Piazzi L.; Cavalli A.; Belluti F.; Bisi A.; Gobbi S.; Rizzo S.; Bartolini M.; Andrisano V.; Recanatini M.; Rampa A., Extensive SAR and computational studies of
3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives., «JOURNAL OF MEDICINAL CHEMISTRY», 2007, 50, pp. 4250 - 4254 [Scientific article]
Rampa A.; Belluti F.; Gobbi S.; Piazzi L.; Bartolini M.; Bisi A., Hybrid drugs for Alzheimer's disease: new indanone derivatives bearing a pharmacophoric fragment of AP2238, in: Frontiers in CNS and oncology medicinal chemistry, SIENA, s.n, 2007, pp. 49 - 50 (atti di: Frontiers in CNS and oncology medicinal chemistry, Siena, 7-9 ottobre 2007) [Abstract]
Gobbi S.; Cavalli A.; Negri M.; Schewe K.E.; Belluti F.; Piazzi L.; Hartmann R.W.; Recanatini M.; Bisi A., Imidazolylmethylbenzophenones as highly potent aromatase inhibitors., «JOURNAL OF MEDICINAL CHEMISTRY», 2007, 50, pp. 3420 - 3422 [Scientific article]
Gobbi S.; Bisi A.; Belluti F.; Piazzi L.; Rampa A.; Cavalli A.; Schede K.; Hartmann R.W., New potent inhibitors of cytochrome P450 aromatase, in: 16th Camerino-Noordwijkerhout Symposium-An overview of receptor chemistry, CAMERINO, s.n, 2007, pp. 113 - 113 (atti di: 16th Camerino-Noordwijkerhout Symposium, Camerino, 9-13 settembre 2007) [Abstract]
M. Bartolini; F. Belluti; M.L. Bolognesi; M. Rosini; V. Andrisano, In vitro methods for characterizing new multi-potent compounds for Alzheimer’s disease, in: 9th International Geneve/Springfield Symposium on advances in Alzheimer Therapy, Abstract Book, s.l, s.n, 2006, pp. 32 - 32 (atti di: 9th International Geneve/Springfield Symposium on advances in Alzheimer Therapy, Geneve Switzerland., April 19-22, 2006) [Abstract]
Gobbi S.; Cavalli A.; Rampa A.; Belluti F.; Piazzi L.; Paluszcak A.; Hartmann R.W.; Recanatini M.; Bisi A., Lead optimization providing a series of flavone derivatives as potent nonsteroidal inhibitors of the cytochrome P450 aromatase enzyme, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 4777 - 4780 [Scientific article]
Gobbi S.; Belluti F.; Bisi A.; Piazzi L.; Rampa A.; Zampiron A.; Barbera M.; Caputo A.; Carrara M., New derivatives of xanthenone-4-acetic acid: synthesis, pharmacological profile and effect on TNF-alpha and NO production by human immune cells, «BIOORGANIC & MEDICINAL CHEMISTRY», 2006, 14, pp. 4101 - 4109 [Scientific article]
Bisi A.; Gobbi S.; Rampa A.; Belluti F.; Piazzi L.; Valenti P.; Gyemant N.; Molnar J., New potent P-glycoprotein inhibitors carrying a polycyclic scaffold, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 3049 - 3051 [Scientific article]
S. Rizzo; A. Rampa; F. Belluti; L. Piazzi; S. Gobbi; A. Bisi, Progettazione e sintesi di derivati benzofuranici per la malattia di Alzheimer, in: Sigma-Aldrich young chemists Symposium
6° SAYCS, RICCIONE, s.n, 2006, pp. P81 - P81 (atti di: Sigma-Aldrich young chemists Symposium
6° SAYCS, Riccione, 9-11 ottobre 2006) [Abstract]
F. Belluti; A. Rampa; L. Piazzi; A. Bisi; S. Gobbi; M. Bartolini; A. Cavalli; P. Valenti, Benzophenone derivatives as Inhibitors of Acetylcholinesterase, in: 15th Noordwijkerhout Camerino Symposium-Trends in drug research, NOORDWIJKERHOUT, s.n, 2005(atti di: 15th Noordwijkerhout Camerino Symposium-Trends in drug research, Noordwijkerhout, 8-13 may) [Abstract]
Belluti, Federica; Rampa, Angela; Piazzi, Lorna; Bisi, Alessandra; Gobbi, Silvia; Bartolini, Manuela; Andrisano, Vincenza; Cavalli, Andrea; Recanatini, Maurizio; Valenti, Piero, Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation., «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48, pp. 4444 - 4456 [Scientific article]
Cavalli A.; Bisi A.; Bertucci C.; Rosini C.; Paluszcak A.; Gobbi S.; Giorgio E.; Rampa A.; Belluti F.; Piazzi L.; Valenti P.; Hartmann R.W.; Recanatini M., Enantioselective nonsteroidal aromatase inhibitors identified through a multidisciplinary medicinal chemistry approach, «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48 (23), pp. 7282 - 7289 [Scientific article]
A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani; P. A. Borea; M. Carrara, Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells, «IL FARMACO», 2005, 60, pp. 135 - 147 [Scientific article]
M. Carrara; A. Zampiron; M. Barbera; A. Caputo; S. Gobbi; F. Belluti; A. Bisi; L. Piazzi; A. Rampa; P. Valenti, In vitro studies of flavon-8-acetic acid analogues, in: 32° Congresso Nazionale della Società Italiana di Farmacologia, NAPOLI, s.n, 2005(atti di: 32° Congresso Nazionale della Società Italiana di Farmacologia, Napoli, 1-4 giugno) [Abstract]
M. Carrara; A. Zampiron; M. Barbera; A. Caputo; A. Bisi; S. Gobbi; F. Belluti; L. Piazzi; A. Rampa; P. Valenti, Mono- or di-fluorinated analogues of Flavone-8-acetic acid: synthesis and in vitro biological activity, «ANTICANCER RESEARCH», 2005, 25, pp. 1179 - 1186 [Scientific article]