Foto del docente

Maria Laura Bolognesi

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Coordinator of PhD Programme in Biotechnological, Biocomputational, Pharmaceutical and Pharmacological Sciences

Publications

M. Staderini; N. Cabezas; M. L. Bolognesi; J. Carlos Menéndez, Solvent- and chromatography-free amination of pi-deficient nitrogen heterocycles under microwave irradiation. A fast, efficient and green route to 9-aminoacridines, 4-aminoquinolines and 4-aminoquinazolines and its application to the synthesis of the drugs amsacrine and bistacrine, «TETRAHEDRON», 2013, 69, pp. 1024 - 1030 [Scientific article]

Michela Rosini; Elena Simoni; Manuela Bartolini; Elena Soriano; José Marco-Contelles; Vincenza Andrisano; Barbara Monti; Manfred Windisch; Birgit Hutter-Paier; David W. McClymont; Ian R. Mellor; Maria Laura Bolognesi, The bivalent ligand approach as a tool for improving the in vitro anti-Alzheimer multitarget profile of dimebon, «CHEMMEDCHEM», 2013, 8, pp. 1276 - 1281 [Scientific article]

G. P. Chiriano; A. De Simone; F. Mancini; D. I. Perez; A. Cavalli; M. L. Bolognesi; G. Legname; A. Martinez; V. Andrisano; P. Carloni; M. Roberti, A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: structure-based design, synthesis, and biological evaluation, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2012, 48, pp. 206 - 213 [Scientific article]

M. L. Bolognesi, Conjugation of quinones with natural polyamines does expand their anti-trypanosomatid profile, in: COST-CM0801: WG1/WG3 Meeting : New Drugs for Neglected Diseases : book of Abstracts, s.l, s.n, 2012, pp. 12 - 12 (atti di: COST-CM0801: WG1/WG3 Meeting : New Drugs for Neglected Diseases, Certosa Di Pontignano, Siena, 31st May - 1st June 2012) [Abstract]

F. Lizzi; G. Veronesi; F. Belluti; C. Bergamini; A. López-Sánchez; M. Kaiser; R. Brun; R. L. Krauth-Siegel; D. G. Hall; L. Rivas; M. L. Bolognesi, Conjugation of Quinones with Natural Polyamines: Toward an Expanded Antitrypanosomatid Profile, «JOURNAL OF MEDICINAL CHEMISTRY», 2012, 55, pp. 10490 - 10500 [Scientific article]

Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Simoni E.; Bolognesi M.L.; Andrisano V.; Bartolini M.; Motori E.; Angeloni C.; Hrelia S., Cystamine-tacrine dimer: A new multi-target-directed ligand as potential therapeutic agent for Alzheimer's disease treatment., «NEUROPHARMACOLOGY», 2012, 62, pp. 997 - 1003 [Scientific article]

Bolognesi; M.L.; Melchiorre; C.; Van der Schyf; C.J.; and Youdim; M.B.H, Discovery of Multi-Target Agents for Neurological Diseases via Ligand Design, in: Designing Multi-Target Drugs, CAMBRIDGE, Royal Society of Chemistry, 2012, pp. 290 - 315 [Chapter or essay]

M. L. Bolognesi, Discovery of multi-target probes for neurodegenerative diseases via ligand design, in: Abstract Book, Basel, September 24-27 2012MipTec and Biovalley Life sciences week, s.l, s.n, 2012, pp. 37 - 37 (atti di: MipTec 2012, Basel, September 24-27 2012) [Abstract]

Cavalli A.; Bolognesi M.L., Multitargeted drugs for the treatment of Alzheimer's disease, in: Polypharmacology in drug discovery, HOBOKEN, Wiley, 2012, pp. 441 - 458 [Chapter or essay]

Simoni E.; Rosini M.; Bartolini M.; Andrisano V.; Soriano E.; Marco-Contelles J.; Melchiorre C.; Bolognesi M.L., Rational design of dimebon bivalent ligands against Alzheimer’s disease, in: Libro degli abstracts, s.l, s.n, 2012, pp. 38 - 38 (atti di: NPCF6-Nuove prospettive in chimica farmaceutica- 6°Meeting, Riccione, 15-17 aprile 2012) [Abstract]

M. L. Bolognesi, Styrylquinolines as amyloid chemical probes and theranostics in Alzheimer’s and prion diseases, in: COST Conference - Personalised Medicine: Better Healthcare for the Future, s.l, s.n, 2012, pp. 36 - 36 (atti di: Personalised Medicine: Better Healthcare for the Future - A Rational Approach Focusing on Bioinformatics, Medicinal Chemistry and Medicine, Larnaca, 17 - 22 June 2012) [Abstract]

Gamberini MT; Bolognesi ML; Nasello AG, The modulatory role of M2 muscarinic receptor on apomorphine-induced yawning and genital grooming, «NEUROSCIENCE LETTERS», 2012, 531, pp. 91 - 95 [Scientific article]

V. González-Ruiz; M. Staderini; M. Bartolini; V. Andrisano; M. L. Bolognesi; N. Cabezas; J. C. Menéndez; A. I. Olives; M. A. Martína, XV International Symposium on Luminescence Spectrometry - Biophysical and Analytical Aspects, Extended Abstracts, 19-22 June 2012, Barcelona,Spain - (ISLS 2012), «LUMINESCENCE», 2012, 27, pp. 534 - 572 [Abstract]

Staderini Matteo; Cabezas Nieves; Bolognesi Maria Laura; Menéndez J. Carlos, A General Protocol for the Solvent- and Catalyst-Free Synthesis of 2-Styrylquinolines under Focused Microwave Irradiation, «SYNLETT», 2011, 17, pp. 2577 - 2579 [Scientific article]

A. Minarini; A. Milelli; V. Tumiatti; E. Simoni; M. L. Bolognesi; V. Andrisano; M. Bartolini; E. Motori; C. Angeloni ; S. Hrelia; C.Melchiorre, Cystamine-tacrine dimer: a new multi-target-directed ligand as potential therapeutic agent for Alzheimer’s disease treatment, in: Atti del XXIV Congresso Nazionale della Società Chimica Italiana, LECCE, 2011 Università del Salento – Coordinamento SIBA-, 2011, pp. 434 - 435 (atti di: XXIV Congresso Nazionale della Società Chimica Italiana, Lecce, 11-16 settembre 2011) [Abstract]