherini G.; Bartoletti M.; Antognoli A.; Laggetta M.; Gagliardi M.; Tufoni M.; Domenicali M.; Waterstradt K.; Paterini P.; Baldan A.; Leoni S.; Bartolini M.; Viale P.; Trevisani F.; Bernardi M.; Caraceni P., Determination of Effective Albumin in Patients With Decompensated Cirrhosis: Clinical and Prognostic Implications, «HEPATOLOGY», 2021, 74, pp. 2058 - 2073 [Scientific article]Open Access
Talibov, Vladimir O; Fabini, Edoardo; FitzGerald, Edward A; Tedesco, Daniele; Cederfeldt, Daniela; Talu, Martin J; Rachman, Moira M; Mihalic, Filip; Manoni, Elisabetta; Naldi, Marina; Sanese, Paola; Forte, Giovanna; Lepore Signorile, Martina; Barril, Xavier; Simone, Cristiano; Bartolini, Manuela; Dobritzsch, Doreen; Del Rio, Alberto; Danielson, U Helena, Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase, «CHEMBIOCHEM», 2021, 22, pp. 1597 - 1608 [Scientific article]Open Access
Ramos, Gd; De Oliveira, As; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L; Fraser, Pe; Abreu, M; Kiametis, As; Gargano, R; Silveira, Er; Brand, Gd; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, Ml; Romeiro, Las, Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties, «RSC MEDICINAL CHEMISTRY», 2021, 12, pp. 1154 - 1163 [Scientific article]Open Access
Albertini C.; Naldi M.; Petralla S.; Strocchi S.; Grifoni D.; Monti B.; Bartolini M.; Bolognesi M.L., From combinations to single-molecule polypharmacology—cromolyn-ibuprofen conjugates for alzheimer’s disease, «MOLECULES», 2021, 26, Article number: 1112 , pp. 1 - 22 [Scientific article]Open Access
Pont, C.; Ginex, T.; Grinan-Ferre, C.; Scheiner, M.; Mattellone, A.; Martinez, N.; Arce, E. M.; Soriano-Fernandez, Y.; Naldi, M.; De Simone, A.; Barenys, M.; Gomez-Catalan, J.; Perez, B.; Sabate, R.; Andrisano, V.; Loza, M. I.; Brea, J.; Bartolini, M.; Bolognesi, M. L.; Decker, M.; Pallas, M.; Luque, F. J.; Munoz-Torrero, D., From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2021, 225, Article number: 113779 , pp. 1 - 25 [Scientific article]Open Access
Montanari S.; Allara M.; Scalvini L.; Kostrzewa M.; Belluti F.; Gobbi S.; Naldi M.; Rivara S.; Bartolini M.; Ligresti A.; Bisi A.; Rampa A., New Coumarin derivatives as cholinergic and cannabinoid system modulators, «MOLECULES», 2021, 26, Article number: 3254 , pp. 1 - 18 [Scientific article]Open Access
De Simone, A.; Naldi, M.; Tedesco, D.; Bartolini, M.; Davani, L.; Andrisano, V., Advanced analytical methodologies in Alzheimer's disease drug discovery, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2020, 178, Article number: 112899 , pp. 1 - 25 [Scientific article]Open Access
Cieslikiewicz-Bouet, Monika; Naldi, Marina; Bartolini, Manuela; Pérez, Belén; Servent, Denis; Jean, Ludovic; Aráoz, Rómulo; Renard, Pierre-Yves, Functional characterization of multifunctional ligands targeting acetylcholinesterase and alpha 7 nicotinic acetylcholine receptor, «BIOCHEMICAL PHARMACOLOGY», 2020, 177, Article number: 114010 , pp. 1 - 11 [Scientific article]Open Access
Palmerini, Tullio; Barozzi, Chiara; Tomasi, Luciana; Riva, Diego Della; Marengo, Mario; Cicoria, Gianfranco; Bruno, Antonio G.; Bacchi-Reggiani, Maria-Letizia; Naldi, Marina; Bartolini, Manuela; Fanti, Stefano; Galiè, Nazzareno; Stone, Gregg W., In vitro thrombogenicity of drug-eluting and bare metal stents, «THROMBOSIS RESEARCH», 2020, 185, pp. 43 - 48 [Scientific article]
Verardi L.; Fiori J.; Andrisano V.; Locatelli A.; Morigi R.; Naldi M.; Bertucci C.; Strocchi E.; Boga C.; Micheletti G.; Calonghi N., Indole derivative interacts with estrogen receptor beta and inhibits human ovarian cancer cell growth, «MOLECULES», 2020, 25, Article number: 4438 , pp. 1 - 15 [Scientific article]Open Access