Foto del docente

Michela Rosini

Professoressa associata

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

Singhal M.; Merino V.; Rosini M.; Cavalli A.; Kalia Y.N., Controlled Iontophoretic Delivery in Vitro and in Vivo of ARN14140 - A Multitarget Compound for Alzheimer's Disease, «MOLECULAR PHARMACEUTICS», 2019, 16, pp. 3460 - 3468 [articolo]

Di Paolo, Maria Luisa; Cervelli, Manuela; Mariottini, Paolo; Leonetti, Alessia; Polticelli, Fabio; Rosini, Michela; Milelli, Andrea; Basagni, Filippo; Venerando, Rina; Agostinelli, Enzo; Minarini, Anna, Exploring the activity of polyamine analogues on polyamine and spermine oxidase: methoctramine, a potent and selective inhibitor of polyamine oxidase, «JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY», 2019, 34, pp. 740 - 752 [articolo]Open Access

Basagni F.; Lanni C.; Minarini A.; Rosini M., Lights and shadows of electrophile signaling: Focus on the Nrf2-Keap1 pathway, «FUTURE MEDICINAL CHEMISTRY», 2019, 11, pp. 707 - 721 [articolo]

Rosini M.; Simoni E.; Caporaso R.; Basagni F.; Catanzaro M.; Abu I.F.; Fagiani F.; Fusco F.; Masuzzo S.; Albani D.; Lanni C.; Mellor I.R.; Minarini A., Merging memantine and ferulic acid to probe connections between NMDA receptors, oxidative stress and amyloid-β peptide in Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 180, pp. 111 - 120 [articolo]Open Access

Catanzaro, Michele; Corsini, Emanuela*; Rosini, Michela; Racchi, Marco; Lanni, Cristina, Immunomodulators inspired by nature: A review on curcumin and Echinacea, «MOLECULES», 2018, 23, Article number: 2778, pp. 1 - 17 [articolo]Open Access

Maria Luisa Di Paolo, Giorgio Cozza, Andrea Milelli, Francesca Zonta, Stefania Sarno, Elirosa Minniti, Michela Rosini, Anna Minarini, Novel targets for “old” polyamine analogues: monoamine oxidases and benextramine derivatives, in: 5th International Conference on Polyamines: Biochemical, Physiological and Clinical Perspectives, 2018, pp. 115 - 115 (atti di: 5th International Conference on Polyamines: Biochemical, Physiological and Clinical Perspectives, Howard Civil Service International House, National Taiwan Ocean University Taipei (Taiwan), September 2nd - 7th, 2018) [atti di convegno-poster]

Serafini, Melania Maria; Catanzaro, Michele; Rosini, Michela; Racchi, Marco; Lanni, Cristina, Curcumin in Alzheimer's disease: Can we think to new strategies and perspectives for this molecule?, «PHARMACOLOGICAL RESEARCH», 2017, 124, pp. 146 - 155 [articolo]

Simoni, Elena; Bartolini, Manuela; Abu, Izuddin F; Blockley, Alix; Gotti, Cecilia; Bottegoni, Giovanni; Caporaso, Roberta; Bergamini, Christian; Andrisano, Vincenza; Cavalli, Andrea; Mellor, Ian R; Minarini, Anna; Rosini, Michela, Multitarget drug design strategy in Alzheimer's disease: focus on cholinergic transmission and amyloid-beta aggregation, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 953 - 963 [articolo]

AMADIO M, Serafini M M, Marchesi N, Catanzaro M, Fagiani F, Simoni E, Pascale A, Rosini M, Lanni C, Nature-inspired Nrf2 activators in retinal pigment epithelial cells: a source for therapeutics in age-related macular degeneration, in: Science for sight: EVER 2017 Abstract book, 2017, pp. 190 - 190 (atti di: XXth EVER Congress 2017, Nizza (Francia), 27-30 settembre 2017) [atti di convegno-abstract]

Minniti, Elirosa; Byl, Jo Ann W.; Riccardi, Laura; Sissi, Claudia; Rosini, Michela; De Vivo, Marco; Minarini, Anna; Osheroff, Neil, Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2017, 27, pp. 4687 - 4693 [articolo]

Maestri, Valentina; Tarozzi, Andrea; Simoni, Elena; Cilia, Antonio; Poggesi, Elena; Naldi, Marina; Nicolini, Benedetta; Pruccoli, Letizia; Rosini, Michela; Minarini, Anna, Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 136, pp. 259 - 269 [articolo]

Simoni, Elena; Serafini, Melania M; Caporaso, Roberta; Marchetti, Chiara; Racchi, Marco; Minarini, Anna; Bartolini, Manuela; Lanni, Cristina; Rosini, Michela, Targeting the Nrf2/Amyloid-Beta Liaison in Alzheimer's Disease: A Rational Approach, «ACS CHEMICAL NEUROSCIENCE», 2017, 8, pp. 1618 - 1627 [articolo]

Reggiani, Angelo M.; Simoni, Elena; Caporaso, Roberta; Meunier, Johann; Keller, Emeline; Maurice, Tangui; Minarini, Anna; Rosini, Michela; Cavalli, Andrea, In vivo characterization of ARN14140, a memantine/galantamine-based multi-target compound for Alzheimer's disease, «SCIENTIFIC REPORTS», 2016, 6, Article number: 33172, pp. 1 - 11 [articolo]Open Access

Rosini, M; Simoni, E; Caporaso, R; Minarini, A, Multitarget strategies in Alzheimer's disease: benefits and challenges on the road to therapeutics, «FUTURE MEDICINAL CHEMISTRY», 2016, 8, pp. 697 - 711 [articolo]

Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela, Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease, «CHEMMEDCHEM», 2016, 11, pp. 1309 - 1317 [articolo]Open Access