Foto del docente

Andrea Bedini

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: BIO/14 Pharmacology

Publications

Alessandra Locatelli;Sandro Cosconati;Matteo Micucci;Alberto Leoni;Luciana Marinelli;Andrea Bedini;Pierfranco Ioan;Santi Mario Spampinato;Ettore Novellino;Alberto Chiarini;Roberta Budriesi, Ligand Based Approach to L-Type Calcium Channel by Imidazo[2,1-b]thiazole-1,4-Dihydropyridines: from Heart Activity to Brain Affinity, «JOURNAL OF MEDICINAL CHEMISTRY», 2013, 56, pp. 3866 - 3877 [Scientific article]

S. Spampinato; A. Bedini; M. Baiula, Prodynorphin-derived peptides, in: Handbok of Biologically Active Peptides, SAN DIEGO, Academic Press, 2013, pp. 1596 - 1601 [Chapter or essay]

C: Petrella; C. Giuli; M. Broccardo; H. Eutamene; C. Cartier; M. Leveque; A. Bedini; S. Spampinato; L. Bueno; V. Theodorou; G. Improta; S. Agostini, Protective and worsening peripheral nociceptin/orphanin FQ receptor-mediated effect in a rat model of experimental colitis, «PHARMACOLOGICAL RESEARCH», 2013, 70, pp. 72 - 79 [Scientific article]

R. De Marco; A. Tolomelli; S. Spampinato; A. Bedini; L. Gentilucci, Opioid Activity Profiles of Oversimplified Peptides Lacking in the Protonable N-Terminus, «JOURNAL OF MEDICINAL CHEMISTRY», 2012, 55, pp. 10292 - 10296 [Scientific article]

Baiula M; Carbonari G; Dattoli SD; Calienni M; Bedini A; Spampinato S., REST is up-regulated by epidermal growth factor in HeLa cells and inhibits apoptosis by influencing histone H3 acetylation, «BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH», 2012, 1823, pp. 1252 - 1263 [Scientific article]

Baiula M; Bedini A; Carbonari G; Dattoli SD; Spampinato S, Therapeutic Targeting of Eosinophil Adhesion and Accumulation in Allergic Conjunctivitis, «FRONTIERS IN PHARMACOLOGY», 2012, 3/203, pp. 1 - 6 [Scientific article]

L. Gentilucci; R. de Marco; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali, A novel family of minimalist opioid peptides deprived of the classic pharmacophores, «PHARMACOLOGICAL REPORTS», 2011, 63, pp. 212 - 212 [Abstract]

R.De Marco; L. Gentilucci; A. Tolomelli; S. Feddersen; S. Spampinato; A. Bedini; R. Artali., DESIGN AND SYNTHESIS OF OPIOID PEPTIDE ANALOGUES AND MIMETICS, «PHARMACOLOGICAL REPORTS», 2011, 63, pp. 226 - 226 [Abstract]

Baiula M; Spartà A; Bedini A; Carbonari G; Bucolo C; Ward KW; Zhang JZ; Govoni P; Spampinato S, Eosinophil as a cellular target of the ocular anti-allergic action of mapracorat, a novel selective glucocorticoid receptor agonist, «MOLECULAR VISION», 2011, 17, pp. 3208 - 3223 [Scientific article]

Bedini A; Vincelli G; Spampinato S, mu-opioid receptor (MOR) expression and opioid-mediated intracellular signalling are altered in glial cells exposed to TNF-alpha, «PHARMACOLOGICAL REPORTS», 2011, 63, pp. 223 - 223 [Abstract]

Gentilucci L; Tolomelli A; De Marco R; Spampinato S; Bedini A; Artali R., The Inverse Type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists., «CHEMMEDCHEM», 2011, 6(9), pp. 1640 - 1653 [Scientific article]

L. Gentilucci; R. De Marco; A. Tolomelli; S. Spampinato; A. Bedini; R. Artali, Ac-D-Trp-PheNH2 AND Ac-D-Trp-Phe-GlyNH2 - A NEW CLASS OF UNUSUAL OPIOID PEPTIDES, in: INRC 2010 - Abstracts Book, INRC, 2010, pp. 79 - 79 (atti di: International Narcotics Research Conference 2010, Malmoe, Sweden, 11-16 luglio 2010) [Abstract]

L. Gentilucci; G. Cardillo; S. Spampinato; A. Tolomelli; F. Squassabia; R. De Marco; A. Bedini; M. Baiula; L. Belvisi; M. Civera, Antiangiogenic Effect of Dual/Selective α5β1/αvβ3 Integrin Antagonists Designed on Partially Modified Retro-Inverso Cyclotetrapeptide Mimetics, «JOURNAL OF MEDICINAL CHEMISTRY», 2010, 53, pp. 106 - 118 [Scientific article]

B. Luppi; F. Bigucci; A. Abruzzo; G. Corace; T. Cerchiara; A. Bedini; S. Spampinato; V. Zecchi, Chitosan-based Polyelectrolyte Complexes for Nasal Drug Delivery, «CRS NEWSLETTER», 2010, 27(6), pp. 15 - 16 [Scientific article]

L. Gentilucci; A.Tolomelli; S. Spampinato; A. Bedini; R. De Marco; R. Artali, DETERMINATION OF THE BIOLOGICALLY ACTIVE STRUCTURE OF THE ATYPICAL MOR-LIGAND c[D-Asp-1-amide-beta-Ala-D-Trp-Phe] AND ANALOGUES BY NMR AND MOLECULAR DOCKING, in: , «BOLETÍN DE LA SOCIEDAD QUÍMICA DE MÉXICO», 2010, 4 n.e., pp. 96 - 96 (atti di: 45° Congreso Mexicano de Quimica, Riviera Maya, Quntana Roo, 18-22 settembre 2010) [Abstract]