Foto del docente

Vincenzo Tumiatti

Full Professor

Department for Life Quality Studies

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Director of Single Cycle Degree in Pharmacy

Publications

De Simone, Angela; Fiori, Jessica; Naldi, Marina; D'Urzo, Annalisa; Tumiatti, Vincenzo; Milelli, Andrea; Andrisano, Vincenza, Application of an ESI-QTOF method for the detailed characterization of GSK-3β inhibitors, «JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS», 2017, 144, pp. 159 - 166 [Scientific article]

Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini, Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna, Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 128, pp. 107 - 122 [Scientific article]

Milelli, Andrea; De Simone, Angela; Ticchi, Nicole; Chen, Huan Huan; Betari, Nibal; Andrisano, Vincenza; Tumiatti, Vincenzo, Tacrine-based Multifunctional Agents in Alzheimer's Disease: an Old Story in Continuous Development, «CURRENT MEDICINAL CHEMISTRY», 2017, 24, pp. 3522 - 3546 [Scientific article]

Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A., Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 117, pp. 283 - 291 [Scientific article]

Marchetti, C.; Minarini, A.; Tumiatti, V.; Moraca, F.; Parrotta, L.; Alcaro, S.; Rigo, R.; Sissi, C.; Gunaratnam, M.; Ohnmacht, S.A.; Neidle, S.; Milelli, A., Macrocyclic naphthalene diimides as G-quadruplex binders, «BIOORGANIC & MEDICINAL CHEMISTRY», 2015, 23, pp. 3819 - 3830 [Scientific article]Open Access

Aloisi, I.; Cai, G.; Tumiatti, V.; Minarini, A.; Del Duca, S., Natural polyamines and synthetic analogs modify the growth and the morphology of Pyrus communis pollen tubes affecting ROS levels and causing cell death, «PLANT SCIENCE», 2015, 239, pp. 92 - 105 [Scientific article]Open Access

Amelia Parise; Andrea Milelli; Vincenzo Tumiatti; Anna Minarini; Paolo Neviani; Guendalina Zuccari, Preparation, characterization and in vitro evaluation of sterically stabilized liposome containing a naphthalenediimide derivative as anticancer agent, «DRUG DELIVERY», 2015, 22, pp. 590 - 597 [Scientific article]Open Access

De Gianni, E.; Turrini, E.; Milelli, A.; Maffei, F.; Carini, M.; Minarini, A.; Tumiatti, V.; Da Ros, T.; Prato, M.; Fimognari, C., Study of the cytotoxic effects of the new synthetic isothiocyanate CM9 and its fullerene derivative on human T-leukemia cells, «TOXINS», 2015, 7, pp. 535 - 552 [Scientific article]Open Access

Zuccari, G.; Milelli, A.; Pastorino, F.; Loi, M.; Petretto, A.; Parise, A.; Marchetti, C.; Minarini, A.; Cilli, M.; Emionite, L.; Di Paolo, D.; Brignole, C.; Piaggio, F.; Perri, P.; Tumiatti, V.; Pistoia, V.; Pagnan, G.; Ponzoni, M., Tumor vascular targeted liposomal-bortezomib minimizes side effects and increases therapeutic activity in human neuroblastoma, «JOURNAL OF CONTROLLED RELEASE», 2015, 211, pp. 44 - 52 [Scientific article]

Anna Minarini; Andrea Milelli; Carmela Fimognari; Elena Simoni; Eleonora Turrini; Vincenzo Tumiatti, Exploring the effects of isothiocyanates on chemotherapeutic drugs, «EXPERT OPINION ON DRUG METABOLISM & TOXICOLOGY», 2014, 10, pp. 25 - 38 [Scientific article]

Milelli A;Fimognari C;Ticchi N;Neviani P;Minarini A;Tumiatti V, Isothiocyanate synthetic analogs: biological activities, structure-activity relationships and synthetic strategies., «MINI-REVIEWS IN MEDICINAL CHEMISTRY», 2014, 14, pp. 963 - 977 [Scientific article]

Welsh, Silje; Li, Huanzhao; Marchetti, Chiara; Tumiatti, Vincenzo; Minarini, Anna; Wallace, Heather, Preliminary evaluation of the cytotoxicity of naphthalene diimide-polyamine conjugates in human cancer cells, in: 50th Congress of the European-Societies-of-Toxicology, ELSEVIER IRELAND LTD, «TOXICOLOGY LETTERS», 2014, 229, pp. S158 - S158 (atti di: 50th Congress of the European-Societies-of-Toxicology, Edinburgh, SCOTLAND, 7 ottobre 2014) [Abstract]

Minarini A.; Milelli A.; Tumiatti V.; Rosini M.; Lenzi M.; Ferruzzi L.; Turrini E.; Hrelia P.; Sestili P.; Calcabrini C.; Fimognari C., Exploiting RNA as a new biomolecular target for synthetic polyamines, «GENE», 2013, 524, pp. 232 - 240 [Scientific article]

Ryotaro Saiki; Yuki Yoshizawa; Anna Minarini; Andrea Milelli; Chiara Marchetti; Vincenzo Tumiatti; Toshihiko Toida; Keiko Kashiwagi; Kazuei Igarashi, In vitro and in vivo evaluation of polymethylene tetraamine derivatives as NMDA receptor channel blockers, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2013, 23, pp. 3901 - 3904 [Scientific article]

Anna Minarini; Andrea Milelli; Elena Simoni; Michela Rosini; Maria Laura Bolognesi; Chiara Marchetti; Vincenzo Tumiatti, Multifunctional Tacrine Derivatives in Alzheimer’s Disease, «CURRENT TOPICS IN MEDICINAL CHEMISTRY», 2013, 13, pp. 1771 - 1786 [Scientific article]