Foto del docente

Manuela Bartolini

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHEM-07/A Chimica farmaceutica

Pubblicazioni

Talibov, Vladimir O; Fabini, Edoardo; FitzGerald, Edward A; Tedesco, Daniele; Cederfeldt, Daniela; Talu, Martin J; Rachman, Moira M; Mihalic, Filip; Manoni, Elisabetta; Naldi, Marina; Sanese, Paola; Forte, Giovanna; Lepore Signorile, Martina; Barril, Xavier; Simone, Cristiano; Bartolini, Manuela; Dobritzsch, Doreen; Del Rio, Alberto; Danielson, U Helena, Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase, «CHEMBIOCHEM», 2021, 22, pp. 1597 - 1608 [articolo]Open Access

Ramos, Gd; De Oliveira, As; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L; Fraser, Pe; Abreu, M; Kiametis, As; Gargano, R; Silveira, Er; Brand, Gd; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, Ml; Romeiro, Las, Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties, «RSC MEDICINAL CHEMISTRY», 2021, 12, pp. 1154 - 1163 [articolo]Open Access

Albertini C.; Naldi M.; Petralla S.; Strocchi S.; Grifoni D.; Monti B.; Bartolini M.; Bolognesi M.L., From combinations to single-molecule polypharmacology—cromolyn-ibuprofen conjugates for alzheimer’s disease, «MOLECULES», 2021, 26, Article number: 1112, pp. 1 - 22 [articolo]Open Access

Pont, C.; Ginex, T.; Grinan-Ferre, C.; Scheiner, M.; Mattellone, A.; Martinez, N.; Arce, E. M.; Soriano-Fernandez, Y.; Naldi, M.; De Simone, A.; Barenys, M.; Gomez-Catalan, J.; Perez, B.; Sabate, R.; Andrisano, V.; Loza, M. I.; Brea, J.; Bartolini, M.; Bolognesi, M. L.; Decker, M.; Pallas, M.; Luque, F. J.; Munoz-Torrero, D., From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2021, 225, Article number: 113779, pp. 1 - 25 [articolo]Open Access

Montanari S.; Allara M.; Scalvini L.; Kostrzewa M.; Belluti F.; Gobbi S.; Naldi M.; Rivara S.; Bartolini M.; Ligresti A.; Bisi A.; Rampa A., New Coumarin derivatives as cholinergic and cannabinoid system modulators, «MOLECULES», 2021, 26, Article number: 3254, pp. 1 - 18 [articolo]Open Access

Gorecki L.; Uliassi E.; Bartolini M.; Janockova J.; Hrabinova M.; Hepnarova V.; Prchal L.; Muckova L.; Pejchal J.; Karasova J.Z.; Mezeiova E.; Benkova M.; Kobrlova T.; Soukup O.; Petralla S.; Monti B.; Korabecny J.; Bolognesi M.L., Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2021, 12, pp. 1698 - 1715 [articolo]Open Access

Rossi, M; Freschi, M; de Camargo Nascente, L; Salerno, A; de Melo Viana Teixeira, S; Nachon, F; Chantegreil, F; Soukup, O; Prchal, L; Malaguti, M; Bergamini, C; Bartolini, M; Angeloni, C; Hrelia, S; Soares Romeiro, La; Bolognesi, Ml., Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease, «JOURNAL OF MEDICINAL CHEMISTRY», 2021, 64, pp. 4972 - 4990 [articolo]Open Access

Perone, R.; Albertini, C.; Uliassi, E.; Di Pietri, F.; de Sena Murteira Pinheiro, P.; Petralla, S.; Rizzardi, N.; Fato, R.; Pulkrabkova, L.; Soukup, O.; Tramarin, A.; Bartolini, M.; Bolognesi, M. L., Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy, «CHEMMEDCHEM», 2021, 16, pp. 187 - 198 [articolo]Open Access

De Simone, A.; Naldi, M.; Tedesco, D.; Bartolini, M.; Davani, L.; Andrisano, V., Advanced analytical methodologies in Alzheimer's disease drug discovery, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2020, 178, Article number: 112899, pp. 1 - 25 [articolo]Open Access

Pérez-Areales, F Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer, Angel; Muñoz-Torrero, Diego, Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6, «JOURNAL OF MEDICINAL CHEMISTRY», 2020, 63, pp. 9360 - 9390 [articolo]Open Access

Guzman, Laura; Besa, Gisela; Linares, Daniela; González, Lara; Pont, Caterina; Bartolini, Manuela; Haigis, Ann-Cathrin; Legradi, Jessica; Muñoz-Torrero, Diego; Gómez-Catalán, Jesús; Barenys, Marta, Evaluation of the effects of acetylcholinesterase inhibitors in the zebrafish touch-evoked response: quantitative vs. qualitative assessment, «ENVIRONMENTAL SCIENCES EUROPE», 2020, 32, Article number: 145, pp. 1 - 12 [articolo]Open Access

Cieslikiewicz-Bouet, Monika; Naldi, Marina; Bartolini, Manuela; Pérez, Belén; Servent, Denis; Jean, Ludovic; Aráoz, Rómulo; Renard, Pierre-Yves, Functional characterization of multifunctional ligands targeting acetylcholinesterase and alpha 7 nicotinic acetylcholine receptor, «BIOCHEMICAL PHARMACOLOGY», 2020, 177, Article number: 114010, pp. 1 - 11 [articolo]Open Access

Palmerini, Tullio; Barozzi, Chiara; Tomasi, Luciana; Riva, Diego Della; Marengo, Mario; Cicoria, Gianfranco; Bruno, Antonio G.; Bacchi-Reggiani, Maria-Letizia; Naldi, Marina; Bartolini, Manuela; Fanti, Stefano; Galiè, Nazzareno; Stone, Gregg W., In vitro thrombogenicity of drug-eluting and bare metal stents, «THROMBOSIS RESEARCH», 2020, 185, pp. 43 - 48 [articolo]

Bua G.; Tedesco D.; Conti I.; Reggiani A.; Bartolini M.; Gallinella G., No G-Quadruplex Structures in the DNA of Parvovirus B19: Experimental Evidence versus Bioinformatic Predictions, «VIRUSES», 2020, 12, Article number: 935, pp. 935 - 935 [articolo]Open Access

Marques C.S.; Lopez O.; Bagetta D.; Carreiro E.P.; Petralla S.; Bartolini M.; Hoffmann M.; Alcaro S.; Monti B.; Bolognesi M.L.; Decker M.; Fernandez-Bolanos J.G.; Burke A.J., N-1,2,3-triazole-isatin derivatives for cholinesterase and β-amyloid aggregation inhibition: A comprehensive bioassay study, «BIOORGANIC CHEMISTRY», 2020, 98, Article number: 103753, pp. 103753 - 103765 [articolo]