Piazzi L.; Cavalli A.; Belluti F.; Bisi A.; Gobbi S.; Rizzo S.; Bartolini M.; Andrisano V.; Recanatini M.; Rampa A., Extensive SAR and computational studies of
3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives., «JOURNAL OF MEDICINAL CHEMISTRY», 2007, 50, pp. 4250 - 4254 [articolo]
Gobbi S.; Cavalli A.; Negri M.; Schewe K.E.; Belluti F.; Piazzi L.; Hartmann R.W.; Recanatini M.; Bisi A., Imidazolylmethylbenzophenones as highly potent aromatase inhibitors., «JOURNAL OF MEDICINAL CHEMISTRY», 2007, 50, pp. 3420 - 3422 [articolo]
Gobbi S.; Cavalli A.; Rampa A.; Belluti F.; Piazzi L.; Paluszcak A.; Hartmann R.W.; Recanatini M.; Bisi A., Lead optimization providing a series of flavone derivatives as potent nonsteroidal inhibitors of the cytochrome P450 aromatase enzyme, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 4777 - 4780 [articolo]
Gobbi S.; Belluti F.; Bisi A.; Piazzi L.; Rampa A.; Zampiron A.; Barbera M.; Caputo A.; Carrara M., New derivatives of xanthenone-4-acetic acid: synthesis, pharmacological profile and effect on TNF-alpha and NO production by human immune cells, «BIOORGANIC & MEDICINAL CHEMISTRY», 2006, 14, pp. 4101 - 4109 [articolo]
Bisi A.; Gobbi S.; Rampa A.; Belluti F.; Piazzi L.; Valenti P.; Gyemant N.; Molnar J., New potent P-glycoprotein inhibitors carrying a polycyclic scaffold, «JOURNAL OF MEDICINAL CHEMISTRY», 2006, 49, pp. 3049 - 3051 [articolo]
Belluti, Federica; Rampa, Angela; Piazzi, Lorna; Bisi, Alessandra; Gobbi, Silvia; Bartolini, Manuela; Andrisano, Vincenza; Cavalli, Andrea; Recanatini, Maurizio; Valenti, Piero, Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation., «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48, pp. 4444 - 4456 [articolo]
Cavalli A.; Bisi A.; Bertucci C.; Rosini C.; Paluszcak A.; Gobbi S.; Giorgio E.; Rampa A.; Belluti F.; Piazzi L.; Valenti P.; Hartmann R.W.; Recanatini M., Enantioselective nonsteroidal aromatase inhibitors identified through a multidisciplinary medicinal chemistry approach, «JOURNAL OF MEDICINAL CHEMISTRY», 2005, 48 (23), pp. 7282 - 7289 [articolo]
A. Rampa; A. Bisi; F. Belluti; S. Gobbi; L. Piazzi; P. Valenti; A. Zampiron; A. Caputo; K. Varani; P. A. Borea; M. Carrara, Homopterocarpanes as bridged triarylethylene analogues: synthesis and antagonistic effects in human MCF-7 breast cancer cells, «IL FARMACO», 2005, 60, pp. 135 - 147 [articolo]
M. Carrara; A. Zampiron; M. Barbera; A. Caputo; A. Bisi; S. Gobbi; F. Belluti; L. Piazzi; A. Rampa; P. Valenti, Mono- or di-fluorinated analogues of Flavone-8-acetic acid: synthesis and in vitro biological activity, «ANTICANCER RESEARCH», 2005, 25, pp. 1179 - 1186 [articolo]
R. Budriesi; A. Bisi; P. Ioan; A. Rampa; S. Gobbi; F. Belluti; L. Piazzi; P. Valenti; A. Chiarini, 1,4-dihydropyridine derivatives as calcium channel modulators: the role of 3-methoxy-flavone moiety, «BIOORGANIC & MEDICINAL CHEMISTRY», 2005, 13, pp. 3423 - 3430 [articolo]
Bisi A.; Rampa A.; Budriesi R.; Gobbi S.; Belluti F.; Ioan P.; Valoti E.; Chiarini A.; Valenti P., Cardiovascular hybrid drugs: New benzazepinone derivatives as bradycardic agents endowed with selective β1-Non-competitive antagonism, «BIOORGANIC & MEDICINAL CHEMISTRY», 2003, 11, pp. 1353 - 1361 [articolo]
Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Piazzi L.; Valenti P.; Caputo A.; Zampiron A.; Carrara M., Synthesis and biological evaluation of 3-alkoxy analogues of flavone-8-acetic acid, «JOURNAL OF MEDICINAL CHEMISTRY», 2003, 46, pp. 3662 - 3669 [articolo]
Piazzi L.; Rampa A.; Bisi A.; Gobbi S.; Belluti F.; Cavalli A.; Bartolini M.; Andrisano V.; Valenti P.; Recanatini M., 3-(4-{[benzyl(methyl)amino]methyl}-phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced β-amyloid aggregation: A dual function lead for Alzheimer's disease therapy, «JOURNAL OF MEDICINAL CHEMISTRY», 2003, 46, pp. 2279 - 2282 [articolo]
Gobbi S.; Rampa A.; Bisi A.; Belluti F.; Valenti P.; Caputo A.; Zampiron A.; Carrara M., Synthesis and antitumor activity of new derivatives of xanthen-9-one-4-acetic acid, «JOURNAL OF MEDICINAL CHEMISTRY», 2002, 45, pp. 4931 - 4939 [articolo]
Recanatini M.; Hartmann R.W.; Bisi A.; Cavalli A.; Belluti F.; Gobbi S.; Rampa A.; Valenti P.; Palzer M.; Palusczak A., A new class of nonsteroidal aromatase inhibitors: Design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17α-hydroxylase/C17,20-lyase, «JOURNAL OF MEDICINAL CHEMISTRY», 2001, 44, pp. 672 - 680 [articolo]
