Foto del docente

Roberta Budriesi

Associate Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/10 Food Chemistry

Publications

Fumagalli L.; Pallavicini M.; Budriesi R.; Bolchi C.; Chiarini A.; Chiodini G.; Gobbi M.; Laurino P.; Micucci M.; Straniero V.; Valoti E., 6-Methoxy7-benzofuranoxy and 6-methoxy-7-indolyloxy analogues of WB4101: discovery of a potent and selective a1D-adrenoceptor antagonist., «JOURNAL OF MEDICINAL CHEMISTRY», 2013, 56, pp. 6402 - 6412 [Scientific article]

Pierfranco Ioan; Alessia Ciogli; Francesco Sirci; Roberta Budriesi; Barbara Cosimelli; Marco Pierini; Elda Severi; Alberto Chiarini; Gabriele Cruciani; Francesco Gasparrini; Domenico Spinelli; Emanuele Carosati, Absolute configuration and biological profile of two thiazinooxadiazol-3-ones with L-type calcium channel activity: a study of the structural effects, «ORGANIC & BIOMOLECULAR CHEMISTRY», 2012, 10, pp. 8994 - 9003 [Scientific article]

Fumagalli L; Pallavicini M; Budriesi R; Gobbi M; Straniero V; Zagami M; Chiodini G; Bolchi C; Chiarini A; Micucci M; Valoti E, Affinity and activity profiling of unichiral 8-substituted 1,4-benzodioxane analogues of WB4101 reveals a potent and selective α1B-adrenoceptor antagonist., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2012, 58, pp. 184 - 191 [Scientific article]

Micucci M; Ioan P; Arroo R; Ruparelia K; Chiarini A; Budriesi R, Castanea sativa mill. Extract: a Co Adjuvant in the Treatment of Colestasis., in: abstracts book, s.l., s.n., 2012, pp. 144 - 144 (atti di: Nuove Prospettive in Chimica Farmaceutica. VI Meeting, Riccione (RN), 15-17 Aprile) [Abstract]

Aldini R; Budriesi R; Roda G; Micucci M; Ioan P; D’Errico-Grigioni A; Sartini A; Guidetti E; Marocchi M; Cevenini M; Rosini F; Montagnani M; Chiarini A; Mazzella G, Curcuma longa Extract Exerts a Myorelaxant Effect on the Ileum and Colon in a Mouse Experimental Colitis Model, Independent of the Anti-Inflammatory Effect, «PLOS ONE», 2012, 7, Article number: e44650 , pp. 1 - 12 [Scientific article]Open Access

Micucci M; Budriesi R; Ioan P; Chiarini A; Giorgini S, Effects of natural extract of chestnut wood in guinea pig ileum and proximal colon., in: Proceedings of first international conference on food digestion, s.l., s.n., 2012, pp. 118 - 118 (atti di: 1st international conference on food digestion, Cesena (FC), March, 19-21) [Abstract]

Micucci M; Aldini R; Mazzella G; Roda G; Chiarini A; Budriesi R, Nutraceuticals and Functional Foods: effects of turmeric towards intestinal motility in acute and chronic Dextrane Sodium Sulphate (DSS) induced colitis in mice., in: Atti, 2012(atti di: ChimALSi 2012-IX Congresso Italiano di Chimica degli Alimenti,, Ischia (Na), 04-07 Giugno 2012) [Poster]

Catalano A; Desaphy J-F; Lentini G; Carocci A; Di Mola A; Bruno C; Carbonara R; De Palma A; Budriesi R; Ghelardini C; Perrone MG; Colabufo NA; Conte Camerino D; Franchini C, Synthesis and Toxicopharmacological Evaluation of meta-Hydroxymexiletine, the First Metabolite of Mexiletine more Potent than the Parent Compound on Voltage-gated Sodium Channels., «JOURNAL OF MEDICINAL CHEMISTRY», 2012, 55, pp. 1418 - 1422 [Scientific article]

Budriesi R, 1,4-DHP scaffold: calcium channel ligand based approach from cardiovascular to neuroprotective activity., in: Book of Abstract, s.l., s.n., 2012, pp. 30 - 30 (atti di: 21st National Meeting on Medicinal Chemistry., Palermo, July 17–20) [Abstract]

E Carosati; P Ioan; M Micucci; F Broccatelli; G Cruciani; BS Zhorov; A Chiarini; R Budriesi, 1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story So Far And Perspectives (Part 2): Action in Other Targets and Antitargets, «CURRENT MEDICINAL CHEMISTRY», 2012, 19, pp. 4306 - 4323 [Scientific article]

R. Budriesi; P. Ioan; A. Leoni; N. Pedemonte; A. Locatelli; M. Micucci; A. Chiarini; L. J. Galietta., Cystic Fibrosis: a New Target for 4-Imidazo[2,1-b]thiazole-1,4- Dihydropyridines., «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 3094 - 3885 [Scientific article]

budriesi, Dalla nutraceutica alla chimica farmaceutica: piante e salute, in: gastrocervia, 2011, pp. 1 - 1 (atti di: gastrocervia, cervia-milano marittima, 17-18 settebre 2011) [Contribution to conference proceedings]

Budriesi R.; Micucci M.; Ioan P.; Malaguti M.; Hrelia S.; Chiarini A., I tannini della Castanea Sativa Mill: caratterizzazione dell'attività cardiovascolare e cardioprotettiva., in: Atti del XVIII Congresso Nazionale della Società Italiana di Ricerche Cardiovascolari, s.l., (sine nomine), 2011, pp. 37 - 37 (atti di: XVIII Congresso Nazionale della Società Italiana di Ricerche Cardiovascolari, Imola (BO), 21-22 ottobre 2011) [Abstract]

M. Viale; C. Cordazzo; D. de Totero; R. Budriesi; C. Rosano; A. Leoni; P. Ioan; C. Aiello; M. Croce; A. Andreani; M. Rambaldi; P. Russo; A. Chiarini; D. Spinelli, Inhibition of MDR1 activity and induction of apoptosis by analogues of nifedipine and diltiazem: an in vitro analysis, «INVESTIGATIONAL NEW DRUGS», 2011, 29, pp. 98 - 109 [Scientific article]

Cosimelli B; Severi E; Novellino E; Cavaccini A; Cataldi M; Budriesi R; Micucci M; Chiarini A; Ioan P, Preliminary Finding on a New Calcium Channel Entry Blocker Chemotype: 5,6-Diamino-4-hydroxy-2-mercaptopyrimidine Derivatives., «JOURNAL OF MEDICINAL CHEMISTRY», 2011, 54, pp. 5597 - 5601 [Scientific article]

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