Foto del docente

Luca Gentilucci

Professore associato confermato

Dipartimento di Chimica "Giacomo Ciamician"

Settore scientifico disciplinare: CHIM/06 CHIMICA ORGANICA

Pubblicazioni

Gentilucci L.; Cardillo G. ; Squassabia F.; Tolomelli A.; Spampinato S.; Sparta A.; Baiula M., Inhibition of cancer cell adhesion by heterochiral Pro-containing RGD mimetics., «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2007, 17, pp. 2329 - 2333 [articolo]

L. Gentilucci; F. Squassabia; R. Artali, Re-discussion of the importance of ionic interactions in stabilizing ligand-opioid receptor complex and in activating signal transduction, «CURRENT DRUG TARGETS», 2007, 8, pp. 185 - 196 [articolo]

F. Benfatti; G. Cardillo; S.Fabbroni; P. Galzerano; L. Gentilucci; R. Juris; A. Tolomelli; M. Baiula; A. Spartà; S.Spampinato, Synthesis and Biological Evaluation of Nonpeptide alpha-v-beta-3/alpha-5-beta-1 Integrin Dual Antagonists containing 5,6-Dihydropyridin-2-one Scaffolds, «BIOORGANIC & MEDICINAL CHEMISTRY», 2007, 15, pp. 7380 - 7390 [articolo]

F. Benfatti; G. Cardillo; L. Gentilucci; A. Tolomelli, Synthesis and biological evaluation of unprecedented classes of spiro-beta-lactams and azido-beta-lactams as acyl-CoA:cholesterol acyltransferase inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2007, 17, pp. 1946 - 1950 [articolo]

F. Benfatti; G. Cardillo; L. Gentilucci; A. Tolomelli, Synthesis of four-membered ring spiro-beta -lactams by epoxide ring-opening., «EUROPEAN JOURNAL OF ORGANIC CHEMISTRY», 2007, 19, pp. 3199 - 3205 [articolo]

L. Gentilucci; A. Tolomelli; F. Squassabia, Topological exploration of cyclic endomorphin-1 analogues, structurally defined models for investigating the bioactive conformation of MOR agonists., «PROTEIN AND PEPTIDE LETTERS», 2007, 14, pp. 51 - 56 [articolo]

L. Gentilucci; G. Cardillo; A. Tolomelli; F. Squassabia; C. Tiozzo, A novel family of minimal PMRI cyclic peptides as versatile scaffolds for generating new molecular topology., «MEDICINAL CHEMISTRY», 2006, 2, pp. 395 - 400 [articolo]

L. Gentilucci; A. Tolomelli; F. Squassabia, Peptides and peptidomimetics in medicine, surgery, and biotecnology, «CURRENT MEDICINAL CHEMISTRY», 2006, 13, pp. 2449 - 2466 [articolo]

F.Benfatti; G.Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli; A. Catapano, Synthesis and Biological Evaluation of Azido- and Aziridino-hydroxyl-beta -lactams through Stereo- and Regioselective Epoxide Ring Opening., «JOURNAL OF ORGANIC CHEMISTRY», 2006, 71, pp. 9229 - 9232 [articolo]

F. Benfatti; G. Cardillo; S. Fabbroni; L. Gentilucci; R. Perciaccante; A. Tolomelli; M. Baiula; S.Spampinato, Synthesis of Enantiomerically Pure alpha-v-beta-3 Integrin ligands Based on a 5,6-Dihydropyridin-2-one Scaffold., «TETRAHEDRON-ASYMMETRY», 2006, 17, pp. 167 - 170 [articolo]

G.Cardillo; L. Gentilucci; A. Tolomelli, Unusual Amino Acids: Synthesis and Introduction into Naturally Occurring Peptides and Biologically Active Analogues, «MINI-REVIEWS IN MEDICINAL CHEMISTRY», 2006, 6, pp. 293 - 304 [articolo]

F. Benfatti; G. Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli, An investigation of the reactivity of MCPBA and alpha-bromoalkenes under traditional or microwave-assisted conditions: Selective formation of epoxides or allylic bromides., «SYNLETT», 2005, 14, pp. 2204 - 2208 [articolo]

L. Gentilucci; F. Squassabia; G. Cardillo; A. Tolomelli, Atypical mu-opioid agonists: reconsideration of the requisites for receptor activation, in: Book of Abstracts, RIMINI, s.n, 2005(atti di: 1st European Conference on Chemistry for Life Sciences, Rimini, 4-8 ottobre 2005) [atti di convegno-abstract]

F. Benfatti; G. Cardillo; L. Gentilucci; R. Perciaccante; A. Tolomelli, Functionalizations of the C3 side chain of densely substituted azetidin-2-ones, in: 20th ICHC Book of Abstracts, PALERMO, s.n, 2005(atti di: 20th International Congress of Heterocyclic Chemistry, Palermo, 31 luglio-5 agosto 2005) [atti di convegno-abstract]

G.Cardillo; S. Fabbroni; L. Gentilucci; R. Perciaccante; F. Piccinelli; A. Tolomelli, Highly Diastereoselective Allylic Azide Formation and Isomerization. Synthesis of 3(2'-Amino)-beta-lactams, «ORGANIC LETTERS», 2005, 7, pp. 533 - 536 [articolo]